Target Poor or Non Binder(s) Information
Target General Information | Top | ||||
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Target ID | T58921 | Target Info | |||
Target Name | Peroxisome proliferator-activated receptor gamma (PPAR-gamma) | ||||
Synonyms |
PPAR-gamma; Nuclear receptor subfamily 1 group C member 3; NR1C3
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Target Type | Successful Target | ||||
Gene Name | PPARG | ||||
Biochemical Class | Nuclear hormone receptor | ||||
UniProt ID |
Poor Binders of This Target (in total, 100 binders) | Download | Top | |||
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Compound Name |
FENOFIBRIC ACID
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Approved | Compound Info | ||
Synonyms |
Fenofibric acid; 42017-89-0; Procetofenic acid; 2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropanoic acid; alpha 1081; NSC 281318; LF 178 acid; UNII-BGF9MN2HU1; 2-[4-(4-chlorobenzoyl)phenoxy]-2-methylpropanoic acid; LF 153; FNF Acid; C17H15ClO4; Trilipix; CCRIS 7302; EINECS 255-626-9; BGF9MN2HU1; CHEMBL981; BRN 2058973; CHEBI:83469; 2-[4-(4-Chlorobenzoyl)phenoxy]-2-methylpropionic Acid; Propanoic acid, 2-(4-(4-chlorobenzoyl)phenoxy)-2-methyl-; AK117112; 2-{4-[(4-chlorophenyl)carbonyl]phenoxy}-2-methylpropanoic acid; W-106287
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Activity |
IC50 ~ 50000 nM
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[1] | |||
Compound Name |
Indomethacin
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Approved | Compound Info | ||
Synonyms |
Aconip; Amuno; Arthrexin; Artracin; Artrinovo; Artrivia; Bonidin; Bonidon; Catlep; Confortid; Dolcidium; Dolovin; Durametacin; Elmetacin; Hicin; IMN; Idomethine; Imbrilon; Inacid; Indacin; Indameth; Indmethacine; Indocid; Indocin; Indomecol; Indomed; Indomee; Indometacin; Indometacina; Indometacine; Indometacinum; Indometacyna; Indomethacine; Indomethacinum; Indomethancin; Indomethazine; Indomethegan; Indomethine; Indometicina; Indomo; Indomod; Indoptic; Indoptol; Indorektal; Indoxen; Inflazon; Infrocin; Lausit; Liometacen; Metacen; Metartril; Methazine; Metindol; Mezolin; Miametan; Mikametan; Mobilan; Novomethacin; Reumacide; Sadoreum; Tannex; Vonum; Bonidon Gel; DESMETHYL INDOMETHACIN; Dolcidium PL;Flexin continus; Indocid Pda; Indocid Sr; Indocin Sr; Indolar SR; Indometacyna [Polish]; Indometicina [Spanish]; Inteban sp; Rhemacin LA; Rheumacin LA; I 7378; IN1454; Indomet 140; Aconip (TN); Apo-Indomethacin; Chibro-amuno; Chrono-indicid; Chrono-indocid; Indo-Lemmon; Indo-Spray; Indo-phlogont; Indo-rectolmin; Indo-tablinen; Indocid (TN); Indocid (pharmaceutical); Indocin (TN); Indocin I.V; Indometacina [INN-Spanish]; Indometacine [INN-French]; Indometacinum [INN-Latin]; Indomethacin (USP); Indomethacin [USAN:BAN]; Novo-Methacin; Indochron E-R (TN); Indocin I.V.; Indocin-SR (TN); Indometacin (JP15/INN); Indomethacin & MAP-30; Indomethacin, Indochron E-R, Indocin-SR, Indocid, Indocin, Indomethacin
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Activity |
EC50 = 50000 nM
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[2] | |||
Compound Name |
Bezafibrate
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Approved | Compound Info | ||
Synonyms |
Azufibrat; Befibrat; Befizal; BezaLande; BezaPuren; Bezabeta; Bezacur; Bezafibrat; Bezafibrato; Bezafibratum; Bezafisal;Bezalip; Bezamerck; Bezatol; Cedur; Difaterol; Durabezur; Eulitop; Lipox; Reducterol; Sklerofibrat; Solibay; Azupharma Brand of Bezafibrate; Bayer Brand of Bezafibrate; Berlin Chemie Brand of Bezafibrate; Betapharm Brand of Bezafibrate; Beza Lande; Beza Puren; Bezafibrat PB; Bezafibrate Azupharma Brand; Bezafibrate Bayer Brand; Bezafibrate Betapharm Brand; Bezafibrate Cryopharma Brand; Bezafibrate Elfar Brand; Bezafibrate Hennig Brand; Bezafibrate Hexal Brand; Bezafibrate Isis Brand; Bezafibrate Lakeside Brand; Bezafibrate Merckle Brand; Bezafibrate Roche Brand; Bezafibrate Synthelabo Brand; Bezafibrate TAD Brand; Bezafibrate Teva Brand; Bezafibrato [Spanish]; Bezalip Retard; Bezatol SR; Boehringer Mannheim Brand of Bezafibrate; Cryopharma Brand of Bezafibrate; Elfar Brand of Bezafibrate;Hennig Brand of Bezafibrate; Hexal Brand of Bezafibrate; Isis Brand of Bezafibrate; Lakeside Brand of Bezafibrate; Merckle Brand of Bezafibrate; Regadrin B; Roche Brand of Bezafibrate; Synthelabo Brand of Bezafibrate; TAD Brand of Bezafibrate; Teva Brand of Bezafibrate; BM 15075; LO 44; BF-759; BM 15.075; BM-15075; BM15.075; Berlin-Chemie Brand of Bezafibrate; Beza-Lande; Beza-Puren; Bezafibrate Berlin-Chemie Brand; Bezafibrato [INN-Spanish]; Bezafibratum [INN-Latin]; Bezalip (TN); Bezatol SR (TN); PB, Bezafibrat; BM-15.075; Bezafibrate (JP15/USAN/INN); Bezafibrate [USAN:BAN:INN:JAN]; A-[4-(4-chlorobenzoylaminoethyl)phenoxy]isobutyric acid; 2-(4-{2-[(4-chlorobenzoyl)amino]ethyl}phenoxy)-2-methylpropanoic acid; 2-(p-(2-(p-Chlorobenzamido)ethyl)phenoxy)-2-methylpropionic acid; 2-[4-(2-[4-Chlorobenzamido]ethyl)-phenoxy]-2-methylpropanoic acid; 2-[4-[2-(4-Chlorobenzamido)ethyl]phenoxy]-2-methylpropanoic acid; 2-[4-[2-(4-Chlorobenzamido)ethyl]phenoxy]isobutyric Acid; 2-[4-[2-[(4-chlorobenzoyl)amino]ethyl]phenoxy]-2-methylpropanoic acid
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Activity |
EC50 = 57200 nM
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[3] | |||
Compound Name |
Gemfibrozil
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Approved | Compound Info | ||
Synonyms |
ApoGemfibrozil; Ausgem; Bolutol; Brozil; Cholespid; Clearol; Decrelip; Elmogan; Fetinor; Fibratol; Fibrocit; GFZ; Gemd; Gemfibril; Gemfibromax; Gemfibrosil; Gemfibrozilo; Gemfibrozilum; Gemhexal; Gemlipid; Gemnpid; GenGemfibrozil; Genlip; Gozid; Hidil; Hipolixan; Innogem; Innogen; Ipolipid; Jezil; Lanaterom; Lifibron; Lipazil; Lipigem; Lipira; Lipizyl; Lipozid; Lipur; Litarek; Lopid; Micolip; Normolip; NuGemfibrozil; Pilder; Polyxit; Progemzal; Reducel; Regulip; Renabrazin; Sinelip; Synbrozil; Taborcil; Tentroc; Trialmin; Alphapharm Brand of Gemfibrozil; Apo Gemfibrozil; Apotex Brand of Gemfibrozil; Bayvit Brand of Gemfibrozil; Bexal Brand of Gemfibrozil; Biochemie Brand of Gemfibrozil; Bull Brand of Gemfibrozil; Cantabria Brand of Gemfibrozil; Chem mart Brand of Gemfibrozil; Chem mart Gemfibrozil; DBL Gemfibrozil; Douglas Brand of Gemfibrozil; Farmasierra Brand of Gemfibrozil; Faulding Brand of Gemfibrozil;Ferrer Brand of Gemfibrozil; Gemfibrozilo Bayvit; Gemfibrozilo Bexal; Gemfibrozilo Ur; Gen Gemfibrozil; GenRX Gemfibrozil; Genpharm Brand of Gemfibrozil; Gevilon Uno; Healthsense Brand of Gemfibrozil; Healthsense Gemfibrozil; Hexal Brand of Gemfibrozil; Ipsen Brand of Gemfibrozil; Lipox Gemfi; Lopid R; Menarini Brand of Gemfibrozil; Novo Gemfibrozil; Novopharm Brand of Gemfibrozil; Nu Gemfibrozil; Nu Pharm Brand of Gemfibrozil; PMS Gemfibrozil; Parke Davis Brand of Gemfibrozil; Pfizer Brand of Gemfibrozil; Pharmascience Brand of Gemfibrozil; Quimifar Brand of Gemfibrozil; SBPA Gemfibrozil; Sigma Brand of Gemfibrozil; TAD Brand of Gemfibrozil; Terry White Chemists Brand of Gemfibrozil; Terry White Chemists Gemfibrozil; United Drug Brand of Gemfibrozil; Warner Lambert Brand of Gemfibrozil; CI719; Gemfi 1A Pharma; Apo-Gemfibrozil; Bayvit, Gemfibrozilo; Gem-S; Gemfibrozil, GenRX; Gemfibrozil, Healthsense; Gemfibrozil, SBPA; Gemfibrozilo [INN-Spanish]; Gemfibrozilum [INN-Latin]; Gen-Fibro;Gen-Gemfibrozil; Jezil (TN); Lopid (TN); Low-Lip; Novo-Gemfibrozil; Nu-Gemfibrozil; Nu-Pharm Brand of Gemfibrozil; PMS-Gemfibrozil; TEVA-A; WL-Gemfibrozil; Warner-Lambert Brand of Gemfibrozil; GEMFIBROZIL (SEE ALSO PEROXISOME PROJECT (GEMFIBROZIL)); Gemfibrozil [USAN:BAN:INN]; Gen-Fibro (TN); PEROXISOME PROJECT (GEMFIBROZIL) (SEE ALSO GEMFIBROZIL); Gemfibrozil (JAN/USP/INN); Gemcor, Lopid, Jezil,Gen-Fibro, Gemfibrozil; 1A Brand of Gemfibrozil; 2,2-Dimethyl-5-(2,5-dimethylphenoxy)pentanoic acid; 2,2-Dimethyl-5-(2,5-dimethylphenoxy)valeriansaeure; 2,2-Dimethyl-5-(2,5-xylyloxy)valeriansaeure; 2,2-Dimethyl-5-(2,5-xylyloxy)valeric acid; 5-(2,5-Dimethyl-Phenoxy)-2,2-Dimethyl-Pentanoic Acid; 5-(2,5-Dimethylphenoxy)-2,2-dimethylpentanoic acid; 5-[(2,5-dimethylphenyl)oxy]-2,2-dimethylpentanoic acid
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Activity |
EC50 = 147800 nM
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[4] | |||
Compound Name |
PIRINIXIC ACID
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Preclinical | Compound Info | ||
Synonyms |
