Target Poor or Non Binder(s) Information

Target General Information

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Target ID

T52067

Target Info

Target Name

Solute carrier family 15 member 2 (SLC15A2)

Synonyms

Peptide transporter 2; PEPT2; Oligopeptide transporter, kidney isoform; Kidney H(+)/peptide cotransporter

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Target Type

Literature-reported Target

Gene Name

SLC15A2

UniProt ID

Q16348

Poor Binders of This Target (in total, 10 binders)

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Compound Name

Cefadroxil

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Approved

Compound Info

Synonyms

CDX; Cefadroxilo; Cefadroxilum; Cephadroxil; Sumacef; Cefadroxil anhydrous; S 578; BL-S 578; BL-S578; Cefadroxil (JP15); Cefadroxilo [INN-Spanish]; Cefadroxilum [INN-Latin]; Curisafe (TN); D-Cefadroxil; S-578; Sumacef (TN); MJF-11567-3; (6R,7R)-7-((R)-2-Amino-2-(p-hydroxyphenyl)acetamido)-3-methyl-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3,4-didehydrocepham-4-carboxylic acid

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Activity

IC50 = 66000 nM

[1]

Compound Name

Cephalexin

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Approved

Compound Info

Synonyms

Adcadina; Ades[prex; Alcephin; Alexin; Alsporin; Ambal; Aristosporin; Azabort; Bactopenor; Beliam; Biocef; CEX; Carnosporin; Cefablan; Cefacet; Cefadal; Cefadin; Cefadina; Cefalekey; Cefaleksin; Cefalessina; Cefalexgobens; Cefalexin; Cefalexina; Cefalexine; Cefalexinum; Cefalin; Cefalival; Cefaloto; Cefaseptin; Cefax; Ceffanex; Cefibacter; Ceflax; Ceforal; Cefovit; Celexin; Cepastar; Cepexin; Cephacillin; Cephalexine; Cephalexinum; Cephalobene; Cephanasten; Cephaxin; Cephin; Cepol; Ceporex; Ceporexin; Ceporexine; Check; Cophalexin; Domucef; Doriman; Durantel; Efemida; Erocetin; Factagard; Felexin; Fexin; Ibilex; Ibrexin; Inphalex; Karilexina; Kefalospes; Keflet; Keflex; Kefolan; Keforal; Keftab; Kekrinal; Kidolex; Lafarine; Larixin; Lenocef; Lexibiotico; Loisine; Lonflex; Lopilexin; Losporal; Madlexin; Maksipor; Mamalexin; Mamlexin; Medolexin; Medoxine; Neokef; Neolexina; Noveol; Novolexin; Nufex; Oracef; Oriphex; Oroxin; Ortisporina; Ospexin; Palitrex; Pectril; Prindex; Pyassan; Rilexine; Roceph; Rogevil; Sanaxin; Sartosona; Sencephalin; Sepexin; Servicef; Servispor; Sialexin; Sinthecillin; Sintolexyn; Sporicef; Sporidex; Syncl; Syncle; Synecl; Tepaxin; Theratrex; Tokiolexin; Uphalexin; Viosporine; Voxxim; Winlex; Zabytrex; Zozarine; Cefalessina [DCIT]; Cefalexin Scand Pharm; Cefalexin Sodium; Cefalexin generics; Cefalexin hydrate; Cefalexin monohydrate; Cefalexina Northia; Cefalexina Richet; Cephalex von ct; Cephalexin hydrate; Cephalexin monohydrate; Ceporex Forte; Durantel DS; Henina Oral; Panixine Disperdose; Roceph Distab; Lilly 66873; S 6437; SQ 20248; Cefa-iskia; Cefalexin (JP15); Cefalexin.H2O; Cefalexina [INN-Spanish]; Cefalexine [INN-French]; Cefalexinum [INN-Latin]; Cephalexin(USP); Cephalexin (anhydrous); Cephalexin 1-hydrate; Cephalexin 1-wasser; Cephalexin [USAN:BAN]; Cephalexin.H2O; Ceporexin-E; Cusisporina-Cefalox; Ed A-Ceph; KS-1134; Keflex (TN); Keftab (TN); L-Keflex; Panixine disperdose (TN); Sporidex (TN); Cephalexin, (6R-(6alpha,7beta))-Isomer; 7-(D-2-Amino-2-phenylacetamido)-3-methyl-delta (sup 3)-cephem-4-carboxylic acid; 7-(D-2-Amino-2-phenylacetamido)-3-methyl-delta3-cephem-4-carboxylic acid; 7-(D-alpha-Aminophenylacetamido)desacetoxycephalosporanic acid

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Activity

Ki = 68200 nM

[1]

