Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T86591 | Target Info | |||
| Target Name | Peroxisome proliferator-activated receptor alpha (PPARA) | ||||
| Synonyms |
Peroxisome proliferater-activated receptor alpha; PPARalpha; PPAR-alpha; PPAR; Nuclear receptor subfamily 1 group C member 1; NR1C1
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| Target Type | Successful Target | ||||
| Gene Name | PPARA | ||||
| Biochemical Class | Nuclear hormone receptor | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 129 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Clofibrate
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|
Approved | Compound Info | ||
| Synonyms |
Amotril; Angiokapsul; Anparton; Antilipid; Antilipide; Apolan; Arterioflexin; Arterosol; Artevil; Ateculon; Ateriosan; Athebrate; Atheromide; Atheropront; Athromidin; Atrolen; Atromid; Atromida; Atromidin; Atrovis; Azionyl; Bioscleran; Bresit; CPIB; Cartagyl; Chlorfenisate; Chlorphenisate; Cinnarizin; Citiflus; Claripex; Cloberat; Clobrat; Clofar; Clofibate; Clofibram; Clofibrat; Clofibrato; Clofibratum; Clofinit; Clofipront; Delipid; Deliva; ELPI; EPIB; Fibralem; Gerastop; Hyclorate; Klofibrat; Klofiran; Levatrom; Lipamid; Lipavil; Lipavlon; Lipidsenker; Lipofacton; Lipomid; Liponorm; Liporeduct; Liporil; Liposid; Liprin; Liprinal; Lobetrin; Miscleron; Misclerone; Miskleron; Negalip; Normalip; Normat; Normet; Normolipol; Novofibrate; Persantinat; Recolip; Regardin; Regelan; Robigram; Scrobin; Serofinex; Serotinex; Skerolip; Sklerepmexe; Sklero; Sklerolip; Skleromex; Skleromexe; Ticlobran; Xyduril; Yoclo; Amotril S; Atromid S; Claripex CPIB; Clofibrato [Spanish]; Dura clofibrat; Ethyl chlorophenoxyisobutyrate; Ethyl clofibrate; Regelan N; Vincamin compositum; AY 61123; C 6643; Lipide 500; Oxan 600; AY-61123; Athranid-wirkstoff; Atromid-S; BML2-F02; Chlorophenoxyisobutyrate, Ethyl; Clobren-5F; Clobren-SF; Clofibrate (CLOF); Clofibrato [INN-Spanish]; Clofibratum [INN-Latin]; Clofibric Acid, Ethyl Ester; Ethyl p-chlorophenoxyisobutyrate; Ethyl para-chlorophenoxyisobutyrate; Neo-Atomid; Neo-Atromid; Sklero-Tablinen; Sklero-tablinene; Sklero-tabuls; ATROMID-S (TN); Atromid-S (TN); Atromid-S, Clofibrate; Ethyl alpha-p-chlorophenoxyisobutyrate; Clofibrate (JP15/USP/INN); Clofibrate [USAN:INN:BAN:JAN]; Ethyl 2-(4-chlorophenoxy)isobutyrate; Ethyl 2-(p-chlorophenoxy)isobutyrate; Ethyl alpha-(4-chlorophenoxy)isobutyrate; Ethyl alpha-(p-chlorophenoxy)isobutyrate; Ethyl-alpha-p-chlorophenoxy-isobutyrate
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| Activity |
EC50 = 55000 nM
|
[1] | |||
| Compound Name |
Gemfibrozil
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Approved | Compound Info | ||
| Synonyms |
ApoGemfibrozil; Ausgem; Bolutol; Brozil; Cholespid; Clearol; Decrelip; Elmogan; Fetinor; Fibratol; Fibrocit; GFZ; Gemd; Gemfibril; Gemfibromax; Gemfibrosil; Gemfibrozilo; Gemfibrozilum; Gemhexal; Gemlipid; Gemnpid; GenGemfibrozil; Genlip; Gozid; Hidil; Hipolixan; Innogem; Innogen; Ipolipid; Jezil; Lanaterom; Lifibron; Lipazil; Lipigem; Lipira; Lipizyl; Lipozid; Lipur; Litarek; Lopid; Micolip; Normolip; NuGemfibrozil; Pilder; Polyxit; Progemzal; Reducel; Regulip; Renabrazin; Sinelip; Synbrozil; Taborcil; Tentroc; Trialmin; Alphapharm Brand of Gemfibrozil; Apo Gemfibrozil; Apotex Brand of Gemfibrozil; Bayvit Brand of Gemfibrozil; Bexal Brand of Gemfibrozil; Biochemie Brand of Gemfibrozil; Bull Brand of Gemfibrozil; Cantabria Brand of Gemfibrozil; Chem mart Brand of Gemfibrozil; Chem mart Gemfibrozil; DBL Gemfibrozil; Douglas Brand of Gemfibrozil; Farmasierra Brand of Gemfibrozil; Faulding Brand of Gemfibrozil;Ferrer Brand of Gemfibrozil; Gemfibrozilo Bayvit; Gemfibrozilo Bexal; Gemfibrozilo Ur; Gen Gemfibrozil; GenRX Gemfibrozil; Genpharm Brand of Gemfibrozil; Gevilon Uno; Healthsense Brand of Gemfibrozil; Healthsense Gemfibrozil; Hexal Brand of Gemfibrozil; Ipsen Brand of Gemfibrozil; Lipox Gemfi; Lopid R; Menarini Brand of Gemfibrozil; Novo Gemfibrozil; Novopharm Brand of Gemfibrozil; Nu Gemfibrozil; Nu Pharm Brand of Gemfibrozil; PMS Gemfibrozil; Parke Davis Brand of Gemfibrozil; Pfizer Brand of Gemfibrozil; Pharmascience Brand of Gemfibrozil; Quimifar Brand of Gemfibrozil; SBPA Gemfibrozil; Sigma Brand of Gemfibrozil; TAD Brand of Gemfibrozil; Terry White Chemists Brand of Gemfibrozil; Terry White Chemists Gemfibrozil; United Drug Brand of Gemfibrozil; Warner Lambert Brand of Gemfibrozil; CI719; Gemfi 1A Pharma; Apo-Gemfibrozil; Bayvit, Gemfibrozilo; Gem-S; Gemfibrozil, GenRX; Gemfibrozil, Healthsense; Gemfibrozil, SBPA; Gemfibrozilo [INN-Spanish]; Gemfibrozilum [INN-Latin]; Gen-Fibro;Gen-Gemfibrozil; Jezil (TN); Lopid (TN); Low-Lip; Novo-Gemfibrozil; Nu-Gemfibrozil; Nu-Pharm Brand of Gemfibrozil; PMS-Gemfibrozil; TEVA-A; WL-Gemfibrozil; Warner-Lambert Brand of Gemfibrozil; GEMFIBROZIL (SEE ALSO PEROXISOME PROJECT (GEMFIBROZIL)); Gemfibrozil [USAN:BAN:INN]; Gen-Fibro (TN); PEROXISOME PROJECT (GEMFIBROZIL) (SEE ALSO GEMFIBROZIL); Gemfibrozil (JAN/USP/INN); Gemcor, Lopid, Jezil,Gen-Fibro, Gemfibrozil; 1A Brand of Gemfibrozil; 2,2-Dimethyl-5-(2,5-dimethylphenoxy)pentanoic acid; 2,2-Dimethyl-5-(2,5-dimethylphenoxy)valeriansaeure; 2,2-Dimethyl-5-(2,5-xylyloxy)valeriansaeure; 2,2-Dimethyl-5-(2,5-xylyloxy)valeric acid; 5-(2,5-Dimethyl-Phenoxy)-2,2-Dimethyl-Pentanoic Acid; 5-(2,5-Dimethylphenoxy)-2,2-dimethylpentanoic acid; 5-[(2,5-dimethylphenyl)oxy]-2,2-dimethylpentanoic acid
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| Activity |
EC50 = 59000 nM
|
[2] | |||
| Compound Name |
FENOFIBRIC ACID
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Approved | Compound Info | ||
| Synonyms |
Fenofibric acid; 42017-89-0; Procetofenic acid; 2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropanoic acid; alpha 1081; NSC 281318; LF 178 acid; UNII-BGF9MN2HU1; 2-[4-(4-chlorobenzoyl)phenoxy]-2-methylpropanoic acid; LF 153; FNF Acid; C17H15ClO4; Trilipix; CCRIS 7302; EINECS 255-626-9; BGF9MN2HU1; CHEMBL981; BRN 2058973; CHEBI:83469; 2-[4-(4-Chlorobenzoyl)phenoxy]-2-methylpropionic Acid; Propanoic acid, 2-(4-(4-chlorobenzoyl)phenoxy)-2-methyl-; AK117112; 2-{4-[(4-chlorophenyl)carbonyl]phenoxy}-2-methylpropanoic acid; W-106287
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| Activity |
IC50 = 68000 nM
|
[3] | |||
| Compound Name |
GW1929
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Investigative | Compound Info | ||
| Synonyms |
GW 1929; GW-1929
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| Activity |
EC50 = 55300 nM
|
[4] | |||
| Compound Name |
(R)-2-(3-(3-(4-Methoxybenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)phenoxy)butanoic acid