Pirinixic acid; 50892-23-4; WY-14643; [4-Chloro-6-(2,3-xylidino)-2-pyrimidinylthio]acetic acid; WY-14,643; WY14643; Wyeth 14,643; Wy 14643; Pirinixic acid [INN]; WY-14643 (Pirinixic Acid); (4-Chloro-6-(2,3-xylidino)-2-pyrimidinylthio)acetic acid; UNII-86C4MRT55A; C14H14ClN3O2S; CCRIS 133; Acidum pirinixicum [INN-Latin]; Acide pirinixique [INN-French]; Acido pirinixico [INN-Spanish]; NSC310038; NSC-310038; NSC 310038; BRN 0759945; ((4-Chloro-6-((2,3-dimethylphenyl)amino)-2-pyrimidinyl)thio)acetic acid; Acetic acid, ((4-chloro-6-(
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Activity |
IC50 = 53700 nM
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[5] | |||
Compound Name |
tagitinin A
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Investigative | Compound Info | ||
Synonyms |
tagitinin A; 59979-61-2; GTPL8701; CHEMBL518700; AC1L48P2; MEGxp0_000075; ACon0_000437; ACon1_000272; BDBM50394802; NCGC00180721-01
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Activity |
IC50 = 55000 nM
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[6] | |||
Compound Name |
(R)-2-(4-Methoxy-3-(4-(trifluoromethyl)benzylcarbamoyl)benzyl)butanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL115604; BDBM50109109; N-[4-(Trifluoromethyl)benzyl]-2-methoxy-5-[(2R)-2-carboxybutyl]benzamide; (R)-2-[4-Methoxy-3-(4-trifluoromethyl-benzylcarbamoyl)-benzyl]-butyric acid; (2R)-2-[[4-methoxy-3-[[4-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
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Activity |
IC50 ~ 50000 nM
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[7] | |||
Compound Name |
3-{4-[2-Amino-6-(4-benzoyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL538875; SCHEMBL2808919; BDBM50296701; 3-[4-[2-amino-6-(4-benzoylpiperazin-1-yl)pyrimidin-4-yl]oxyphenyl]-2-methyl-2-phenoxypropanoic acid
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Activity |
EC50 ~ 50000 nM
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[8] | |||
Compound Name |
2-Phenyl-2-(4-propanoylphenoxy)acetic Acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL427520; CTK6C6508; BDBM50169228; AKOS000165384; AKOS017276395; Phenyl-(4-propionyl-phenoxy)-acetic acid
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
3-{4-{2-Amino-6-[4-(4-propyl-benzoyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL538945; SCHEMBL2808154; BDBM50296702
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Activity |
EC50 ~ 50000 nM
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[8] | |||
Compound Name |
3-[4-[2-Amino-6-[4-(pyridin-2-ylmethyl)piperazin-1-yl]pyrimidin-4-yl]oxyphenyl]-2-methyl-2-phenoxypropanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL551928; SCHEMBL2806755
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Activity |
EC50 ~ 50000 nM
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[8] | |||
Compound Name |
(R)-2-(3-((3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)methyl)phenoxy)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL461571; SCHEMBL2902118; BDBM50244809
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
(2R)-2-[5-[[3-(4-Tert-butylphenyl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]-2-chlorophenoxy]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1946568; BDBM50362951
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
(R)-5-[2-(2-Chloro-4-trifluoromethoxy-phenoxy)-ethoxy]-2-isopropyl-2,3-dihydro-benzofuran-2-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL363006; SCHEMBL4422445; BDBM50171995
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Activity |
IC50 ~ 50000 nM
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[11] | |||
Compound Name |
(4-Isopropyl-phenyl)-(4-propionyl-2,6-dipropyl-phenylamino)-acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL187612; BDBM50169257
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
Plantagineoside A
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2159605; BDBM50394346
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Activity |
EC50 ~ 50000 nM
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[12] | |||
Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-chloro-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1946570; BDBM50362952
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
(2,6-Dimethyl-4-propionyl-phenoxy)-phenyl-acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL189950; BDBM50169229
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
(2R,3R,4S,5S,6R)-2-[(3R,5R)-1-(3,4-Dihydroxyphenyl)-5-hydroxy-7-(4-hydroxyphenyl)heptan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
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Investigative | Compound Info | ||
Synonyms |
CHEMBL458899; BDBM50394342; [(1R,3R)-1-(3,4-Dihydroxyphenethyl)-3-hydroxy-5-(4-hydroxyphenyl)pentyl]beta-D-glucopyranoside
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Activity |
EC50 ~ 50000 nM
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[12] | |||
Compound Name |
(2R,3R,4S,5S,6R)-2-[(3R,5R)-1,7-Bis(3,4-dihydroxyphenyl)-5-hydroxyheptan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
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Investigative | Compound Info | ||
Synonyms |
CHEMBL465800; BDBM50394341; [(1R,3R)-1-(3,4-Dihydroxyphenethyl)-3-hydroxy-5-(3,4-dihydroxyphenyl)pentyl]beta-D-glucopyranoside
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Activity |
EC50 ~ 50000 nM
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[12] | |||
Compound Name |
(2R)-2-[2-Chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1947143; BDBM50362953
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
(2R)-2-[4-Chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1947146; BDBM50362948
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
3-[4-[2-Amino-6-[4-(furan-2-carbonyl)piperazin-1-yl]pyrimidin-4-yl]oxyphenyl]-2-methyl-2-phenoxypropanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL559112
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Activity |
EC50 ~ 50000 nM
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[8] | |||
Compound Name |
(R)-2-Tert-Butyl-5-[2-(2-chloro-4-trifluoromethoxy-phenoxy)-ethoxy]-2,3-dihydro-benzofuran-2-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL191489; SCHEMBL4424683; BDBM50171998
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Activity |
IC50 ~ 50000 nM
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[11] | |||
Compound Name |
(S)-2-Ethyl-5-{3-[4-(2,2,2-trifluoro-ethoxy)-phenoxy]-propoxy}-2,3-dihydro-benzofuran-2-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL193459; BDBM50171990
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Activity |
IC50 ~ 50000 nM
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[11] | |||
Compound Name |
(2,6-Dichloro-4-propionyl-phenoxy)-phenyl-acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL366220; BDBM50169256
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
(2,6-Di-sec-butyl-4-propionyl-phenoxy)-phenyl-acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL371112; BDBM50169255
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
(5R)-5-[4-Chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1947147; SCHEMBL14261739; BDBM50362949
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Activity |
EC50 ~ 50000 nM
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[10] | |||
Compound Name |
2-(4-Isopropyl-phenyl)-3-(4-propionyl-2,6-dipropyl-phenyl)-propionic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL371832; BDBM50169241
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Activity |
IC50 ~ 50000 nM
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[9] | |||
Compound Name |
(2R,3R,4S,5S,6R)-2-[(3R,5R)-5-Hydroxy-1,7-bis(4-hydroxyphenyl)heptan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
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Investigative | Compound Info | ||
Synonyms |
CHEMBL516827; BDBM50394343; [(1R,3R)-1-(4-Hydroxyphenethyl)-3-hydroxy-5-(4-hydroxyphenyl)pentyl]beta-D-glucopyranoside
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Activity |
EC50 ~ 50000 nM
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[12] | |||
Compound Name |
(S)-5-[3-(2-Chloro-4-trifluoromethoxy-phenoxy)-propoxy]-2-isopropyl-2,3-dihydro-benzofuran-2-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL192791; BDBM50172005
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Activity |
IC50 ~ 50000 nM
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[11] | |||
Compound Name |
Plantagineoside C
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2159607; BDBM50394344
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Activity |
EC50 ~ 50000 nM
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[12] | |||
Compound Name |