Compound Name

Glycylglycine

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Investigative

Compound Info

Synonyms

Diglycine; N-GLYCYLGLYCINE; Gly-Gly; Glycine, glycyl-; Glycyl-glycine; Glycine dipeptide; 2-(2-Aminoacetamido)Acetic Acid; Glycine, N-glycyl-; H-Gly-Gly-OH; Gly-Gly-OH; 2-(Aminoacetamido)acetic acid; 2-[(2-aminoacetyl)amino]acetic acid; alpha-Glycylglycine; MFCD00008130; [(Aminoacetyl)amino]acetic acid; UNII-10525P22U0; CHEMBL292467; Glycylglycine, 99+%; 10525P22U0; glycylglycine zwitterion; ((aminoacetyl)amino)acetic acid; 2-(2-aminoacetylamino)acetic acid; Glycyl Glycine; Glycylgycine; EINECS 209-127-8; H-Gly-Gly; Glycylglycine, DL-; NSC 49346; .alpha.-Glycylglycine; n-GLYCYL- Glycine; PubChem14973; ACMC-1AWKP; AI3-62521; Glycylglycine (GLYGLY); Gly-Gly, 98%; B-GLYGLY250; SCHEMBL14934; KSC492E0P; CTK3J2207; DTXSID90862194; Gly-Gly, >=99% (titration); [(Aminoacetyl)amino]acetic acid #; HY-D0889; NSC49346; ZINC5112515; ANW-32355; BBL018705; BDBM50169222; NSC-49346; s4810; SBB067231; STL194277; AKOS001045997; CCG-231053; MCULE-1239116894; KS-000002A7; Gly-Gly, BioXtra, >=99.0% (NT); AK-46058; AS-14771; Gly-Gly, BioUltra, >=99.5% (NT); SC-17448; ST099026; SY018005; Gly-Gly, Vetec(TM) reagent grade, 99%; AB0006830; DB-002742; CS-0015211; FT-0626788; G0124; T7982; C02037; G-6000; G-6001; Glycylglycine, 0.2M buffer solution, pH 8.0; Glycylglycine, 0.2M buffer solution, pH 8.5; 556G503; Q665455; F2191-0195; 2,3,6,2',3',4',6'-Hepta-O-acetyl-a-D-lactosyl bromide; 33903968-DDB2-47F2-9B6C-7C232D1962DA; Dyglycine, United States Pharmacopeia (USP) Reference Standard; Gly-Gly, BioPerformance Certified, cell culture tested, >=99%

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Activity

Ki = 53703.18 nM

[2]

Compound Name

Glycylsarcosine

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Investigative

Compound Info

Synonyms

Glycyl-sarcosine; Gly-Sar; H-Gly-Sar-OH; 2-(2-amino-N-methylacetamido)acetic acid; N-Glycylsarcosine; Gly-Sarcosin; 2-[(2-aminoacetyl)-methylamino]acetic acid; UNII-2JE8SG6VDT; 2JE8SG6VDT; CHEMBL175737; MFCD00038193; N-glycyl-Sar-OH; EINECS 249-875-2; Gly-Sar-OH; [3H]GlySar; NSC 206288; glycyl-N-methylglycine; [3H]-GlySar; tritiated glycylsarcosine; N-glycyl-N-methylglycine; ACMC-209hb7; Glycine, N-glycyl-N-methyl-; SCHEMBL510835; GTPL4659; GTPL9505; CTK8B1399; DTXSID50183953; KS-000012VZ; ZINC1742265; 7028AH; ANW-26705; BDBM50188516; NSC206288; [(ammonioacetyl)(methyl)amino]acetate; AKOS009157522; NSC-206288; [(Aminoacetyl)(methyl)amino]acetic acid; AS-56734; [(Aminoacetyl)(methyl)amino]acetic acid #; FT-0760838; G0138; [(2-Amino-acetyl)-methyl-amino]-acetic acid; K-7194; J-017657

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Activity

Ki = 64000 nM

[1]

Compound Name

Ceftibuten

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Investigative

Compound Info

Synonyms

Cedax; Ceftibuteno; Ceftibutenum; Ceftibutene; Sch 39720; cis-ceftibuten; UNII-IW71N46B4Y; Cephem; cis-Ceftibutin; Sch-39720; Ceftibuten hydrate; 7432-S; Antibiotic 7432S; Cephalosporin 7432-S; IW71N46B4Y; 97519-39-6 (free); Isocef; MFCD00864918; Ceftibutene [INN-French]; Ceftibutenum [INN-Latin]; Ceftibuteno [INN-Spanish]; Ceftibuten [USAN:INN:BAN]; S 7432; Ceprifran; Ceftem; Keimax; NCGC00095137-01; Ceftibuten, 95%; Ceftibuten (USAN/INN); Spectrum5_001558; CHEMBL1605; DSSTox_CID_25925; DSSTox_RID_81227; DSSTox_GSID_45925; SCHEMBL37054; ACHN383; BSPBio_002733; SPECTRUM1505207; ACHN-383; DTXSID4045925; HMS1922L17; HMS2093K18; HMS3715P10; Pharmakon1600-01505207; HY-B0698; ZINC3871967; Tox21_111446; BDBM50370586; CC0255; CCG-39440; NSC758925; AKOS005146205; AKOS015854930; DB01415; NSC-758925; NCGC00178501-01; NCGC00178501-04; SC-27736; SBI-0206740.P001; C08117; D00922; AB01563048_01; 519C396; Ceftibuten, Antibiotic for Culture Media Use Only; Q419521; SR-05000001989; SR-05000001989-1

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Activity

Ki = 90000 nM

[3]

Compound Name

(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Amino-3-methylbutanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acid