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Investigative | Compound Info | ||
| Synonyms |
MK-0533; CHEMBL490029; UNII-J17152066B; MK0533; J17152066B; SCHEMBL671319; BDBM50267991; ZINC49878561; DB15242
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| Activity |
IC50 ~ 50000 nM
|
[5] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-3-(3-hydroxy-phenoxy)-1H-indole-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL426294; BDBM50173342
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| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
3-(5,7-Dipropyl-3-trifluoromethyl-benzo[d]isoxazol-6-yloxy)-2,2-dimethyl-propionic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL190352; BDBM50164209
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| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
Plantagineoside B
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2159606; BDBM50394345
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| Activity |
EC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
(5r)-5-(3-{[3-(6-Methoxy-1,2-Benzoxazol-3-Yl)-2-Oxo-2,3-Dihydro-1h-Benzimidazol-1-Yl]methyl}phenyl)-5-Methyl-1,3-Oxazolidine-2,4-Dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947144; SCHEMBL4950298; BDBM50362954; Q27449900
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
2-Phenyl-2-(4-propanoylphenoxy)acetic Acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL427520; CTK6C6508; BDBM50169228; AKOS000165384; AKOS017276395; Phenyl-(4-propionyl-phenoxy)-acetic acid
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| Activity |
IC50 ~ 50000 nM
|
[10] | |||
| Compound Name |
(S)-2-(3-((3-(4-Methoxybenzoyl)-2,6-dimethyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL510180; SCHEMBL13959211; BDBM50244656
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(S)-2-(4-Fluoro-3-((6-methoxy-3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL462378; BDBM50244699
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946753; BDBM50362974
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(5-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946572; BDBM50362973
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(5R)-5-[3-[[3-(6-Chloro-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947145; SCHEMBL14261747; BDBM50362968
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(S)-2-(4-Fluoro-3-((3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL455127; BDBM50244609
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-3-(3-trifluoromethyl-phenoxy)-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL197848; BDBM50173370
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| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
(2S)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946952; BDBM50362959
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(S)-2-(4-Chloro-3-((6-methoxy-3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL460073; BDBM50244701
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(2R)-2-[5-[[3-(4-Tert-butylphenyl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]-2-chlorophenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946568; BDBM50362951
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(S)-2-(4-Chloro-3-((3-(4-chlorophenoxy)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL452054; SCHEMBL13959273; BDBM50244611
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| Activity |
IC50 ~ 50000 nM
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[11] | |||
| Compound Name |
(S)-2-(4-Chloro-3-((3-(4-chlorophenoxy)-6-fluoro-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL461378; BDBM50244747
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(5R)-5-[3-[[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947140; SCHEMBL14261717; BDBM50362965
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-[(4-chlorophenyl)methyl]-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946566; BDBM50362969
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(4-Isopropyl-phenyl)-(4-propionyl-2,6-dipropyl-phenylamino)-acetic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL187612; BDBM50169257
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| Activity |
IC50 ~ 50000 nM
|
[10] | |||
| Compound Name |
5-Benzyl-2-Ethyl-3-{(1s)-5-[2-(1h-Tetrazol-5-Yl)phenyl]-2,3-Dihydro-1h-Inden-1-Yl}-3,5-Dihydro-4h-Imidazo[4,5-C]pyridin-4-One
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2322437; BDBM50426774; Q27451681; 14R
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| Activity |
EC50 ~ 50000 nM
|
[12] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(4-chlorobenzoyl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946567; BDBM50362970
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-6-chloro-3-(3-methanesulfonyl-phenoxy)-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL197823; BDBM50173346
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| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
1-(4-Methoxy-phenyl)-3-(3-trifluoromethyl-phenoxy)-1H-indole-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL198605; BDBM50173355
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| Activity |
IC50 ~ 50000 nM
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[6] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-3-(3-ethoxy-phenoxy)-1H-indole-2-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL372107; BDBM50173352
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| Activity |
IC50 ~ 50000 nM
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[6] | |||
| Compound Name |
(5R)-5-[4-[[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947139; BDBM50362964
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946755; BDBM50362955
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-chloro-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946570; BDBM50362952
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(2R)-2-[4-Chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946953; BDBM50362960
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(S)-2-(2-Chloro-5-((6-chloro-3-(4-chlorophenoxy)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL461944; SCHEMBL13959441; BDBM50244750
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| Activity |
IC50 ~ 50000 nM
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[11] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethoxy)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946756; BDBM50362956
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
(2R)-2-[3-[[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]butanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946955; BDBM50362962