3-[4-[2-Amino-6-[4-(2-methoxybenzoyl)piperazin-1-yl]pyrimidin-4-yl]oxyphenyl]-2-methyl-2-phenoxypropanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL554773; SCHEMBL2806770
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Activity |
EC50 ~ 50000 nM
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[8] | |||
Compound Name |
2-((4S,5S)-1-(4-((1-(2-Fluoro-5-methoxyphenyl)piperidin-4-yl)oxy)phenyl)-4-methyl-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-5-yl)acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL4105324; SCHEMBL15710748; BDBM50243976
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Activity |
EC50 ~ 50000 nM
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[13] | |||
Compound Name |
Phenylpropanoic acid derivative, 74
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Investigative | Compound Info | ||
Synonyms |
CHEMBL477690; SCHEMBL6385019; BDBM34035
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Activity |
IC50 ~ 50000 nM
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[14] | |||
Compound Name |
1-[4-[2-(Benzenesulfonamido)ethyl]phenyl]sulfonyl-3-(4-methylphenyl)thiourea
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Investigative | Compound Info | ||
Synonyms |
CHEMBL465132; BDBM50269537
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Activity |
IC50 = 50000 nM
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[15] | |||
Compound Name |
Chembl4284250
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Investigative | Compound Info | ||
Synonyms |
SCHEMBL2266225; BDBM50466689; 5-[[4-[(2R)-2-(5-ethylpyridin-2-yl)-2-hydroxyethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
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Activity |
IC50 = 50140 nM
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[16] | |||
Compound Name |
(S)-3-(4-(2-(5-Methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-p-tolylpiperazin-1-yl)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1090860; BDBM50315308
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Activity |
EC50 = 50220 nM
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[17] | |||
Compound Name |
(2E,4E,8Z)-N-(2-Methylpropyl)dodeca-2,4,8,10-tetraenamide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2011545; BDBM50379799
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Activity |
EC50 = 52300 nM
|
[18] | |||
Compound Name |
Phenylpropanoic acid derivative, 32
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL477940; SCHEMBL5727584; BDBM34022
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||||
Activity |
IC50 = 53000 nM
|
[14] | |||
Compound Name |
2-[4-[2-(4-Benzoylphenoxy)ethyl]phenoxy]-2-methylpropanoic acid
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2204687; BDBM50402001
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||||
Activity |
EC50 = 54600 nM
|
[19] | |||
Compound Name |
3-[4-[[[3-[[Benzoyl(ethyl)amino]methyl]benzoyl]-ethylamino]methyl]phenyl]propanoic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2403501; BDBM50492345
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|
||||
Activity |
IC50 = 56200 nM
|
[20] | |||
Compound Name |
Chembl4217589
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Investigative | Compound Info | ||
Synonyms |
BDBM50456438
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|
||||
Activity |
EC50 = 56710 nM
|
[21] | |||
Compound Name |
Chembl4172253
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
BDBM50286281
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|
||||
Activity |
EC50 = 56900 nM
|
[22] | |||
Compound Name |
Epipinoresinol
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
(+)-Epipinoresinol; epi-pinoresinol; Pinoresinol; UNII-6YKG9JJC1S; 6YKG9JJC1S; Q63408653; (+)-epi-pinoresinol; MLS002473314; CHEMBL487611; SCHEMBL10019016; HMS2196C10; BDBM50379794; ZINC12153081; SMR001397395
Click to Show/Hide
|
||||
Activity |
EC50 = 58600 nM
|
[18] | |||
Compound Name |
5-[[4-[Bis[2-[(4-methoxyphenyl)methoxy]ethyl]amino]phenyl]methylidene]-1,3-diazinane-2,4,6-trione
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3753560; BDBM50137104
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|
||||
Activity |
IC50 = 59100 nM
|
[23] | |||
Compound Name |
N-(1-Adamantyl)-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazole-5-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070234; BDBM50389765
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[2-(4-Methylsulfonyl-3-nitrophenyl)-4-phenyl-1,3-thiazol-5-yl]-piperidin-1-ylmethanone
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070232; BDBM50389763
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[2-(4-Methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazol-5-yl]-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070236; BDBM50389767
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
3,4-Dihydro-1H-isoquinolin-2-yl-[2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazol-5-yl]methanone
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070094; BDBM50389754
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[4-Methyl-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-piperidin-1-ylmethanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070235; BDBM50389766
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
(2-Methyl-2,3-dihydroindol-1-yl)-[2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazol-5-yl]methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070093; BDBM50389755
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
N-Benzyl-N-methyl-2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazole-5-carboxamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070096; BDBM50389752
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
N-[(2-Fluorophenyl)methyl]-N-methyl-2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazole-5-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070095; BDBM50389753
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
2-(4-Methylsulfonyl-3-nitrophenyl)-N-phenyl-N-propyl-1,3-thiazole-4-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070090; BDBM50389758
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
N-[(3-Fluorophenyl)methyl]-N-methyl-2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazole-5-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070238; BDBM50389751
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[4-Methyl-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-(4-methylpiperidin-1-yl)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070091; BDBM50389757
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
(4-Methylpiperidin-1-yl)-[2-(4-methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazol-5-yl]methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070097; BDBM50389760
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[2-(4-Methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-piperidin-1-ylmethanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070099; BDBM50389762
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[2-(4-Methylsulfonyl-3-nitrophenyl)-4-(trifluoromethyl)-1,3-thiazol-5-yl]-piperidin-1-ylmethanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070098; BDBM50389761
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[4-Methyl-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070092; BDBM50389756
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[4-Ethyl-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070237; BDBM50389768
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
[4-Ethyl-2-(4-methylsulfonyl-3-nitrophenyl)-1,3-thiazol-5-yl]-piperidin-1-ylmethanone
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2070233; BDBM50389764
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|
||||
Activity |
IC50 ~ 60000 nM
|
[24] | |||
Compound Name |
3-[4-[[[3-(Benzamidomethyl)benzoyl]amino]methyl]phenyl]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2403509; BDBM50492346
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|
||||
Activity |
IC50 = 62700 nM
|
[20] | |||
Compound Name |
{4-[4-(6-Isopropoxypyridin-3-yl)-5-(4-trifluoromethoxyphenyl)-oxazol-2-ylmethoxy]-2-methylphenoxy}acetic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL1080699; SCHEMBL2786407; BDBM50312476
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|
||||
Activity |
EC50 = 70000 nM
|
[25] | |||
Compound Name |
Phenylpropanoic acid derivative, 17k
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL593320; BDBM33295
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|
||||
Activity |
IC50 ~ 70000 nM
|
[26] | |||
Compound Name |
2-Methyl-2-[4-[3-(4-phenoxyphenoxy)propyl]phenoxy]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2204691; BDBM50401997