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Investigative

Compound Info

Synonyms

CHEMBL1814497; BDBM50350485

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Activity

Ki = 109647.82 nM

[2]

Compound Name

d-Alanyl-l-alanine

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Investigative

Compound Info

Synonyms

H-D-Ala-Ala-OH; L-Alanine, D-alanyl-; N-ALANYLALANINE; UNII-C7641UJG3Q; C7641UJG3Q; CHEMBL1814491; (2S)-2-[[(2R)-2-aminopropanoyl]amino]propanoic acid; (S)-2-((R)-2-Aminopropanamido)propanoic acid; d-alanylalanine; NSC-203792; D-Ala-Ala-OHHCl; D-Ala-L-Ala-OH; D-Ala-Ala-OH HCl; N-D-Alanyl-L-alanine; H-D-Ala-Ala-OH HCl; SCHEMBL574263; CTK0I2831; DTXSID901016946; ZINC1575494; 7092AH; BDBM50350475; MFCD00066039; AKOS017430148; UNII-3CUV6EVI23 component DEFJQIDDEAULHB-DMTCNVIQSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-DMTCNVIQSA-N

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Activity

Ki = 128824.96 nM

[2]

Compound Name

Asp-Asp

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Compound Info

Synonyms

H-ASP-ASP-OH; (S)-2-((S)-2-Amino-3-carboxypropanamido)succinic acid; CHEMBL17171; Aspartyl-aspartic Acid; Asp-Asp-OH; L-Asp-L-Asp; NH2-Asp-Asp-COOH; alpha-aspartylaspartic acid; L-Aspartyl-L-aspartic acid; SCHEMBL434560; L-alpha-aspartyl-L-aspartic acid; ZINC1575288; BDBM50169127; MFCD00055820; 2-(2-Amino-3-carboxy-propionylamino)-succinic acid; Q27140532; (S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succinic acid

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Activity

Ki = 150000 nM

[2]

Compound Name

Ala-Ala-Asp

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Investigative

Compound Info

Synonyms

CHEMBL1814485; L-alanyl-L-alanyl-L-aspartic acid; L-Ala-L-Ala-L-Asp; Alanyl-alanyl-aspartic acid; A-A-D; BDBM50350459; ZINC13520692; (2S)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]propanoyl]amino]butanedioic Acid; Q27140433

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Activity

Ki = 158489.32 nM

[2]

Compound Name

(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Aminopropanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acid

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Investigative

Compound Info

Synonyms

CHEMBL1814486; BDBM50350460

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Activity

Ki = 190000 nM

[2]

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Non Binders of This Target (in total, 28 non binders)

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Compound Name

Dicloxacillin

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Approved

Compound Info

Synonyms

Dichloroxacillin; Diclossacillina; Dicloxaciclin; Dicloxacilin; Dicloxacilina; Dicloxacilline; Dicloxacillinum; Dicloxacycline; Dycill; Dynapen; Maclicine; Methyldichlorophenylisoxazolylpenicillin; Pathocil; Diclossacillina [DCIT]; Dicloxacillin sodium; BRL 1702; Diclocil (TN); Dicloxacilina [INN-Spanish]; Dicloxacilline [INN-French]; Dicloxacillinum [INN-Latin]; R-13423; Dicloxacillin (USAN/INN); Dicloxacillin [USAN:INN:BAN]; Dicloxacillin, Monosodium Salt, Mono-Hydrate; (2S,5R,6R)-6-({[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-({[3-(2,6-dichlorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-[[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolylpenicillin; 6-(3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(3-(2,6-Dichlorophenyl)-5-methyl-4-isoxazolecarboxamido)penicillanic acid; 6beta-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]carboxamido}-2,2-dimethylpenam-3alpha-carboxylic acid

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Activity

Ki = 416869.38 nM

[2]