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R)-2-[3-[[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946954; BDBM50362961
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(5R)-5-[3-[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947141; BDBM50362966
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(S)-2-(2-Chloro-5-((6-methoxy-3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL459466; BDBM50244702
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(2R,3R,4S,5S,6R)-2-[(3R,5R)-1,7-Bis(3,4-dihydroxyphenyl)-5-hydroxyheptan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL465800; BDBM50394341; [(1R,3R)-1-(3,4-Dihydroxyphenethyl)-3-hydroxy-5-(3,4-dihydroxyphenyl)pentyl]beta-D-glucopyranoside
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| Activity |
EC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
CID 11592357
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947142; SCHEMBL4947295; BDBM50362967
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| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-6-chloro-3-[3-(4-trifluoromethyl-1H-pyrrol-2-yl)-phenoxy]-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL198365; BDBM50173368
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947143; BDBM50362953
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R)-2-[4-Chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947146; BDBM50362948
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(S)-2-(2-Chloro-5-((3-(4-chlorophenoxy)-6-fluoro-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL518499; BDBM50244748
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(5R)-5-[2-[[3-(6-Methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947138; BDBM50362963
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
5-(4-(2-(5-Methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-phenyl-2H-1,2,3-triazole-4-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL489506; BDBM50248411
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[13] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-5-hydroxy-3-(3-trifluoromethyl-phenoxy)-1H-indole-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL373048; BDBM50173367
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
(S)-7-{3-[2-Chloro-4-(2,2,2-trifluoro-ethoxy)-phenoxy]-propoxy}-2-methyl-chroman-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL180928; SCHEMBL6797892; BDBM50168569
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[14] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-5-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946757; BDBM50362957
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(S)-2-(2-Fluoro-5-((3-(4-methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL507477; BDBM50244610
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(S)-2-(2-Chloro-5-((3-(4-chlorophenoxy)-2-methyl-6-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL517436; BDBM50244808
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(S)-2-(3-((3-(4-Chlorophenoxy)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)-4-fluorophenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL509369; BDBM50244654
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(S)-2-(3-((3-(4-Methoxybenzoyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)phenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL455126; BDBM50244608
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
(3S,4S)-4-[[4-[2-(5-Methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3398452; SCHEMBL12617588; BDBM50063488
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[15] | |||
| Compound Name |
(5R)-5-[4-Chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1947147; SCHEMBL14261739; BDBM50362949
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R,3R,4S,5S,6R)-2-[(3R,5R)-5-Hydroxy-1,7-bis(4-hydroxyphenyl)heptan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL516827; BDBM50394343; [(1R,3R)-1-(4-Hydroxyphenethyl)-3-hydroxy-5-(4-hydroxyphenyl)pentyl]beta-D-glucopyranoside
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
(2S)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}pentanoic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL560160; BDBM50293850
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[16] | |||
| Compound Name |
(S)-2-(5-((3-(4-Chlorophenoxy)-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)-2-fluorophenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL455130; BDBM50244655
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
1-(4-Tert-Butyl-phenyl)-3-[4-(4-trifluoromethyl-1H-pyrrol-2-yl)-phenoxy]-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL426105; BDBM50173345
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(7-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946571; BDBM50362972
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(S)-2-(5-((3-(4-Chlorophenoxy)-6-fluoro-2-methyl-1H-pyrrolo[2,3-b]pyridin-1-yl)methyl)-2-fluorophenoxy)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL461379; BDBM50244749
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
Plantagineoside C
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2159607; BDBM50394344
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-5-(trifluoromethoxy)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946758; BDBM50362958
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
3-(3-Hydroxy-phenoxy)-1-(3-isopropyl-phenyl)-1H-indole-2-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL372850; BDBM50173360
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-chloro-1,3-benzothiazol-2-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946569; BDBM50362971
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
(2R)-2-[2-Chloro-5-[[3-(5-chloro-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1946754; BDBM50362975
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[9] | |||
| Compound Name |
N-(Benzenesulfonyl)-2-[(5-chloro-1,3-benzothiazol-2-yl)sulfanyl]octanamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1808555; BDBM50349443
Click to Show/Hide
|
||||
| Activity |
EC50 = 50600 nM
|
[17] | |||
| Compound Name |
7-Chloro-8-methyl-2-phenylquinoline-4-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
4-quinolinecarboxylic acid, 7-chloro-8-methyl-2-phenyl-; NSC40306; MLS000737014; CHEMBL1565327; Oprea1_131928; SCHEMBL17211711; CTK4J1990; DTXSID80285050; HMS2751B15; ALBB-000648; ZINC1671896; 4334AE; BBL016961; BDBM50462441; MFCD03422093; NSC-40306; NSC400903; STK437244; AKOS003323222; MCULE-9589916425; NSC-400903; SMR000393970; VS-05726; ST50843130; Y-0452
Click to Show/Hide
|
||||
| Activity |