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|
||||
Activity |
EC50 = 75200 nM
|
[19] | |||
Compound Name |
5-[[4-[Bis(2-phenylmethoxyethyl)amino]phenyl]methylidene]-1,3-diazinane-2,4,6-trione
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3754461; BDBM50137107
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|
||||
Activity |
IC50 = 78400 nM
|
[23] | |||
Compound Name |
Chembl4286980
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|
Investigative | Compound Info | ||
Synonyms |
SCHEMBL6928620; BDBM50466692
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|
||||
Activity |
IC50 = 78450 nM
|
[16] | |||
Compound Name |
5-[[4-[2-[(4-Methoxyphenyl)methoxy]ethyl-(2-pyridin-2-yloxyethyl)amino]phenyl]methylidene]-1,3-diazinane-2,4,6-trione
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3753871; BDBM50137105
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|
||||
Activity |
IC50 = 84000 nM
|
[23] | |||
Compound Name |
Glycine, N-((5-((2-(4-chlorophenyl)-5-methyl-4-oxazolyl)methoxy)-2-fluorophenyl)methyl)-N-(methoxycarbonyl)-
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
BMS-711939; UNII-E2C4891M77; BMS 711939; E2C4891M77; SCHEMBL2742707; CHEMBL3828718; BDBM28802; BMS711939; Q27276778
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|
||||
Activity |
IC50 ~ 98400 nM
|
[27] | |||
Compound Name |
Chembl4237449
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|
Investigative | Compound Info | ||
Synonyms |
SCHEMBL21370574; BDBM50462439
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|
||||
Activity |
EC50 ~ 100000 nM
|
[28] | |||
Compound Name |
N-(4-(4-Trifluoromethylbenzyl)carbamoylphenyl)-3-((4R)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3601088; SCHEMBL16385852; BDBM50109262
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|
||||
Activity |
EC50 ~ 100000 nM
|
[29] | |||
Compound Name |
Bisphenol A diglycidyl ether
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
BADGE; 2,2-Bis(4-glycidyloxyphenyl)propane; Epoxide A; Epophen EL 5; Dian diglycidyl ether; Diglycidyl bisphenol A; epi-Rez 510; Diglycidyl bisphenol A ether; Bpdge; DGEBA; DGEBPA; Diglycidyl ether of bisphenol A; Diomethane diglycidyl ether; Dian-bis-glycidylether; 2,2-Bis(4'-glycidyloxyphenyl)propane; Epi-Rez 508; 2,2-Bis(p-glycidyloxyphenyl)propane; Oligomer 340; Diglycidyl diphenylolpropane ether; 4,4'-Isopropylidenediphenol diglycidyl ether; Bis(4-glycidyloxyphenyl)dimethylmethane; ERL-2774; EP 274; 2,2-Bis[4-(2,3-epoxypropoxy)phenyl]propane; D.E.R. 332; Diglycidyl ether of 4,4'-isopropylidenediphenol; UNII-F3XRM1NX4H; NSC 5022; 2,2-Bis(phenyl-4-glycidoxy)propane; 2,2-Bis(4-hydroxyphenyl)propane diglycidyl ether; 4,4'-Bis(2,3-epoxypropoxy)diphenyldimethylmethane; 2,2-Bis(p-(2,3-epoxypropoxy)phenyl)propane; 2,2-Bis(4-(2,3-epoxypropyloxy)phenyl)propane; MFCD00080480; F3XRM1NX4H; 2,2-Bis(4-hydroxyphenyl)propane, diglycidyl ether; 2,2-Bis(p-hydroxyphenyl)propane, diglycidyl ether; Propane, 2,2-bis(4-(2,3-epoxypropoxy)phenyl)-; 2,2-Bis[4-(glycidyloxy)phenyl]propane; BISPHENOLFDIGLYCIDYLETHER; CHEMBL258558; 2,2-Bis[p-(2,3-epoxypropoxy)phenyl]propane; 2,2-Bis(p-hydroxyphenyl)propane diglycidyl ether; Propane, 2,2-bis(p-(2,3-epoxypropoxy)phenyl)-; Propane, 2,2-bis[p-(2,3-epoxypropoxy)phenyl]-; 2,2-bis-(4-Glycidyloxyphenyl)propane; DSSTox_CID_4624; 2,2-bis(4-(2,3-epoxypropoxy)phenyl)propane; 2,2-Bis[4-(2,3-epoxypropyloxy)phenyl]propane; DSSTox_RID_77472; DSSTox_GSID_24624; Epotuf 37-140; CCRIS 1965; Dian-bis-glycidylether [Czech]; HSDB 331; 2,2-bis(4-(2,3-epoxypropoxy)phenyl)-propane; 2,2-Bis(p-(2,3-epoxypropoxy)phenyl)-Propane; 2,2-Bis[4-(2,3-epoxypropoxy)phenyl]-Propane; 2,2-Bis[p-(2,3-epoxypropoxy)phenyl]-Propane; SR-01000597404; EINECS 216-823-5; GY 6010; Bisphenol A, diglycidyl ether; hexyloxypropylamine; Propane, 2,2-bis (p-(2,3-epoxypropoxy)phenyl); 2, diglycidyl ether; BISPHENOL A DIGLYCIDYL ETHER RESIN; ACMC-209dwr; Spectrum5_001987; Bisphenol-A diglycidylether; 4,3-epoxypropoxy)benzene]; D.E.R.trade mark 332; 11391red; bisphenol-a diglycidyl ether; isphenol a, diglycidyl ether; SCHEMBL22121; BSPBio_001468; KBioGR_000188; KBioSS_000188; Bis(4-glycidyloxyphenyl)propane; diglycidyl ether of bisphenol-A; 2,3-epoxypropoxy)phenyl]propane; DTXSID6024624; NIOSH/SL1998000; BCBcMAP01_000157; CTK3J3495; KBio2_000188; KBio2_002756; KBio2_005324; KBio3_000375; KBio3_000376; NSC5022; 2,3-epoxypropyloxy)phenyl]propane; Bio1_000378; Bio1_000867; Bio1_001356; Bio2_000188; Bio2_000668; HMS1361J10; HMS1791J10; HMS1989J10; HMS3267P05; HMS3402J10; HMS3414L19; HMS3649C20; HMS3678L17; WLN: T3OTJ B1OR D- 2X; KS-00000UP7; NSC-5022; 2,2-bis(4-glycidyloxypheny)propane; Bisphenol A diglycidyl ether, tech.; Tox21_202141; Tox21_303315; 1642AH; ANW-22297; BDBM50241439; 2, 2-Bis(4-glycidyloxyphenyl)propane; 2, 2-Bis(p-glycidyloxyphenyl)propane; AKOS003609360; Bis(4-glycidyloxyphenyl)dimethyamethane; DB14083; MCULE-9203373672; 2, 2-Bis(4'-glycidyloxyphenyl)propane; 2,2-[Bis(4-glycidyloxyphenyl)]propane; 4,3-epoxypropoxy)diphenyldimethylmethane; IDI1_033938; NCGC00025114-02; NCGC00025114-03; NCGC00025114-04; NCGC00025114-05; NCGC00025114-06; NCGC00025114-07; NCGC00025114-08; NCGC00257039-01; NCGC00259690-01; AS-33346; FT-0609175; FT-0663368; SL19980000; ST50826240; 4, 4'-Isopropylidenediphenol diglycidyl ether; D.E.R.(TM) 332, used as embedding medium; Propane,2-bis[(p-2,3-epoxypropoxy)phenyl]-; Propane,2-bis[4-(2,3-epoxypropoxy)phenyl]-; Propane,2-bis[p-(2,3-epoxypropoxy)phenyl]-; 2,2-Bis[(p-2,3-epoxypropoxy)phenyl]-Propane; Bis[4-(2,3-epoxypropoxy)phenyl]-(2)-propane; C14348; p,p'-Dimethylmethylenediphenol diglycidyl ether; 4,4'-Isopropylidene diphenol, diglycidyl ether-; Bisphenol A diglycidyl ether, analytical standard; Diglycidyl ether of 4, 4'-isopropylidenediphenol; 2, 2-Bis(4-hydroxyphenyl)propane diglycidyl ether; 2, 2-Bis(p-hydroxyphenyl)propane diglycidyl ether; Q2080808; SR-01000597404-1; SR-01000597404-3; SR-01000597404-4; W-107909; BRD-A16694057-001-01-9
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Activity |
IC50 = 100000 nM
|
[30] | |||
Compound Name |
(S)-3-(3-Bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-phenylpiperazin-1-yl)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1090557; SCHEMBL4482985; BDBM50315310
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||||
Activity |
EC50 ~ 100000 nM
|
[17] | |||
Compound Name |
Phenylpropanoic acid derivative, 75
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL516129; SCHEMBL6384196; BDBM34036
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||||
Activity |
IC50 ~ 100000 nM
|
[14] | |||
Compound Name |
2-[3-[(4-Methylphenyl)carbamoyl]-4-piperidin-1-ylphenyl]indazole-6-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL3746821; SCHEMBL17317386; BDBM50500150
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|
||||
Activity |
EC50 ~ 100000 nM
|
[31] | |||
Compound Name |
N-[4-[4-[3-[1-[(4-Tert-butylphenyl)methyl]-4-ethyl-5-oxo-1,2,4-triazol-3-yl]propyl]phenyl]phenyl]-4-(4-methoxyphenyl)benzenesulfonamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3264936; BDBM50013725
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||||
Activity |
IC50 ~ 100000 nM
|
[32] | |||
Compound Name |
(Z)-5-(4-(3-(Piperidin-1-yl)propoxy)benzylidene)-2-thioxothiazolidin-4-one
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1081073; BDBM50313117
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||||
Activity |
EC50 ~ 100000 nM
|
[33] | |||
Compound Name |
(2R)-3,3,3-Trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]-2-hydroxypropanamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2323021; SCHEMBL3628001; HSD-621; BDBM50426478
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||||
Activity |
IC50 ~ 100000 nM
|
[34] | |||
Compound Name |
3-[[(4R)-4-Benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]-N-[4-(cyclohexylmethylcarbamoyl)phenyl]benzamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3601092; SCHEMBL16385917; BDBM50109196
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||||
Activity |
EC50 ~ 100000 nM
|
[29] | |||
Compound Name |
2-Ethyl-3-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]-5H-imidazo[4,5-c]pyridin-4-one
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2322177; BDBM50426775
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||||
Activity |
EC50 ~ 100000 nM
|
[35] | |||
Compound Name |
N-(4-Dodecylcarbamoylphenyl)-3-((4R)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3601090; SCHEMBL17744950; BDBM50109199; 3-[[(4R)-4-benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]-N-[4-(dodecylcarbamoyl)phenyl]benzamide
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||||