Compound Name

Amoxicillin

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Approved

Compound Info

Synonyms

AMPC; Actimoxi; Amoclen; Amolin; Amopen; Amopenixin; Amoxi; Amoxibiotic; Amoxicaps; Amoxicilina; Amoxicillanyl; Amoxicilline; Amoxicillinum; Amoxiden; Amoxil; Amoxivet; Amoxycillin; Anemolin; Aspenil; Biomox; Bristamox; Cemoxin; Clamoxyl; Delacillin; DisperMox; Efpenix; Flemoxin; Hiconcil; Histocillin; Hydroxyampicillin; Ibiamox; Imacillin; Lamoxy; Larotid; Moxacin; Moxal; Moxatag; Ospamox; Pamoxicillin; Piramox; Polymox; Robamox; Sumox; Tolodina; Trimox; Unicillin; Utimox; Vetramox; Wymox; AMOXICILLIN CRYSTALLINE; AMOXICILLIN PEDIATRIC; Amoxicillin anhydrous; Amoxicilline [INN]; Amoxycillin Trihydrate; Metafarma capsules; Metifarma capsules; Sawamox PM; BLP 1410; AMK (TN); Actimoxi (TN); Alphamox (TN); Amoksibos (TN); Amoksiklav (TN); Amoxi-Mast; Amoxibiotic (TN); Amoxicilina (TN); Amoxicilina [INN-Spanish]; Amoxicillin (INN); Amoxicillin (TN); Amoxicillin (anhydrous); Amoxicilline [INN-French]; Amoxicillinum [INN-Latin]; Amoxiclav (TN); Amoxidal (TN); Amoxil (TN); Amoxin (TN); Apo-Amoxi; Augmentin (TN); BL-P 1410; BRL-2333; Bactox (TN); Betalaktam (TN); Cilamox (TN); Clamoxyl (TN); Curam (TN); D-Amoxicillin; Dedoxil (TN); Dispermox (TN); Duomox (TN); Enhancin (TN); Geramox (TN); Gimalxina (TN); Hiconcil (TN); Isimoxin (TN); Klavox (TN); Lamoxy (TN); Moxatag (TN); Moxilen (TN); Moxypen (TN); Moxyvit (TN); Nobactam (TN); Novamoxin (TN); Ospamox (TN); P-Hydroxyampicillin; Pamoxicillin (TN); Panamox (TN); Panklav (TN); Polymox (TN); Ro 10-8756; Samthongcillin (TN); Sandoz (TN); Senox (TN); Sinacilin (TN); Tolodina (TN); Trimox (TN); Wymox (TN); Yucla (TN); Zerrsox (TN); Zimox (TN); Apo-Amoxi (TN); Alpha-Amino-p-hydroxybenzylpenicillin; D-2-Amino-2-(4-hydroxyphenyl)acetamidopenicillanic acid; D-(-)-alpha-Amino-p-hydroxybenzylpenicillin; (-)-6-(2-Amino-2-(P-hydroxyphenyl)acetamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo-(3.2.0)heptane-2-carboxylic acid; (2S,5R,6R)-6-[[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-{[(2R)-2-amino-2-(4-hydroxyphenyl)acetyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 4-Thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid, 6-(2-amino-2-(p-hydroxyphenyl)acetamido)-3,3-dimethyl-7-oxo-, D-(8CI); 6-(D-(-)-alpha-Amino-p-hydroxyphenylacetamido)penicillanic acid; 6-(D-(-)-p-Hydroxy-alpha-aminobenzyl)penicillin; 6-(p-Hydroxy-alpha-aminophenylacetamido)penicillanic acid; 6beta-[(2R)-2-amino-2-(4-hydroxyphenyl)acetamido]-2,2-dimethylpenam-3alpha-carbonyl; 6beta-[(2R)-2-amino-2-(4-hydroxyphenyl)acetamido]-2,2-dimethylpenam-3alpha-carboxylic acid

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Activity

Ki = 426579.52 nM

[2]

Compound Name

Cyclacillin

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Approved

Compound Info

Synonyms

Aminocyclohexylpenicillin; Bastcillin; Calthor; Ciclacilina; Ciclacillin; Ciclacilline; Ciclacillinum; Ciclacillum; Citosarin; Cyclapen; Noblicil; Orfilina; Peamezin; Syngacillin; Ultracillin; Vastcillin; Vipicil; Wyvital; Aminocyclohexyl penicillin; Cyclacillin [USAN]; AC 98; WY 4508; WY4508; C-12104; Ciclacilina [INN-Spanish]; Ciclacilline [INN-French]; Ciclacillinum [INN-Latin]; Cyclacillin (USAN); Cyclapen (TN); Cyclapen-W; Vastcillin (TN); Wy-4508; Ciclacillin (JP15/INN); Cyclapen-W (TN); (1-Aminocyclohexyl)penicillin; (2S,5R,6R)-6-[(1-aminocyclohexanecarbonyl)amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-{[(1-aminocyclohexyl)carbonyl]amino}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 4-Thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid, 6-(1-aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-(8CI); 6-(1-Aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(1-Aminocyclohexanecarboxamido)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; 6-(1-Aminocyclohexanecarboxamido)penicillanic acid; 6-(1-Aminocyclohexylcarboxamido)penicillanic acid; 6beta-(1-aminocyclohexanecarboxamido)-2,2-dimethylpenam-3alpha-carboxylic acid

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Activity

IC50 = 610000 nM

[1]

Compound Name

Cloxacillin

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Compound Info

Synonyms

Chloroxacillin; Clossacillina; Cloxacilina; Cloxacilline; Cloxacillinum; MCIPC; Orbenin; Syntarpen; Tegopen; Clossacillina [DCIT]; Cloxacillin sodium; Methocillin S; BRL 1621; Cloxacilina [INN-Spanish]; Cloxacillin (INN); Cloxacillin [INN:BAN]; Cloxacilline [INN-French]; Cloxacillinum [INN-Latin]; Cloxapen (TN); Cloxapen (sodium monohydrate); Methylchlorphenylisoxazoryl-penicillin; Novo-Cloxin; Nu-Cloxi; Orbenin (TN); Tegopen (sodium monohydrate); BRL-1621 (sodium monohydrate); P-25 (sodium monohydrate); [3-(O-CHLOROPHENYL)-5-METHYL-4-ISOXAZOLYL]PENICILLIN; (2S,5R,6R)-6-({[3-(2-chlorophenyl)-5-methylisoxazol-4-yl]carbonyl}amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-6-[[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (3-(o-Chlorophenyl)-5-methyl-4-isoxazolyl)penicillin; 6-(((3-(2-Chlorophenyl)-5-methyl-4-isoxazolyl)carbonyl)amino)-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylic acid; 6-(3-(o-Chlorophenyl)-5-methyl-4-isoxazolecarboxamido)penicillanic acid