EC50 = 52400 nM
|
[18] | |||
| Compound Name |
4-[(3R,3As,6R,6aS)-3-(1,3-benzodioxol-5-yl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-6-yl]-2-methoxyphenol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2011540; BDBM50379798
Click to Show/Hide
|
||||
| Activity |
EC50 = 53200 nM
|
[19] | |||
| Compound Name |
(S)-2-(5-Chlorobenzo[d]thiazol-2-ylthio)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL583796; BDBM50299266
Click to Show/Hide
|
||||
| Activity |
EC50 = 55900 nM
|
[20] | |||
| Compound Name |
(R)-2-(5-Methoxybenzo[d]thiazol-2-ylthio)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL572662; BDBM50299265
Click to Show/Hide
|
||||
| Activity |
EC50 = 57300 nM
|
[20] | |||
| Compound Name |
(S)-3-(3-((E)-1-(4-Hydroxybenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL488991; BDBM50264412
Click to Show/Hide
|
||||
| Activity |
EC50 = 58800 nM
|
[21] | |||
| Compound Name |
Pluviatilol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2011539; BDBM50379793; Q15425255
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 60000 nM
|
[19] | |||
| Compound Name |
Epipinoresinol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
(+)-Epipinoresinol; epi-pinoresinol; Pinoresinol; UNII-6YKG9JJC1S; 6YKG9JJC1S; Q63408653; (+)-epi-pinoresinol; MLS002473314; CHEMBL487611; SCHEMBL10019016; HMS2196C10; BDBM50379794; ZINC12153081; SMR001397395
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 60000 nM
|
[19] | |||
| Compound Name |
4-[(3R,3Ar,6S,6aR)-3-(1,3-benzodioxol-5-yl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-6-yl]-2,6-dimethoxyphenol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2011538; BDBM50379792
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 60000 nM
|
[19] | |||
| Compound Name |
2,2-Dimethyl-5-[4-[(E)-3-phenylprop-2-enoyl]phenoxy]pentanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1828828; BDBM50353759
Click to Show/Hide
|
||||
| Activity |
EC50 = 61500 nM
|
[22] | |||
| Compound Name |
2-[(5-Chlorobenzothiazole)-2-ylthio]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL566081
Click to Show/Hide
|
||||
| Activity |
EC50 = 62500 nM
|
[20] | |||
| Compound Name |
2-Methyl-2-[4-[2-[4-[(E)-3-phenylprop-2-enoyl]phenoxy]ethyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2204701; BDBM50402004
Click to Show/Hide
|
||||
| Activity |
EC50 = 64000 nM
|
[23] | |||
| Compound Name |
Lithium;5-(3-carboxyphenyl)-2-[(2,4-dichlorobenzoyl)amino]benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL325172
Click to Show/Hide
|
||||
| Activity |
Ki = 67000 nM
|
[24] | |||
| Compound Name |
4-Chloro-N-[2-[4-[1-(methanesulfonamido)-2-methyl-1-oxopropan-2-yl]oxyphenyl]ethyl]benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2153842; BDBM50392680
Click to Show/Hide
|
||||
| Activity |
IC50 = 68500 nM
|
[25] | |||
| Compound Name |
2-[(6-Ethoxy-1,3-benzothiazol-2-yl)thio]-2-methylpropanoic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL583065; BDBM50299267
Click to Show/Hide
|
||||
| Activity |
EC50 = 69300 nM
|
[20] | |||
| Compound Name |
(R)-2-(5-Chlorobenzo[d]thiazol-2-ylthio)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL567389; BDBM50299269
Click to Show/Hide
|
||||
| Activity |
EC50 = 73500 nM
|
[20] | |||
| Compound Name |
2-[4-(2-Hydroxyethyl)phenoxy]-2-methylpropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2204684; SCHEMBL3845467; BDBM50402007
Click to Show/Hide
|
||||
| Activity |
EC50 = 75100 nM
|
[23] | |||
| Compound Name |
Trp-glu
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
H-Trp-Glu-OH; G3335; tryptophanyl-glutamic acid; CHEMBL39176; Tryptophyl-Glutamate; (2S)-2-[[(2S)-2-amino-3-(1H-indol-3-yl)propanoyl]amino]pentanedioic acid; tryptophylglutamic acid; L-Trp-L-Glu; L-tryptophyl-L-glutamic acid; L-Tryptophan-L-glutamic acid; l-tryptophanyl-l-glutamic acid; TRYPTOPHYL-GLUTAMIC ACID; SCHEMBL3547828; N-L-Tryptophyl-L-glutamic acid; CTK7J1923; ZINC2384989; BDBM50240464; Q27144978; PPARgamma Antagonist III, G3335 - CAS 36099-95-3; 2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-pentanedioic acid; (S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-propionylamino]-pentanedioic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 83400 nM
|
[26] | |||
| Compound Name |
Rac-2-[(6-Bromo-1,3-benzothiazol-2-yl)thio]propanoic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL575316; BDBM50299268
Click to Show/Hide
|
||||
| Activity |
EC50 = 84300 nM
|
[20] | |||
| Compound Name |
5-Chloro-2-[(E)-3-[2-(4-methoxybenzoyl)-4-methylpyrrol-1-yl]prop-1-enyl]-N-methylsulfonylbenzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1641708; SCHEMBL2327521; SCHEMBL2327530; SMP-534; BDBM50334217
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 90000 nM
|
[27] | |||
| Compound Name |
2,2-Dimethyl-5-[4-[(E)-2-naphthalen-2-ylethenyl]phenoxy]pentanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3752362
Click to Show/Hide
|
||||
| Activity |
EC50 = 90000 nM
|
[2] | |||
| Compound Name |
Phenylpropanoic acid derivative, 60
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL514696; SCHEMBL5727707; BDBM34033; (2S)-3-[4-[3-(N-methylanilino)propyl]phenyl]-2-pyrrol-1-ylpropanoic acid
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[28] | |||
| Compound Name |
6-Methoxy-1-oxo-3-phenyl-1H-indene-2-carboxylic acid ethyl ester
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL213547; SCHEMBL3572575; CTK3C9392; DTXSID40631539; BDBM50191605; Ethyl 6-methoxy-1-oxo-3-phenyl-1H-indene-2-carboxylate; ETHYL 5-METHOXY-3-OXO-1-PHENYLINDENE-2-CARBOXYLATE; 1-Oxo-3-phenyl-6-methoxy-1H-indene-2-carboxylic acid ethyl ester; 1H-Indene-2-carboxylic acid, 6-methoxy-1-oxo-3-phenyl-, ethyl ester
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
N-(4-(4-Trifluoromethylbenzyl)carbamoylphenyl)-3-((4R)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3601088; SCHEMBL16385852; BDBM50109262
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[30] | |||
| Compound Name |
CID 71721539
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
NXT629; CHEMBL3264932; SCHEMBL15272225; BDBM50013726; HY-114263; CS-0080837
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
(S)-3-(3-Bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-phenylpiperazin-1-yl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1090557; SCHEMBL4482985; BDBM50315310
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[32] | |||
| Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)phenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL374682; SCHEMBL1400652; Indanylacetic Acid Analog, 34z; BDBM21811
Click to Show/Hide
|
||||
| Activity |
EC50 = 100000 nM
|