Activity |
EC50 ~ 100000 nM
|
[29] | |||
Compound Name |
N-(4-Benzylcarbamoylphenyl)-3-((4R)-2-oxo-4-benzyloxazolidine-3-yl)methylbenzamide
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|
Investigative | Compound Info | ||
Synonyms |
CHEMBL3600934; SCHEMBL16385824; BDBM50109159; N-[4-(benzylcarbamoyl)phenyl]-3-[[(4R)-4-benzyl-2-oxo-1,3-oxazolidin-3-yl]methyl]benzamide
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||||
Activity |
EC50 ~ 100000 nM
|
[29] | |||
Compound Name |
Chembl4240338
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|
Investigative | Compound Info | ||
Synonyms |
SCHEMBL21370444; BDBM50462437
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|
||||
Activity |
EC50 ~ 100000 nM
|
[28] | |||
Compound Name |
(2E,6E,10E)-2,6,10-Trimethyl-12-(3-methylfuran-2-yl)dodeca-2,6,10-trienoic acid
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Investigative | Compound Info | ||
Synonyms |
saurufuran B; CHEMBL494383; SaurufuranB; BDBM50260284
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||||
Activity |
EC50 ~ 100000 nM
|
[36] | |||
Compound Name |
Lithium;5-(3-carboxyphenyl)-2-[(2,4-dichlorobenzoyl)amino]benzoate
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Investigative | Compound Info | ||
Synonyms |
CHEMBL325172
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|
||||
Activity |
EC50 ~ 100000 nM
|
[37] | |||
Compound Name |
2-Methyl-5-[4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)butyl]-1,3-dioxane-2-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL401616; CHEMBL401712; SCHEMBL5856320; SCHEMBL5995415; BDBM50373021; BDBM50373027
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||||
Activity |
EC50 = 100000 nM
|
[38] | |||
Compound Name |
Phenylpropanoic acid derivative, 76
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL478563; SCHEMBL6388891; BDBM34037
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||||
Activity |
IC50 ~ 100000 nM
|
[14] | |||
Compound Name |
2-[2-Ethyl-4-oxo-3-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazo[4,5-c]pyridin-5-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2322440; BDBM50426771
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||||
Activity |
EC50 ~ 100000 nM
|
[35] | |||
Compound Name |
2-[2-Ethyl-4-oxo-3-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL2322438; BDBM50426773
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Activity |
EC50 ~ 100000 nM
|
[35] | |||
Compound Name |
2-[(1S)-5-{3-[2-Chloro-4-(4H-1,2,4-triazol-4-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220990; SCHEMBL1400260; Indanylacetic Acid Analog, 17w; BDBM21776; 2-[(1S)-5-[3-[2-chloro-4-(1,2,4-triazol-4-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Activity |
EC50 = 117489.76 nM
|
[39] | |||
Compound Name |
Dihydroformononetin
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
7-Hydroxy-4'-methoxyisoflavanone; CHEMBL3343011; SCHEMBL2069507; BDBM50102651; LMPK12050448; 7-hydroxy-3-(4-methoxyphenyl)-2,3-dihydrochromen-4-one
Click to Show/Hide
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||||
Activity |
IC50 = 124000 nM
|
[40] | |||
Compound Name |
2-[(1S)-5-[3-(3-Methylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220628; SCHEMBL1400621; Indanylacetic Acid Analog, 17i; BDBM21761
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Activity |
EC50 = 125892.54 nM
|
[39] | |||
Compound Name |
Mifobate
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
SR-202; SR 202; Clenicor; (4-Chlorophenyl)(dimethoxyphosphinyl)methyl phosphoric acid dimethyl ester; Phosphoric acid, (4-chlorophenyl)(dimethoxyphosphinyl)methyl dimethyl ester; CHEMBL284768; NCGC00092299-01; (4-chlorophenyl)(dimethoxyphosphoryl)methyl dimethyl phosphate; DSSTox_CID_25741; DSSTox_RID_81086; DSSTox_GSID_45741; Mifobatum [Latin]; Mifobato [Spanish]; Mifobato; Mifobatum; Mifobate [USAN:INN]; C11H17ClO7P2; BRN 5985350; Clenicor (TN); CLANICLOR; Dimethyl alpha-(dimethoxyphosphinyl)-p-chlorobenzyl phosphate; Mifobate (USAN/INN); Dimethyl (p-chloro-alpha-hydroxybenzyl)phosphonate, dimethyl phosphate; MLS004712055; SCHEMBL635294; DTXSID6045741; CTK8G3195; HMS3268H09; HMS3413C19; HMS3677C19; [(4-chlorophenyl)-dimethoxyphosphorylmethyl] dimethyl phosphate; Tox21_111190; BDBM50240444; MFCD00864813; AKOS005067403; Tox21_111190_1; NCGC00092299-02; SMR002530311; DB-056081; HY-100277; SR-202, >=98% (HPLC), crystalline; CS-0018429; FT-0630844; V4185; D05030; BRD-A72066420-001-01-1; Q27163636; Dimethyl (alpha-dimethoxyphosphinyl-p-chlorobenzyl) phosphate; Dimethyl .alpha.-(dimethoxyphosphinyl)-p-chlorobenzyl phosphate; (4-CHLOROPHENYL)(DIMETHOXYPHOSPHINYL)METHYLPHOSPHORICACIDDIMETHYLESTER; Dimethyl (p-chloro-.alpha.-hydroxybenzyl)phosphonate, dimethyl phosphate
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Activity |
IC50 = 140000 nM
|
[30] | |||
Compound Name |
2-[(1S)-5-[3-(4-Ethylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220421; SCHEMBL1400619; Indanylacetic Acid Analog, 17b; BDBM21754
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Activity |
EC50 = 162181.01 nM
|
[39] | |||
Compound Name |
(3R,4S)-4-[[4-[2-(5-Methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL255930; SCHEMBL12616772; BDBM50377302
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||||
Activity |
EC50 = 165000 nM
|
[41] | |||
Compound Name |
2-[(1S)-5-[3-[4-(Trifluoromethyl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(trifluoromethyl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220422; SCHEMBL1400241; Indanylacetic Acid Analog, 17c; BDBM21755
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||||
Activity |
EC50 = 181970.09 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-{3-[2-Acetamido-4-(1H-1,2,3-triazol-1-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219817; Indanylacetic Acid Analog, 17v; BDBM21775
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Activity |
EC50 = 181970.09 nM
|
[39] | |||
Compound Name |
5-[[4-[2-[(4-Methoxyphenyl)methoxy]ethyl-(2-phenylmethoxyethyl)amino]phenyl]methylidene]-1,3-diazinane-2,4,6-trione
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Investigative | Compound Info | ||
Synonyms |
CHEMBL3753308; BDBM50137096
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||||
Activity |
IC50 = 191000 nM
|
[23] | |||
Click to Show/Hide the Information of All Poor Binders |
Non Binders of This Target (in total, 87 non binders) | Download | Top | |||
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Compound Name |
Fenofibrate
Click to Show/Hide
|
Approved | Compound Info | ||
Synonyms |
Ankebin; Antara; Controlip; Durafenat; Elasterate; Elasterin; FNF; Fenobeta; Fenobrate; Fenofanton; Fenofibrato; Fenofibratum; Fenogal; Fenoglide; Fenomax; Fenotard; Finofibrate; Fulcro; Lipanthyl; Lipantil; Liparison; Lipidex; Lipidil; Lipifen; Lipirex; Lipoclar; Lipofen; Lipofene; Liposit; Lipsin; Lofibra; Luxacor; Nolipax; Pharmavit; Phenofibrate; Procetofen; Procetofene; Proctofene; Protolipan; Secalip; Sedufen; Supralip; Tricor; Triglide; AbZ Brand of Procetofen; Abbott Brand of Procetofen; Aliud Brand of Procetofen; Antara Micronized Procetofen; Anto Brand of Procetofen; Apo Feno Micro; Apo Fenofibrate; Apotex Brand of Procetofen; Azupharma Brand of Procetofen; Betapharm Brand of Procetofen; Bouchara Brand of Procetofen; Ct Arzneimittel Brand of Procetofen; Fenofibrat AL; Fenofibrat AZU; Fenofibrat AbZ; Fenofibrat FPh; Fenofibrat Heumann; Fenofibrat Hexal; Fenofibrat Stada; Fenofibrat ratiopharm; Fenofibrat von ct; Fenofibrate Debat; Fenofibrate MSD; Fournier Brand of Procetofen; GNR Pharma Brand of Procetofen; Gate Brand of Procetofen; Gen Fenofibrate; Genpharm Brand of Procetofen; Heumann Brand of Procetofen; Hexal Brand of Procetofen; Knoll Brand of Procetofen; Lichtenstein Brand of Procetofen; Lipidil Micro; Lipidil Supra; Lipidil Ter; MTW Brand of Procetofen; MTW Fenofibrat; Merck dura Brand of Procetofen; Novartis Brand of Procetofen; Novo Fenofibrate; Novopharm Brand of Procetofen; Nu Fenofibrate; Nu Pharm Brand of Procetofen; PMS Fenofibrate Micro;Pharmascience Brand of Procetofen; Procetofen Reliant Brand; Q Pharm Brand of Procetofen; Ratiopharm Brand of Procetofen; Reliant Brand of Procetofen; Schering Plough Brand of Procetofen; Stadapharm Brand of Procetofen; United Drug Brand of Procetofen; F 6020; LF 178; LF178; AZU, Fenofibrat; Antara (TN); Antara (micronized); Apo-Fenofibrate; CIP-Fenofibrate; Ct-Arzneimittel Brand of Procetofen; Debat, Fenofibrate; FENOFIBRATE (MICRONIZED); Fenofibrat-ratiopharm; Fenofibrate IDD-P; Fenofibrate [INN:BAN]; Fenofibrato [INN-Spanish]; Fenofibratum [INN-Latin]; Fenogal (TN); GNR-Pharma Brand of Procetofen; GRS-027; Gen-Fenofibrate; Heumann, Fenofibrat; Hexal, Fenofibrat; LCP-Feno; LCP-FenoChol; LF-178; Lipanthyl (TN); Lipantil (TN); Lipidil (TN); Lipidil-Ter; Lipofen (TN); Lofibra (TN); MTW-Fenofibrat; Micronized Procetofen, Antara; Novo-Fenofibrate; Nu-Fenofibrate; Nu-Pharm Brand of Procetofen; PMS-Fenofibrate Micro; Procetofen, Antara Micronized; Q-Pharm Brand of Procetofen; Schering-Plough Brand of Procetofen; Stada, Fenofibrat; TRICOR (MICRONIZED); Tricor (TN); Triglide (TN); Trilipix (TN); Apo-Feno-Micro; Fenocor-67 (TN); Fenofibrate (JAN/INN); Isopropyl 2-[4-(4-chlorobenzoyl)phenoxy]-2-methylpropanoate; Isopropyl 2-(4-(4-chlorobenzoyl)phenoxy)-2-methylpropionate; Isopropyl 2-(p-(p-chlorobenzoyl)phenoxy)-2-methylpropionate