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Activity

Ki = 950000 nM

[2]

Compound Name

Ampicillin

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Approved

Compound Info

Synonyms

ABPC; Acillin; Adobacillin; Alpen; Amblosin; Amcill; Amfipen; Aminobenzylpenicillin; Ampen; Ampichel; Ampicil; Ampicilina; Ampicillanyl; Ampicillina; Ampicilline; Ampicillinum; Ampicin; Ampifarm; Ampikel; Ampimed; Ampipenin; Ampiscel; Ampisyn; Ampivax; Ampivet; Amplacilina; Amplin; Amplipenyl; Amplisom; Amplital; Austrapen; Binotal; Bonapicillin; Britacil; Campicillin; Cimex; Copharcilin; Delcillin; Deripen; Divercillin; Doktacillin; Duphacillin; Grampenil; Guicitrina; Guicitrine; Lifeampil; Morepen; Norobrittin; Nuvapen; Omnipen; Orbicilina; Penbristol; Penbritin; Penbrock; Penicline; Penimic; Pensyn; Pentrex; Pentrexl; Pentrexyl; Polycillin; Ponecil; Princillin; Principen; QIDamp; Racenacillin; Rosampline;Roscillin; Semicillin; Servicillin; Sumipanto; Supen; Synpenin; Texcillin; Tokiocillin; Tolomol; Totacillin; Totalciclina; Totapen; Trifacilina; Ukapen; Ultrabion; Ultrabron; Vampen; Viccillin; Wypicil; Amfipen V; Amipenix S; Ampicillin A; Ampicillin Anhydrous; Ampicillin Base; Ampicillin acid; Ampicillin anhydrate; Ampicillina [DCIT]; Anhydrous ampicillin; Olin Kid; Pen A; Pen A Oral; Pen Ampil;Penbritin paediatric; Penbritin syrup; Pfizerpen A; Semicillin R; Viccillin S; AY 6108; BA 7305; BRL 1341; Bayer 5427; HI 63; P 50; Principen 125; Principen 250; Principen 500; SQ 17382; AB-PC; AB-PCSol; AY-6108; Ambidrin (TN); Ampi-Co; Ampi-Tab; Ampi-bol; Ampicilina [INN-Spanish]; Ampicilline [INN-French]; Ampicillinum [INN-Latin]; Ampipenin, nt3; Ampy-Penyl; Anhydrous ampicillin (JP15); BRL-1341; D-Ampicillin; D-Cillin; KS-R1; Novo-ampicillin; OMNIPEN (AMPICILLIN); Omnipen (TN); Omnipen-N; P-50; Penbritin-S; Penicillin, Aminobenzyl; Pfizerpen-A; Polycillin-N; Polyflex (Veterinary); Ro-Ampen; SK-Ampicillin; Totacillin (sodium); Totacillin-N; WY-5103; Ampicillin (USP/INN); AMPICILLIN (SEE ALSO AMPICILLIN TRIHYDRATE 7177-48-2); Ampicillin [USAN:BAN:INN:JAN]; Ampicillin [USAN:INN:BAN:JAN];D-(-)-Ampicillin; D-(-)-alpha-Aminobenzylpenicillin; D-(-)-alpha-Aminopenicillin; D-(-)-6-(alpha-Aminophenylacetamido)penicillanic acid; 6-(D(-)-alpha-Aminophenylacetamido)penicillanic acid; 6beta-[(2R)-2-amino-2-phenylacetamido]-2,2-dimethylpenam-3alpha-carbonyl; 6beta-[(2R)-2-amino-2-phenylacetamido]-2,2-dimethylpenam-3alpha-carboxylic acid

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Activity

Ki = 1288249.55 nM

[2]

Compound Name

Cefixime

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Approved

Compound Info

Synonyms

CFIX; Cefixima; Cefiximum; Denvar; Necopen; Tricef; CL-284635; FK-027; FR-17027; Ofex (TN); Suprax (TN); Cefixime (JP15/USP/INN); (6R,7R)-7-({(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(carboxymethoxy)imino]acetyl}amino)-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(carboxymethyloxyimino)acetyl]amino]-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-{[(carboxymethyl)oxy]imino}acetyl]amino}-3-ethenyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6r,7r)-7-[-2-(2-amino-thiazol-4-yl)-2-carboxymethoxyimino-acetylamino]-8-oxo-3-vinyl-5-thia-1-aza-b; 7beta-{(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(carboxymethoxy)imino]acetamido}-3-ethenyl-3,4-didehydrocepham-4-carboxylic acid

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Activity

Ki = 2570395.78 nM

[2]

Compound Name

Cefamandole

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Approved

Compound Info

Synonyms

Cefadole; Cefamandolum; Cefamandole (USAN/INN); (6R,7R)-7-(R)-Mandelamido-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-carboxylic acid; (6R,7R)-7-[[(2R)-2-hydroxy-2-phenylacetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-hydroxy-2-phenylacetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-{[(2R)-2-hydroxy-2-phenylacetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)thio]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7beta-[(2R)-2-hydroxy-2-phenylacetamido]-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}ceph-3-em-4-carboxylic acid