[33] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-(3-ethoxyphenyl)benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL118852
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[24] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-(2-pyridin-2-ylethoxy)benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL420525; SCHEMBL7036028
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[24] | |||
| Compound Name |
Phenylpropanoic acid derivative, 32
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL477940; SCHEMBL5727584; BDBM34022
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[28] | |||
| Compound Name |
2-[3-[(4-Methylphenyl)carbamoyl]-4-piperidin-1-ylphenyl]indazole-6-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3746821; SCHEMBL17317386; BDBM50500150
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[34] | |||
| Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-methoxyphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL427080; SCHEMBL1400614; BDBM21813; Indanylacetic Acid Analog, 34ab
Click to Show/Hide
|
||||
| Activity |
EC50 = 100000 nM
|
[33] | |||
| Compound Name |
Lithium;5-(6-chloropyrazin-2-yl)oxy-2-[(2,4-dichlorobenzoyl)amino]benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL119111; SCHEMBL7040743
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[24] | |||
| Compound Name |
(2R)-3,3,3-Trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]-2-hydroxypropanamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2323021; SCHEMBL3628001; HSD-621; BDBM50426478
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[35] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-(3-nitropyridin-2-yl)oxybenzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL330938; SCHEMBL7155567
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[24] | |||
| Compound Name |
3-[[(4R)-4-Benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]-N-[4-(cyclohexylmethylcarbamoyl)phenyl]benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3601092; SCHEMBL16385917; BDBM50109196
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[30] | |||
| Compound Name |
(2R)-3-[4-[3-(5-Methyl-2-phenyl-1,3-oxazol-4-yl)propyl]phenyl]-2-(triazol-1-yl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL595440
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[36] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-[(4-ethoxyphenyl)methoxy]benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL119798; SCHEMBL7034813
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[24] | |||
| Compound Name |
(S)-3-(4-(2-(5-Methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-p-tolylpiperazin-1-yl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1090860; BDBM50315308
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[32] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-(5-nitropyridin-2-yl)oxybenzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL118546; SCHEMBL7040861
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[24] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-quinolin-8-ylbenzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL119078
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[24] | |||
| Compound Name |
Phenylpropanoic acid derivative, 33
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL477941; SCHEMBL5726606; BDBM34023; (2S)-3-[4-[3-(N-methylanilino)prop-1-ynyl]phenyl]-2-pyrrol-1-ylpropanoic acid
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[28] | |||
| Compound Name |
3-[[(4S)-4-Benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]-N-[4-[[4-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3601094; BDBM50109165
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[30] | |||
| Compound Name |
N-(4-Benzylcarbamoylphenyl)-3-((4R)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3600934; SCHEMBL16385824; BDBM50109159; N-[4-(benzylcarbamoyl)phenyl]-3-[[(4R)-4-benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]benzamide
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[30] | |||
| Compound Name |
(S)-2-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1090861; SCHEMBL4484300; BDBM50315309
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[32] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-(2-thiophen-2-ylethoxy)benzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL119278; SCHEMBL7034820
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[24] | |||
| Compound Name |
Lithium;2-[(2,4-dichlorobenzoyl)amino]-5-pyrimidin-2-yloxybenzoate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL118206; SCHEMBL7033049
Click to Show/Hide
|
||||
| Activity |
Ki ~ 100000 nM
|
[24] | |||
| Compound Name |
N-(4-Pentylcarbamoylphenyl)-3-((4S)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3601095; BDBM50109164
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[30] | |||
| Compound Name |
(2R)-3-[4-[3-(5-Methyl-2-phenyl-1,3-oxazol-4-yl)propyl]phenyl]-2-(1,2,4-triazol-1-yl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL605520
Click to Show/Hide
|
||||
| Activity |
EC50 ~ 100000 nM
|
[36] | |||
| Compound Name |
2,2-Dimethyl-5-[4-[(E)-2-pyridin-4-ylethenyl]phenoxy]pentanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3751930
Click to Show/Hide
|
||||
| Activity |
EC50 = 103200 nM
|
[2] | |||
| Compound Name |
2-[(1S)-5-[3-(2,4-Dimethylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220785; SCHEMBL3019471; Indanylacetic Acid Analog, 17l; BDBM21765
Click to Show/Hide
|
||||
| Activity |
EC50 = 106831.67 nM
|
[33] | |||
| Compound Name |
N-(4-Acetamidophenyl)sulfonyl-2-[(5-chloro-1,3-benzothiazol-2-yl)sulfanyl]pentanamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781940; BDBM50155327
Click to Show/Hide
|
||||
| Activity |
IC50 = 108000 nM
|
[37] | |||
| Compound Name |
2-[(1S)-5-{3-[2-Acetamido-4-(1H-1,2,3-triazol-1-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219817; Indanylacetic Acid Analog, 17v; BDBM21775
Click to Show/Hide
|
||||
| Activity |
EC50 = 108692.61 nM
|
[33] | |||
| Compound Name |
5-[4-[(E)-3-Phenylprop-2-enoyl]phenoxy]pentanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1828827; BDBM50353758
Click to Show/Hide
|
||||
| Activity |
EC50 = 109300 nM
|
[22] | |||
| Compound Name |
2-[(1S)-5-[3-(4-Cyano-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL375747; SCHEMBL1400667; Indanylacetic Acid Analog, 17s; BDBM21772
Click to Show/Hide
|
||||
| Activity |