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|
||||
Activity |
EC50 = 300000 nM
|
[42] | |||
Compound Name |
Clofibrate
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Approved | Compound Info | ||
Synonyms |
Amotril; Angiokapsul; Anparton; Antilipid; Antilipide; Apolan; Arterioflexin; Arterosol; Artevil; Ateculon; Ateriosan; Athebrate; Atheromide; Atheropront; Athromidin; Atrolen; Atromid; Atromida; Atromidin; Atrovis; Azionyl; Bioscleran; Bresit; CPIB; Cartagyl; Chlorfenisate; Chlorphenisate; Cinnarizin; Citiflus; Claripex; Cloberat; Clobrat; Clofar; Clofibate; Clofibram; Clofibrat; Clofibrato; Clofibratum; Clofinit; Clofipront; Delipid; Deliva; ELPI; EPIB; Fibralem; Gerastop; Hyclorate; Klofibrat; Klofiran; Levatrom; Lipamid; Lipavil; Lipavlon; Lipidsenker; Lipofacton; Lipomid; Liponorm; Liporeduct; Liporil; Liposid; Liprin; Liprinal; Lobetrin; Miscleron; Misclerone; Miskleron; Negalip; Normalip; Normat; Normet; Normolipol; Novofibrate; Persantinat; Recolip; Regardin; Regelan; Robigram; Scrobin; Serofinex; Serotinex; Skerolip; Sklerepmexe; Sklero; Sklerolip; Skleromex; Skleromexe; Ticlobran; Xyduril; Yoclo; Amotril S; Atromid S; Claripex CPIB; Clofibrato [Spanish]; Dura clofibrat; Ethyl chlorophenoxyisobutyrate; Ethyl clofibrate; Regelan N; Vincamin compositum; AY 61123; C 6643; Lipide 500; Oxan 600; AY-61123; Athranid-wirkstoff; Atromid-S; BML2-F02; Chlorophenoxyisobutyrate, Ethyl; Clobren-5F; Clobren-SF; Clofibrate (CLOF); Clofibrato [INN-Spanish]; Clofibratum [INN-Latin]; Clofibric Acid, Ethyl Ester; Ethyl p-chlorophenoxyisobutyrate; Ethyl para-chlorophenoxyisobutyrate; Neo-Atomid; Neo-Atromid; Sklero-Tablinen; Sklero-tablinene; Sklero-tabuls; ATROMID-S (TN); Atromid-S (TN); Atromid-S, Clofibrate; Ethyl alpha-p-chlorophenoxyisobutyrate; Clofibrate (JP15/USP/INN); Clofibrate [USAN:INN:BAN:JAN]; Ethyl 2-(4-chlorophenoxy)isobutyrate; Ethyl 2-(p-chlorophenoxy)isobutyrate; Ethyl alpha-(4-chlorophenoxy)isobutyrate; Ethyl alpha-(p-chlorophenoxy)isobutyrate; Ethyl-alpha-p-chlorophenoxy-isobutyrate
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Activity |
EC50 ~ 500000 nM
|
[42] | |||
Compound Name |
Fibrates
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Investigative | Compound Info | ||
Synonyms |
clofibric acid; 882-09-7; 2-(4-Chlorophenoxy)-2-methylpropanoic acid; Chlorofibrinic acid; Clofibrinic acid; Chlorfibrinic acid; Clofibrin; 2-(4-CHLOROPHENOXY)-2-METHYLPROPIONIC ACID; Chlorophibrinic acid; PCIB; Clofibrate free acid; Clofibrinsaeure; Regulipid; Regadrin; PCPIB; 2-(p-Chlorophenoxy)-2-methylpropionic acid; 2-(4-Chlorophenoxy)isobutyric Acid; 4-CPIB; 2-(p-Chlorophenoxy)isobutyric acid; Propanoic acid, 2-(4-chlorophenoxy)-2-methyl-; alpha-(p-Chlorophenoxy)isobutyric acid; Acido clofibrico; Acide clofibrique; Acidum c
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Activity |
EC50 > 300000 nM
|
[43] | |||
Compound Name |
GW1929
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Investigative | Compound Info | ||
Synonyms |
GW 1929; GW-1929
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Activity |
Ki = 113240036.3 nM
|
[44] | |||
Compound Name |
2-[N-(2-Phenylmethoxyethyl)-4-[(2,4,6-trioxo-1,3-diazinan-5-ylidene)methyl]anilino]ethyl acetate
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL3754373; BDBM50137106
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Activity |
IC50 > 200000 nM
|
[23] | |||
Compound Name |
3-(2,3,10,11-Tetramethoxy-1,4-dihydroisoquinolino[2,1-b]isoquinolin-7-ium-8-yl)propanoic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1783069; BDBM50346517; 8-(2-Carboxy-ethyl)-2,3,10,11-tetramethoxy-1,4-dihydro-isoquino[3,2-a]isoquinolinylium
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Activity |
EC50 = 220000 nM
|
[45] | |||
Compound Name |
Chembl4171403
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Investigative | Compound Info | ||
Synonyms |
BDBM50286278
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Activity |
EC50 = 236400 nM
|
[22] | |||
Compound Name |
2-[(1S)-5-[3-[4-(Furan-3-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(furan-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL376418; SCHEMBL1400869; Indanylacetic Acid Analog, 29b; BDBM21779
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Activity |
EC50 = 245470.89 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-Methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220627; SCHEMBL1400338; Indanylacetic Acid Analog, 17e; BDBM21757
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Activity |
EC50 = 338844.16 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2,4-Dimethylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220785; SCHEMBL3019471; Indanylacetic Acid Analog, 17l; BDBM21765
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Activity |
EC50 = 467735.14 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{4-[5-(Trifluoromethyl)pyridin-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220570; SCHEMBL1400566; Indanylacetic Acid Analog, 29i; BDBM21785
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Activity |
EC50 = 562341.33 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2-Methoxy-4-methylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220060; SCHEMBL1400278; Indanylacetic Acid Analog, 17q; BDBM21770
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Activity |
EC50 = 602559.59 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-Ethyl-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220681; SCHEMBL1400818; Indanylacetic Acid Analog, 17r; BDBM21771
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Activity |
EC50 = 616595 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2-Propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL375098; SCHEMBL3019309; Indanylacetic Acid Analog, 17m; BDBM21766
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Activity |
EC50 = 660693.45 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2-Ethoxy-4-methylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220430; SCHEMBL1400329; Indanylacetic Acid Analog, 17t; BDBM21773
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Activity |
EC50 = 812830.52 nM
|
[39] | |||
Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-methoxyphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL427080; SCHEMBL1400614; BDBM21813; Indanylacetic Acid Analog, 34ab
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Activity |
EC50 = 1000000 nM
|
[39] | |||
Compound Name |
1-[4-[2-(Benzenesulfonamido)ethyl]phenyl]sulfonyl-3-(4-methoxyphenyl)thiourea
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Investigative | Compound Info | ||
Synonyms |
CHEMBL465746; BDBM50269538
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|
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Activity |
IC50 = 1000000 nM
|
[15] | |||
Compound Name |
2-[(1S)-5-[3-[4-(Trifluoromethoxy)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(trifluoromethoxy)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL373605; SCHEMBL1400262; Indanylacetic Acid Analog, 17d; BDBM21756
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Activity |
EC50 = 1000000 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220059; SCHEMBL1400323; Indanylacetic Acid Analog, 34c; BDBM21788
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Activity |
EC50 = 1047128.55 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-{3-[4-(Pyrimidin-5-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220448; SCHEMBL1400268; Indanylacetic Acid Analog, 29f; BDBM21763; 2-[(1S)-5-[3-(4-pyrimidin-5-ylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Activity |
EC50 = 1047128.55 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-Ethoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL220507; SCHEMBL1400700; Indanylacetic Acid Analog, 17f; BDBM21758
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Activity |