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Activity

Ki = 2800000 nM

[2]

Compound Name

Oxacillin

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Approved

Compound Info

Synonyms

Bactocill; Ossacillina; Oxacilina; Oxacilline; Oxacillinum; Oxazocillin; Oxazocilline; Prostaphlin; Prostaphlyn; OXACILLIN SODIUM; Ossacillina [DCIT]; Sodium oxacillin; Bactocill (TN); MPI-penicillin; MPi-PC; Oxacilina (TN); Oxacilina [INN-Spanish]; Oxacillin (INN); Oxacillin [INN:BAN]; Oxacilline [INN-French]; Oxacillinum [INN-Latin]; Penicillin, Methylphenylisoxazolyl; Oxacillin, Monosodium Salt, Anhydrous; (2S,5R,6R)-3,3-dimethyl-6-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (2S,5R,6R)-3,3-dimethyl-6-{[(5-methyl-3-phenylisoxazol-4-yl)carbonyl]amino}-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid; (5-methyl-3-phenyl-4-isoxazolyl)penicillin; 2,2-dimethyl-6beta-(5-methyl-3-phenyl-1,2-oxazole-4-carboxamido)penam-3alpha-carboxylic acid; 5-Methyl-3-phenyl-4-isoxazolyl-penicillin; 6beta-(5-methyl-3-phenylisoxazol-4-yl)penicillanic acid

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Activity

Ki = 3300000 nM

[2]

Compound Name

Cefmetazole

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Approved

Compound Info

Synonyms

CMZ; Cefmetazolo; Cefmetazolum; Cefmetazole Monosodium Salt; CS 1170; SKF 83088; U 72791; CS-1170; Cefmetazole [USAN:INN]; Cefmetazolo [INN-Spanish]; Cefmetazolum [INN-Latin]; U-72791A; Cefmetazole (USP/INN); (6R,7S)-7-(2-((Cyanomethyl)thio)acetamido)-7-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thio)methyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; (6R,7S)-7-(2-((Cyanomethyl)thio)acetamido)-7-methoxy-3-(((1-methyl-1H-tetrazol-5-yl)thiomethyl)-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, sodium salt; (6R,7S)-7-({[(cyanomethyl)sulfanyl]acetyl}amino)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7S)-7-({[(cyanomethyl)thio]acetyl}amino)-7-(methyloxy)-3-{[(1-methyl-1H-tetrazol-5-yl)thio]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7S)-7-[[2-(cyanomethylsulfanyl)acetyl]amino]-7-methoxy-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 6beta-{[(cyanomethyl)sulfanyl]acetamido}-6alpha-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}ceph-3-em-4-carboxylic acid

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Activity

Ki = 4265795.19 nM

[2]

Compound Name

Cefalotin

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Approved

Compound Info

Synonyms

Cefalothin; Cefalotina; Cefalotine; Cefalotinum; Cemastin; Cephalothinum; Cephalotin; Coaxin; Cefalotina fabra; Cephalothin Monosodium Salt; Averon-1; Cefalotin (BAN); Cefalotina [INN-Spanish]; Cefalotina fabra (TN); Cefalotine [INN-French]; Cefalotinum [INN-Latin]; Keflin (TN); (6R,7R)-3-(acetyloxymethyl)-8-oxo-7-[(2-thiophen-2-ylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-3-[(acetyloxy)methyl]-8-oxo-7-[(2-thienylacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 3-(Acetoxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid; 3-(Hydroxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-5-thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid acetate; 3-ACETOXYMETHYL-8-OXO-7-(2-THIOPHEN-2-YL-ACETYLAMINO)-5-THIA-1-AZA-BICYCLO[4.2.0]OCT-2-ENE-2-CARBOXYLIC ACID; 3-Acetoxymethyl-7-(2-thienylacetamido)-3-cephem-4-carboxylic acid; 5-Thia-1-azabicyclo(4.2.0)oct-2-ene-2-carboxylic acid, 3-(hydroxymethyl)-8-oxo-7-(2-(2-thienyl)acetamido)-, acetate (ester); 6R-trans-3-((Acetyloxy)methyl)-8-oxo-7-((2-thienylacetyl)amino)-5-thia-1-azabicyclo(4.2.0)-oct-2-ene-2-carboxylic acid; 7-(2-(2-Thienyl)acetylamido)cephalosporanic acid; 7-(2-Thienylacetamido)cephalosporanic acid; 7-(Thiophene-2-acetamido)cephalosporanic acid; 7-(Thiophene-2-acetamido)cephalosporin; 7beta-(thiophen-2-ylacetamido)-3-acetoxymethyl-3,4-didehydrocepham-4-carboxylic acid

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Activity

Ki = 8300000 nM

[2]