EC50 = 127320.99 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-{3-[4-(Pyrimidin-5-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220448; SCHEMBL1400268; Indanylacetic Acid Analog, 29f; BDBM21763; 2-[(1S)-5-[3-(4-pyrimidin-5-ylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 137372.56 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-{3-[2-Chloro-4-(4H-1,2,4-triazol-4-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220990; SCHEMBL1400260; Indanylacetic Acid Analog, 17w; BDBM21776; 2-[(1S)-5-[3-[2-chloro-4-(1,2,4-triazol-4-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 145982.23 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(Trifluoromethoxy)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(trifluoromethoxy)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL373605; SCHEMBL1400262; Indanylacetic Acid Analog, 17d; BDBM21756
Click to Show/Hide
|
||||
| Activity |
EC50 = 147061.84 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(1H-Indol-6-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(1H-indol-6-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220893; SCHEMBL1400787; Indanylacetic Acid Analog, 29c; BDBM21780
Click to Show/Hide
|
||||
| Activity |
EC50 = 151530.48 nM
|
[33] | |||
| Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-(hydroxymethyl)-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL424933; SCHEMBL1400982; BDBM21814; Indanylacetic Acid Analog, 34ac
Click to Show/Hide
|
||||
| Activity |
EC50 = 154099.06 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(4-Cyanophenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220508; SCHEMBL1400780; Indanylacetic Acid Analog, 17g; BDBM21759
Click to Show/Hide
|
||||
| Activity |
EC50 = 175428.44 nM
|
[33] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 71 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
N-(2-adamantyl)-N'-propylsulfamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL218643; SCHEMBL3117688; BDBM50202584; ZINC35091103
Click to Show/Hide
|
||||
| Activity |
EC50 > 10000000 nM
|
[38] | |||
| Compound Name |
[2'-[(Cyclopropanecarbonyl-ethyl-amino)-methyl]-4'-(6-ethoxy-pyridin-3-yl)-6-methoxy-biphenyl-3-yl]-acetic acid sodium salt
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1668898
Click to Show/Hide
|
||||
| Activity |
IC50 > 250000 nM
|
[39] | |||
| Compound Name |
2-[(1S)-5-[3-(4-Cyano-2-propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219661; SCHEMBL1400255; Indanylacetic Acid Analog, 17o; BDBM21768
Click to Show/Hide
|
||||
| Activity |
EC50 = 253162.86 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(Furan-3-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(furan-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL376418; SCHEMBL1400869; Indanylacetic Acid Analog, 29b; BDBM21779
Click to Show/Hide
|
||||
| Activity |
EC50 = 305844.02 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{4-[5-(Trifluoromethyl)pyridin-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220570; SCHEMBL1400566; Indanylacetic Acid Analog, 29i; BDBM21785
Click to Show/Hide
|
||||
| Activity |
EC50 = 344826 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL374545; SCHEMBL1400856; Indanylacetic Acid Analog, 34u; BDBM21806
Click to Show/Hide
|
||||
| Activity |
EC50 = 395275.59 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{4-[4-(Carboxymethyl)-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL375072; SCHEMBL3120428; BDBM21815; Indanylacetic Acid Analog, 34ad
Click to Show/Hide
|
||||
| Activity |
EC50 = 403180.95 nM
|
[33] | |||
| Compound Name |
2-Isopropoxy-3-(4-(2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL77040; BDBM50103954; 2-Isopropoxy-3-{4-[2-(5-phenyl-[1,2,4]oxadiazol-3-yl)-ethoxy]-phenyl}-propionic acid; alpha-Isopropoxy-4-[2-(5-phenyl-1,2,4-oxadiazole-3-yl)ethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 500034.53 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-(4-Ethylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220421; SCHEMBL1400619; Indanylacetic Acid Analog, 17b; BDBM21754
Click to Show/Hide
|
||||
| Activity |
EC50 = 505126.32 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-{3-[4-(Pyridin-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219944; SCHEMBL1400495; Indanylacetic Acid Analog, 29d; BDBM21781; 2-[(1S)-5-[3-(4-pyridin-3-ylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 591697.86 nM
|
[33] | |||
| Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL222247; SCHEMBL1400267; BDBM21812; Indanylacetic Acid Analog, 34aa
Click to Show/Hide
|
||||
| Activity |
EC50 = 591697.86 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(Trifluoromethyl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(trifluoromethyl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220422; SCHEMBL1400241; Indanylacetic Acid Analog, 17c; BDBM21755
Click to Show/Hide
|
||||
| Activity |
EC50 = 621155.02 nM
|
[33] | |||
| Compound Name |
3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1209170; SCHEMBL4283477; BDBM50323530
Click to Show/Hide
|
||||
| Activity |
EC50 = 680000 nM
|
[41] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(4-ethyl-1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220635; SCHEMBL1400693; Indanylacetic Acid Analog, 34d; BDBM21789
Click to Show/Hide
|
||||
| Activity |
EC50 = 781267.93 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220837; SCHEMBL1400266; Indanylacetic Acid Analog, 34j; BDBM21795
Click to Show/Hide
|
||||
| Activity |
EC50 = 800018.44 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(trifluoromethyl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[2-propyl-4-(trifluoromethyl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL219686; SCHEMBL1400334; Indanylacetic Acid Analog, 17n; BDBM21767
Click to Show/Hide
|
||||
| Activity |
EC50 = 877202.78 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{4-[5-(Dimethylcarbamoyl)-4-methyl-1,3-thiazol-2-yl]-2-methoxyphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220173; SCHEMBL1400660; Indanylacetic Acid Analog, 34y; BDBM21810
Click to Show/Hide
|
||||
| Activity |
EC50 = 1245374.59 nM
|
[33] | |||
| Compound Name |
3-(4-(2-(5-(4-Fluorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL262981; BDBM50103951; 3-(4-{2-[5-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-2-isopropoxy-propionic acid; alpha-Isopropoxy-4-[2-[5-(4-fluorophenyl)-1,2,4-oxadiazole-3-yl]ethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 1267651.87 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4-methoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL222508; SCHEMBL1400402; BDBM21817; Indanylacetic Acid Analog, 34af
Click to Show/Hide
|
||||
| Activity |
EC50 = 1324646.51 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(4-Ethyl-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220681; SCHEMBL1400818; Indanylacetic Acid Analog, 17r; BDBM21771
Click to Show/Hide
|
||||
| Activity |