EC50 = 1071519.31 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(4-ethyl-1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220635; SCHEMBL1400693; Indanylacetic Acid Analog, 34d; BDBM21789
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Activity |
EC50 = 1148153.62 nM
|
[39] | |||
Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1h-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-(hydroxymethyl)-1,3-thiazole-5-carboxylic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL424933; SCHEMBL1400982; BDBM21814; Indanylacetic Acid Analog, 34ac
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Activity |
EC50 = 1148153.62 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL223748; SCHEMBL1400573; BDBM21818; Indanylacetic Acid Analog, 34ag
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Activity |
EC50 = 1348962.88 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(1H-Indol-6-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
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Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(1H-indol-6-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220893; SCHEMBL1400787; Indanylacetic Acid Analog, 29c; BDBM21780
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Activity |
EC50 = 1380384.26 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-Cyano-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL375747; SCHEMBL1400667; Indanylacetic Acid Analog, 17s; BDBM21772
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Activity |
EC50 = 1445439.77 nM
|
[39] | |||
Compound Name |
3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL1209170; SCHEMBL4283477; BDBM50323530
Click to Show/Hide
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||||
Activity |
EC50 = 1450000 nM
|
[46] | |||
Compound Name |
2-[(1S)-5-{3-[4-(Thiophen-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL375748; SCHEMBL1400569; Indanylacetic Acid Analog, 29a; BDBM21778
Click to Show/Hide
|
||||
Activity |
EC50 = 1548816.62 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-Cyano-2-propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219661; SCHEMBL1400255; Indanylacetic Acid Analog, 17o; BDBM21768
Click to Show/Hide
|
||||
Activity |
EC50 = 1778279.41 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-{3-[4-(Pyridin-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219944; SCHEMBL1400495; Indanylacetic Acid Analog, 29d; BDBM21781; 2-[(1S)-5-[3-(4-pyridin-3-ylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
||||
Activity |
EC50 = 1819700.86 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-{3-[4-(6-Methylpyridin-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220325; SCHEMBL1400382; Indanylacetic Acid Analog, 29h; BDBM21784
Click to Show/Hide
|
||||
Activity |
EC50 = 1819700.86 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-{3-[4-(1H-1,2,4-Triazol-1-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220431; Indanylacetic Acid Analog, 17u; BDBM21774
Click to Show/Hide
|
||||
Activity |
EC50 = 1819700.86 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Methoxypyridin-3-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(4-methoxypyridin-3-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220388; SCHEMBL1400769; Indanylacetic Acid Analog, 29e; BDBM21782
Click to Show/Hide
|
||||
Activity |
EC50 = 2089296.13 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL374545; SCHEMBL1400856; Indanylacetic Acid Analog, 34u; BDBM21806
Click to Show/Hide
|
||||
Activity |
EC50 = 2089296.13 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[2-methoxy-4-(1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220124; SCHEMBL1400868; Indanylacetic Acid Analog, 34b; BDBM21787
Click to Show/Hide
|
||||
Activity |
EC50 = 2691534.8 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{2-Methoxy-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219687; SCHEMBL1400842; Indanylacetic Acid Analog, 34i; BDBM21794
Click to Show/Hide
|
||||
Activity |
EC50 = 3090295.43 nM
|
[39] | |||
Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)phenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL374682; SCHEMBL1400652; Indanylacetic Acid Analog, 34z; BDBM21811
Click to Show/Hide
|
||||
Activity |
EC50 = 3235936.57 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(trifluoromethyl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[2-propyl-4-(trifluoromethyl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL219686; SCHEMBL1400334; Indanylacetic Acid Analog, 17n; BDBM21767
Click to Show/Hide
|
||||
Activity |
EC50 = 3311311.21 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(2,4-Dimethoxypyrimidin-5-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(2,4-dimethoxypyrimidin-5-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL425116; SCHEMBL1400636; Indanylacetic Acid Analog, 29g; BDBM21783
Click to Show/Hide
|
||||
Activity |
EC50 = 3388441.56 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Methoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic Acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[4-(4-methoxy-1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL220224; SCHEMBL1400374; BDBM21816; Indanylacetic Acid Analog, 34ae
Click to Show/Hide
|
||||
Activity |
EC50 = 3388441.56 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4,5,6,7-Tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL375812; SCHEMBL1400287; Indanylacetic Acid Analog, 34o; BDBM21800
Click to Show/Hide
|
||||
Activity |
EC50 = 3467368.5 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220837; SCHEMBL1400266; Indanylacetic Acid Analog, 34j; BDBM21795
Click to Show/Hide
|
||||
Activity |
EC50 = 3630780.55 nM
|
[39] | |||
Compound Name |
2-[4-(3-{[(1S)-1-(Carboxymethyl)-2,3-dihydro-1H-inden-5-yl]oxy}propoxy)-3-propylphenyl]-4-methyl-1,3-thiazole-5-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL222247; SCHEMBL1400267; BDBM21812; Indanylacetic Acid Analog, 34aa
Click to Show/Hide
|
||||
Activity |
EC50 = 4265795.19 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(1,3-Benzothiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL424939; SCHEMBL1400421; Indanylacetic Acid Analog, 34t; BDBM21805
Click to Show/Hide
|
||||
Activity |
EC50 = 4677351.41 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219609; SCHEMBL1400824; BDBM21825; Indanylacetic Acid Analog, 34an
Click to Show/Hide
|
||||
Activity |
EC50 = 5623413.25 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2-Methoxy-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL375427; Indanylacetic Acid Analog, 34s; BDBM21804
Click to Show/Hide
|
||||
Activity |
EC50 = 5623413.25 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220152; SCHEMBL1400686; BDBM21824; Indanylacetic Acid Analog, 34am
Click to Show/Hide
|
||||
Activity |
EC50 = 5754399.37 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{2-Methyl-4-[3-(trifluoromethyl)-1,2,4-thiadiazol-5-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219688; SCHEMBL1400498; Indanylacetic Acid Analog, 17x; BDBM21777
Click to Show/Hide
|
||||
Activity |
EC50 = 6456542.29 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}-2-methoxyphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL222248; SCHEMBL1400371; Indanylacetic Acid Analog, 34n; BDBM21799
Click to Show/Hide
|
||||
Activity |
EC50 = 8709635.9 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(4-{4H,5H,6H-Cyclopenta[d][1,3]thiazol-2-yl}-2-propylphenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220223; SCHEMBL3117156; Indanylacetic Acid Analog, 34m; BDBM21798
Click to Show/Hide
|
||||
Activity |
EC50 = 10715193.05 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219617; SCHEMBL1400681; Indanylacetic Acid Analog, 34q; BDBM21802
Click to Show/Hide
|
||||
Activity |
EC50 = 12022644.35 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Methoxy-4-(4-methoxy-1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL222508; SCHEMBL1400402; BDBM21817; Indanylacetic Acid Analog, 34af
Click to Show/Hide
|
||||
Activity |
EC50 = 14791083.88 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220557; SCHEMBL1400349; Indanylacetic Acid Analog, 34f; BDBM21791
Click to Show/Hide
|
||||
Activity |
EC50 = 15488166.19 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{2-Propyl-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL374090; SCHEMBL1400786; Indanylacetic Acid Analog, 34h; BDBM21793
Click to Show/Hide
|
||||
Activity |
EC50 = 18197008.59 nM
|
[39] | |||
Compound Name |
Methyl 2-(5-(2-(2-(biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetate
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL1784949; BDBM50345808
Click to Show/Hide
|
||||
Activity |