Compound Name

Cefepime

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Approved

Compound Info

Synonyms

Axepim; CFPM; Cefepima; Cefepimum; Cepimax; Cepimex; Maxcef; Maxipime; Cefepima [Spanish]; Cefepimum [Latin]; BMY 28142; Axepim (TN); BMY-28142; Cefepime [USAN:INN]; Cepimax (TN); Cepimex (TN); Maxcef (TN); Maxipime (TN); Cefepime (USAN/INN); (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-[(1-methylpyrrolidin-1-ium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate; (6R,7R)-7-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}-3-[(1-methylpyrrolidinium-1-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate; 1-(((6R,7R)-7-(2-(2-Amino-4-thiazolyl)glyoxylamido)-2-carboxy-8-oxo-5-thia-1-azabicyclo(4.2.0)oct-2-en-3-yl)methyl)-1-methylpyrrolidinium hydroxide, inner salt, 7(sup 2)-(Z)-(O-methyloxime); 7beta-[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetamido]-3-[(1-methylpyrrolidinium-1-yl)methyl]-3,4-didehydrocepham-4-carboxylate

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Activity

Ki = 10964781.96 nM

[2]

Compound Name

Cefpodoxime

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Approved

Compound Info

Synonyms

CPDX; Cefpodoxima; Cefpodoximum; Epoxim; Cefpodoxim acid; Cefpodoxima [Spanish]; Cefpodoximum [Latin]; RU 51807; Cefpodoxime (INN); Cefpodoxime [INN:BAN]; Epoxim (TN); Vantin (TN); (6R,7R)-7-({(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-[(methyloxy)imino]acetyl}amino)-3-[(methyloxy)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2E)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; (6R,7R)-7-[[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-methoxyiminoacetyl]amino]-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid; 7-{[(2-amino-1,3-thiazol-4-yl)(methoxyimino)acetyl]amino}-3-(methoxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid

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Activity

Ki = 30902954.33 nM

[2]

Compound Name

Benzylpenicillin

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Phase 3

Compound Info

Synonyms

penicillin g; Benzylpenicillinic acid; Free penicillin II; Pencillin G; 61-33-6; Benzylpenicillin G; Bencilpenicilina; Benzylpenicillinum; Benzyl penicillin; Free penicillin G; Dropcillin; Pharmacillin; Gelacillin; Liquacillin; Benzopenicillin; Cilopen; Pradupen; Benzylpenicilline; Specilline G; Cilloral; Cosmopen; Ursopen; Galofak; Free benzylpenicillin; Compocillin G; Phenylacetamidopenicillanic acid; 6-(2-Phenylacetamido)penicillanic acid; Pfizerpen; Benzyl-6-aminopenicillinic acid

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Activity

Ki = 10964781.96 nM

[2]

Compound Name

Cephaloridine

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Withdrawn from market

Compound Info

Synonyms

cephaloridine; cefaloridine; Cefaloridin; Cephaloridin; Cephaloridinum; Cepaloridin; Cefalorizin; Cephalomycine; Cefaloridinum; Cepalorin; Cefaloridina; Loridine; Ceflorin; 50-59-9; Kefloridin; Glaxoridin; Ceporin; Vioviantine; Intrasporin; Sefacin; Keflordin; Deflorin; Cilifor; Ceporan; Sasperin; Faredina; Ceporine; Keflodin; Verolgin; Lloncefal; Kefspor; Ampligram; Betaine cephaloridine; CHEBI:3537; UNII-LVZ1VC61HB; Cefaloridinum [INN-Latin]; Cefaloridina [INN-Spanish]; N-(7-(2'-Thienylacetamidoceph-3-ylmethyl))-pyridinium-2-carboxylate; SCH

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Activity

Ki = 8500000 nM

[2]

Compound Name

Laevulinic Acid

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Investigative

Compound Info

Synonyms

Levulinic acid; LEVULINIC ACID; 4-Oxopentanoic acid; 123-76-2; Laevulinic acid; Pentanoic acid, 4-oxo-; 4-Oxovaleric acid; Levulic acid; 3-Acetylpropionic acid; 4-Ketovaleric acid; LEVA; gamma-Ketovaleric acid; Acetopropionic acid; Levulinsaeure; Laevulic acid; Valeric acid, 4-oxo-; beta-Acetylpropionic acid; USAF CZ-1; 4-oxo-pentanoic acid; Propionic acid, 3-acetyl-; 4-Oxopentansaeure; Acidum laevulinicum; 3-Acetylpropionsaeure; 3-Ketobutane-1-carboxylic acid; UNII-RYX5QG61EI; NSC 3716; Acetylpropionic acid; FEMA No 2627; Pentanoic acid, 4-oxo; Levulinic Acid

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Activity

Ki = 229086.77 nM

[2]

Compound Name

(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Amino-3-phenylpropanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acid

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Investigative

Compound Info

Synonyms

CHEMBL1814496; BDBM50350484

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Activity

Ki = 239883.29 nM

[2]

Compound Name

Alanyl-D-alanine

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Investigative

Compound Info

Synonyms

H-ALA-D-ALA-OH; D-Alanine, L-alanyl-; l-alanyl-d-alanine; Ala-D-Ala-OH; (2R)-2-[[(2S)-2-aminopropanoyl]amino]propanoic acid; CHEMBL1814487; UNII-A8235021UP; A8235021UP; L-Ala-D-Ala-OH; N-L-Alanyl-D-alanine; SCHEMBL380600; CTK1C3694; DTXSID201016945; ZINC1575495; 7042AH; BDBM50350461; MFCD00066040; AKOS010842226; NSC 186898; (R)-2-((S)-2-Aminopropanamido)propanoic acid; K-8204; Q27896855; UNII-3CUV6EVI23 component DEFJQIDDEAULHB-IUYQGCFVSA-N; UNII-3EE68A29TN component DEFJQIDDEAULHB-IUYQGCFVSA-N