EC50 = 1428564.98 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220151; SCHEMBL1400676; Indanylacetic Acid Analog, 34w; BDBM21808
Click to Show/Hide
|
||||
| Activity |
EC50 = 1785665.06 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(1,3-Benzothiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL424939; SCHEMBL1400421; Indanylacetic Acid Analog, 34t; BDBM21805
Click to Show/Hide
|
||||
| Activity |
EC50 = 1901078.28 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{2-Methyl-4-[3-(trifluoromethyl)-1,2,4-thiadiazol-5-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219688; SCHEMBL1400498; Indanylacetic Acid Analog, 17x; BDBM21777
Click to Show/Hide
|
||||
| Activity |
EC50 = 1923091.73 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219609; SCHEMBL1400824; BDBM21825; Indanylacetic Acid Analog, 34an
Click to Show/Hide
|
||||
| Activity |
EC50 = 1923091.73 nM
|
[33] | |||
| Compound Name |
3-(4-(2-(5-(3-Fluorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL305723; BDBM50103960; 3-(4-{2-[5-(3-Fluoro-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-2-isopropoxy-propionic acid; alpha-Isopropoxy-4-[2-[5-(3-fluorophenyl)-1,2,4-oxadiazole-3-yl]ethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 2004472.03 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-(3-{2-Methoxy-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219687; SCHEMBL1400842; Indanylacetic Acid Analog, 34i; BDBM21794
Click to Show/Hide
|
||||
| Activity |
EC50 = 2288231.71 nM
|
[33] | |||
| Compound Name |
2-Isopropoxy-3-(4-(2-(5-(2-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL433316; BDBM50103945
Click to Show/Hide
|
||||
| Activity |
EC50 = 2500345.36 nM
|
[40] | |||
| Compound Name |
3-(4-(2-(5-(4-Chlorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL305854; BDBM50103944; 3-(4-{2-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-2-isopropoxy-propionic acid; alpha-Isopropoxy-4-[2-[5-(4-chlorophenyl)-1,2,4-oxadiazole-3-yl]ethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 2500345.36 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4,5,6,7-Tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL375812; SCHEMBL1400287; Indanylacetic Acid Analog, 34o; BDBM21800
Click to Show/Hide
|
||||
| Activity |
EC50 = 2557407.89 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(2-Methoxy-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL375427; Indanylacetic Acid Analog, 34s; BDBM21804
Click to Show/Hide
|
||||
| Activity |
EC50 = 3048596.87 nM
|
[33] | |||
| Compound Name |
3-(4-(2-(5-(3-Chlorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL78442; BDBM50103953; 3-(4-{2-[5-(3-Chloro-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-2-isopropoxy-propionic acid; alpha-Isopropoxy-4-[2-[5-(3-chlorophenyl)-1,2,4-oxadiazole-3-yl]ethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 3126079.37 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220059; SCHEMBL1400323; Indanylacetic Acid Analog, 34c; BDBM21788
Click to Show/Hide
|
||||
| Activity |
EC50 = 3731642.24 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[2-methoxy-4-(1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220124; SCHEMBL1400868; Indanylacetic Acid Analog, 34b; BDBM21787
Click to Show/Hide
|
||||
| Activity |
EC50 = 3921931.46 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220557; SCHEMBL1400349; Indanylacetic Acid Analog, 34f; BDBM21791
Click to Show/Hide
|
||||
| Activity |
EC50 = 3937313.54 nM
|
[33] | |||
| Compound Name |
3-[4-[2-(5-Cyclohexyl-1,2,4-oxadiazol-3-yl)ethoxy]phenyl]-2-propan-2-yloxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2262883; BDBM50487311
Click to Show/Hide
|
||||
| Activity |
EC50 = 4168693.83 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-(2-(5-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL80791; BDBM50103941
Click to Show/Hide
|
||||
| Activity |
EC50 = 5000345.35 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-(3-{2-Propyl-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL374090; SCHEMBL1400786; Indanylacetic Acid Analog, 34h; BDBM21793
Click to Show/Hide
|
||||
| Activity |
EC50 = 5075747.39 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{2-Methoxy-4-[4-(propan-2-yloxy)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219669; SCHEMBL1400978; BDBM21822; Indanylacetic Acid Analog, 34ak
Click to Show/Hide
|
||||
| Activity |
EC50 = 5555203.85 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219668; SCHEMBL1400300; Indanylacetic Acid Analog, 34v; BDBM21807
Click to Show/Hide
|
||||
| Activity |
EC50 = 5714786.37 nM
|
[33] | |||
| Compound Name |
3-(4-((5-(4-Fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL78523; BDBM50103952; alpha-Isopropoxy-4-[5-(4-fluorophenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid; 3-{4-[5-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-2-isopropoxy-propionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 6251726.93 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-phenyl-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL311429; BDBM50103938; 2-Isopropoxy-3-[4-(5-phenyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid; alpha-Isopropoxy-4-(5-phenyl-1,2,4-oxadiazole-3-ylmethoxy)benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 6251726.93 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220152; SCHEMBL1400686; BDBM21824; Indanylacetic Acid Analog, 34am
Click to Show/Hide
|
||||
| Activity |
EC50 = 6666532.49 nM
|
[33] | |||
| Compound Name |
((1S)-5-{3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl)acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL373813; SCHEMBL3023128; Indanylacetic Acid Analog, 34e; BDBM21790
Click to Show/Hide
|
||||
| Activity |
EC50 = 6802992.62 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-(3-{4-[5-(Dimethylcarbamoyl)-4-methyl-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220662; SCHEMBL1400162; Indanylacetic Acid Analog, 34x; BDBM21809
Click to Show/Hide
|
||||
| Activity |
EC50 = 7143318.26 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL221101; SCHEMBL3122256; Indanylacetic Acid Analog, 34l; BDBM21797
Click to Show/Hide
|
||||
| Activity |
EC50 = 8928941.96 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[2-propyl-4-(1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL374901; SCHEMBL1400247; Indanylacetic Acid Analog, 34a; BDBM21786
Click to Show/Hide
|
||||
| Activity |
EC50 = 9009485.69 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL387350; SCHEMBL1400331; BDBM21819; Indanylacetic Acid Analog, 34ah
Click to Show/Hide
|
||||
| Activity |