EC50 = 20000000 nM
|
[47] | |||
Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220151; SCHEMBL1400676; Indanylacetic Acid Analog, 34w; BDBM21808
Click to Show/Hide
|
||||
Activity |
EC50 = 20417379.45 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(1,3-thiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
2-[(1S)-5-{3-[2-propyl-4-(1,3-thiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid; CHEMBL374901; SCHEMBL1400247; Indanylacetic Acid Analog, 34a; BDBM21786
Click to Show/Hide
|
||||
Activity |
EC50 = 20892961.31 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{4-[4-(Propan-2-yloxy)-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL436514; SCHEMBL1400496; BDBM21821; Indanylacetic Acid Analog, 34aj
Click to Show/Hide
|
||||
Activity |
EC50 = 22387211.39 nM
|
[39] | |||
Compound Name |
((1S)-5-{3-[4-(4-Ethyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl)acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL373813; SCHEMBL3023128; Indanylacetic Acid Analog, 34e; BDBM21790
Click to Show/Hide
|
||||
Activity |
EC50 = 22387211.39 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-(3-{2-Methoxy-4-[4-(propan-2-yloxy)-1,3-thiazol-2-yl]phenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219669; SCHEMBL1400978; BDBM21822; Indanylacetic Acid Analog, 34ak
Click to Show/Hide
|
||||
Activity |
EC50 = 22908676.53 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-(2-Propyl-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
SCHEMBL1400218; CHEMBL2236890; Indanylacetic Acid Analog, 34r; BDBM21803
Click to Show/Hide
|
||||
Activity |
EC50 = 23988329.19 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL387350; SCHEMBL1400331; BDBM21819; Indanylacetic Acid Analog, 34ah
Click to Show/Hide
|
||||
Activity |
EC50 = 24547089.16 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Ethoxy-5-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL373791; SCHEMBL1400704; BDBM21823; Indanylacetic Acid Analog, 34al
Click to Show/Hide
|
||||
Activity |
EC50 = 29512092.27 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4,5-Dimethyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL374925; SCHEMBL1400962; Indanylacetic Acid Analog, 34k; BDBM21796
Click to Show/Hide
|
||||
Activity |
EC50 = 30902954.33 nM
|
[39] | |||
Compound Name |
2-(5-(2-(2-(Biphenyl-4-yl)-5-methyloxazol-4-yl)ethoxy)-1-(4-chlorobenzoyl)-2-methyl-1H-indol-3-yl)acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL1784948; BDBM50345807
Click to Show/Hide
|
||||
Activity |
EC50 = 40000000 nM
|
[47] | |||
Compound Name |
2-[(1S)-5-(3-{4-[5-(Dimethylcarbamoyl)-4-methyl-1,3-thiazol-2-yl]-2-propylphenoxy}propoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220662; SCHEMBL1400162; Indanylacetic Acid Analog, 34x; BDBM21809
Click to Show/Hide
|
||||
Activity |
EC50 = 50118723.36 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(4-Tert-butyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL220117; SCHEMBL1400351; Indanylacetic Acid Analog, 34g; BDBM21792
Click to Show/Hide
|
||||
Activity |
EC50 = 56234132.52 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)-2-propylphenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL219668; SCHEMBL1400300; Indanylacetic Acid Analog, 34v; BDBM21807
Click to Show/Hide
|
||||
Activity |
EC50 = 58884365.54 nM
|
[39] | |||
Compound Name |
2-[(1S)-5-[3-[2-Propyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
SCHEMBL1400467; CHEMBL2113263; Indanylacetic Acid Analog, 34p; BDBM21801
Click to Show/Hide
|
||||
Activity |
EC50 = 85113803.82 nM
|
[39] | |||
Compound Name |
(S)-3-[4-[2-[Methyl(benzoxazol-2-yl)amino]ethoxy]phenyl]-2-[(2-benzoylphenyl)amino]propionic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL423026; SCHEMBL7914542; BDBM50418564; (2S)-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylanilino)propanoic acid
Click to Show/Hide
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||||
Activity |
Ki = 112201845.4 nM
|
[44] | |||
Compound Name |
3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[2-(2-phenylacetyl)anilino]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL146822; BDBM50418568
Click to Show/Hide
|
||||
Activity |
Ki = 118032063.6 nM
|
[44] | |||
Compound Name |
(2S)-3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-phenoxyanilino)propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL1785077; BDBM50418576
Click to Show/Hide
|
||||
Activity |
Ki = 118850222.7 nM
|
[44] | |||
Compound Name |
3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9,10-dioxoanthracen-1-yl)amino]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL358137; BDBM50418575
Click to Show/Hide
|
||||
Activity |
Ki = 120781383.5 nM
|
[44] | |||
Compound Name |
(2S)-2-(2-Benzoylanilino)-3-[4-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]phenyl]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL148301; BDBM50418563
Click to Show/Hide
|
||||
Activity |
Ki = 120781383.5 nM
|
[44] | |||
Compound Name |
(2S)-2-(2-Benzoylanilino)-3-[4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl]propanoic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
Synonyms |
CHEMBL346219; BDBM50418571
Click to Show/Hide
|
||||
Activity |
Ki = 122179966 nM
|
[44] | |||
Compound Name |
3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenyl)sulfanylpropanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL146322; BDBM50418566
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Activity |
Ki = 132129563.4 nM
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[44] | |||
Compound Name |
2-[[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]methyl]-3-(2-benzoylphenyl)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1785075; BDBM50418565
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Activity |
Ki = 132739445.8 nM
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[44] | |||
Compound Name |
3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenoxy)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL147694; BDBM50418573
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Activity |
Ki = 133659551.7 nM
|
[44] | |||
Compound Name |
(2S)-2-(2-Benzoylanilino)-3-[4-[(1-methylcyclohexyl)methoxy]phenyl]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL357479; BDBM50418562
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Activity |
Ki = 137404197.5 nM
|
[44] | |||
Compound Name |
3-[4-[2-[1,3-Benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9-oxofluoren-1-yl)amino]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL148060; BDBM50418567
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Activity |
Ki = 141579378 nM
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[44] | |||
Compound Name |
(2S)-2-[(2-Benzoylcyclohexen-1-yl)amino]-3-(4-phenylmethoxyphenyl)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1785031; CHEMBL346415; SCHEMBL9994772; BDBM50418560
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Activity |
Ki = 147570653.3 nM
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[44] | |||
Compound Name |
2-[2-(Benzenesulfonyl)anilino]-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL146123; BDBM50418574
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||||
Activity |
Ki = 147570653.3 nM
|
[44] | |||
Compound Name |
(2S)-2-(2-Benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL359377; BDBM50418572
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||||
Activity |
Ki = 164058977.3 nM
|
[44] | |||
Compound Name |
(2S)-2-(4-Benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid
Click to Show/Hide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL147042; BDBM50418561
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||||
Activity |
Ki = 169824365.3 nM
|
[44] | |||
Compound Name |
Methyl 2-(1-(4-chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetate
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1784945; BDBM50345806
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Activity |
EC50 = 620000000 nM
|
[47] | |||
Compound Name |
2-(1-(4-Chlorobenzoyl)-2-methyl-5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-1H-indol-3-yl)acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1784944; BDBM50345805
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||||
Activity |
EC50 = 1230000000 nM
|
[47] | |||
Compound Name |
2-(4-(Benzyloxy)-2-(2,6-dichlorophenylamino)phenyl)acetic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL1784954; BDBM50345809
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Activity |
EC50 = 6030000000 nM
|
[47] | |||
Click to Show/Hide the Information of All Non Binders |
References | Top | ||||
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