EC50 = 9523574.86 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(2-Propyl-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL1400218; CHEMBL2236890; Indanylacetic Acid Analog, 34r; BDBM21803
Click to Show/Hide
|
||||
| Activity |
EC50 = 9901477.39 nM
|
[33] | |||
| Compound Name |
N-Hexadecylsulfamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL218795; 1-(sulfamoylamino)hexadecane; SCHEMBL3124345; BDBM50202581; ZINC43543918
Click to Show/Hide
|
||||
| Activity |
EC50 > 10000000 nM
|
[38] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL223748; SCHEMBL1400573; BDBM21818; Indanylacetic Acid Analog, 34ag
Click to Show/Hide
|
||||
| Activity |
EC50 = 10000000 nM
|
[33] | |||
| Compound Name |
N-Octadecylsulfamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL218794; 1-(sulfamoylamino)octadecane; SCHEMBL1228645; CTK4J1791; BDBM50202579; ZINC43543913
Click to Show/Hide
|
||||
| Activity |
EC50 > 10000000 nM
|
[38] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Tert-butyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL220117; SCHEMBL1400351; Indanylacetic Acid Analog, 34g; BDBM21792
Click to Show/Hide
|
||||
| Activity |
EC50 = 11494762.43 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL374925; SCHEMBL1400962; Indanylacetic Acid Analog, 34k; BDBM21796
Click to Show/Hide
|
||||
| Activity |
EC50 = 12047585.03 nM
|
[33] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-m-tolyl-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL80301; BDBM50103956; 2-Isopropoxy-3-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid; alpha-Isopropoxy-4-[5-(3-methylphenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 12676518.66 nM
|
[40] | |||
| Compound Name |
3-(4-((5-(3-Fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL80772; BDBM50103958; alpha-Isopropoxy-4-[5-(3-fluorophenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid; 3-{4-[5-(3-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-2-isopropoxy-propionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 13212956.34 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL373791; SCHEMBL1400704; BDBM21823; Indanylacetic Acid Analog, 34al
Click to Show/Hide
|
||||
| Activity |
EC50 = 16394568.85 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL222248; SCHEMBL1400371; Indanylacetic Acid Analog, 34n; BDBM21799
Click to Show/Hide
|
||||
| Activity |
EC50 = 18866876.21 nM
|
[33] | |||
| Compound Name |
3-(4-(2-(5-(3,5-Bis(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL80979; BDBM50103957
Click to Show/Hide
|
||||
| Activity |
EC50 = 20044720.27 nM
|
[40] | |||
| Compound Name |
2-[(1S)-5-(3-{4-[4-(Propan-2-yloxy)-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL436514; SCHEMBL1400496; BDBM21821; Indanylacetic Acid Analog, 34aj
Click to Show/Hide
|
||||
| Activity |
EC50 = 21276490.8 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL219617; SCHEMBL1400681; Indanylacetic Acid Analog, 34q; BDBM21802
Click to Show/Hide
|
||||
| Activity |
EC50 = 22724796.35 nM
|
[33] | |||
| Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL1400467; CHEMBL2113263; Indanylacetic Acid Analog, 34p; BDBM21801
Click to Show/Hide
|
||||
| Activity |
EC50 = 23254124.86 nM
|
[33] | |||
| Compound Name |
3-[4-[[5-[4-(2-Methylpropyl)phenyl]-1,2,4-oxadiazol-3-yl]methoxy]phenyl]-2-propan-2-yloxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2262884; BDBM50487310; alpha-Isopropoxy-4-[5-(4-isobutylphenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 25003453.62 nM
|
[40] | |||
| Compound Name |
3-(4-((5-(4-Bromophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL310962; BDBM50103947; alpha-Isopropoxy-4-[5-(4-bromophenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid; 3-{4-[5-(4-Bromo-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-2-isopropoxy-propionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 25003453.62 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-o-tolyl-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL433306; BDBM50103939; 2-Isopropoxy-3-[4-(5-o-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid; alpha-Isopropoxy-4-[5-(2-methylphenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 25003453.62 nM
|
[40] | |||
| Compound Name |
3-(4-((5-(3,5-Difluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL309778; SCHEMBL18644985; BDBM50103946; 3-{4-[5-(3,5-Difluoro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-2-isopropoxy-propionic acid; alpha-Isopropoxy-4-[5-(3,5-difluorophenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 25003453.62 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-(4-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL312791; BDBM50103949
Click to Show/Hide
|
||||
| Activity |
EC50 = 31260793.67 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-p-tolyl-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL310426; BDBM50103948; 2-Isopropoxy-3-[4-(5-p-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid; alpha-Isopropoxy-4-[5-(4-methylphenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
Click to Show/Hide
|
||||
| Activity |
EC50 = 40086671.76 nM
|
[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-(4-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
Click to Show/Hide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL80905; BDBM50103959
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| Activity |
EC50 = 50003453.5 nM
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[40] | |||
| Compound Name |
3-(4-((5-(4-Chlorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL80671; BDBM50103943; alpha-Isopropoxy-4-[5-(4-chlorophenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid; 3-{4-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-2-isopropoxy-propionic acid
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| Activity |
EC50 = 77090346.91 nM
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[40] | |||
| Compound Name |
2-Isopropoxy-3-(4-((5-(4-isopropylphenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL80364; 2-Isopropoxy-3-{4-[5-(4-isopropyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid; BDBM50103950; alpha-Isopropoxy-4-[5-(4-isopropylphenyl)-1,2,4-oxadiazole-3-ylmethoxy]benzenepropionic acid
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| Activity |
EC50 = 77090346.91 nM
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[40] | |||
| Compound Name |
3-(4-((5-(3,5-Bis(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL307728; BDBM50103940
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| Activity |
EC50 = 166724721.3 nM
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[40] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
| References | Top | ||||
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