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Activity

Ki = 269153.48 nM

[2]

Compound Name

(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-Aminopropanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]propanoic acid

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Investigative

Compound Info

Synonyms

CHEMBL1814490; BDBM50350466

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Activity

Ki = 549540.87 nM

[2]

Compound Name

Metampicillin

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Investigative

Compound Info

Synonyms

METHAMPICILLIN; UNII-G0H6U7VSTK; Magnipen; G0H6U7VSTK; METAMPICILLIN SODIUM; 6beta-[(2R)-2-(methylideneamino)-2-phenylacetamido]penicillanic acid; metampilene; Metampicillinum; Celinmicina; Elatocilline; Metampicilina; Metampicillina; Metampicilline; Pangocilin; Relyothenate; Blomopen; Bonopen; Filorex; Metambac; Micinovo; Probiotic; Ruticina; Rutizina; Sedomycin; Suvipen; Viderpen; Viderpin; Vioplex; Teonicon Trofen; Italcina kapseln; Suvipen ampullen; Rastomycin K; Meta-Alvar; Metiskia ampullen; Micinovo ampullen; Rutizina ampullen; Tampilen ampullen; Fedacilina kapseln; Metabacter ampullen; Metampicillina [DCIT]; Metampicilina [Spanish]; Metampicilline [French]; Metampicillinum [Latin]; Metampicillin [INN:DCF]; Metampicilina [INN-Spanish]; Metampicillinum [INN-Latin]; EINECS 229-365-6; Metampicillin (INN); (alpha-(Methyleneamino)benzyl)penicillin; CB 28020; D-(-)-alpha-Methyleneaminobenzylpenicillin; Prestwick0_000235; Prestwick1_000235; Prestwick2_000235; Prestwick3_000235; Epitope ID:141487; SCHEMBL34032; BSPBio_000309; SPBio_002230; BPBio1_000341; CHEMBL1908324; DTXSID5048479; ZINC3874216; BDBM50370588; DB13836; D07234; BRD-K83350436-236-03-4

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Activity

Ki = 724435.96 nM

[2]

Compound Name

(2S)-6-Amino-2-[[(2S)-3-phenyl-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoyl]amino]hexanoic Acid

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Investigative

Compound Info

Synonyms

Pro-Phe-Lys; CHEMBL426809; H-Pro-Phe-Lys-OH; Prolyl-phenylalanyl-lysine; L-Prolyl-L-phenylalanyl-L-lysine; ZINC4899895; BDBM50169183; (S)-6-Amino-2-{(S)-3-phenyl-2-[((S)-pyrrolidine-2-carbonyl)-amino]-propionylamino}-hexanoic acid

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Activity

Ki = 891250.94 nM

[2]

Compound Name

Pro-Asp

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Investigative

Compound Info

Synonyms

H-Pro-Asp-OH; L-prolyl-L-aspartic acid; CHEMBL190704; (2S)-2-[[(2S)-pyrrolidine-2-carbonyl]amino]butanedioic acid; Prolyl-Aspartate; l-pro l-asp; prolyl-aspartic acid; L-Pro-L-Asp; L-Aspartic acid, L-prolyl-; CTK3C9100; ZINC4029831; BDBM50169195; MFCD00057886; STL527058; AKOS030494433; MCULE-3726564210; AS-56431; Q27144883; (S)-2-[((S)-Pyrrolidine-2-carbonyl)-amino]-succinic acid

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Activity

Ki = 2089296.13 nM

[2]

Compound Name

Prolylglutamic acid

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Investigative

Compound Info

Synonyms

Pro-glu; L-Prolyl-L-glutamic acid; CHEMBL190027; Prolyl-Glutamate; H-Pro-Glu-OH; pro glu; Prolyl-glutamic acid; L-Pro-L-Glu; N-L-Prolyl-L-glutamic acid; L-Glutamic acid, L-prolyl-; SCHEMBL5408968; L-Glutamic acid, N-L-prolyl-; CTK5C6473; DTXSID70987011; C10H16N2O5; ZINC3776573; BDBM50169114; MFCD00037872; STL527174; AKOS010408434; MCULE-1644415057; AS-58357; N-[Hydroxy(pyrrolidin-2-yl)methylidene]glutamic acid; Q27144887; (2S)-2-{[(2S)-pyrrolidin-2-yl]formamido}pentanedioic acid

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Activity

Ki = 2570395.78 nM

[2]

Compound Name

Glycyl-l-histidyl-l-lysine

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Investigative

Compound Info

Synonyms

Gly-his-lys; Glycyl-histidyl-lysine; Glycylhistidyllysine; L-Lysine, glycyl-L-histidyl-; Liver cell growth factor; UNII-39TG2H631E; NSC 379527; Copper Peptide; CHEMBL1814493; 39TG2H631E; Copper(II)ghk; Prezatide; Copper glycyl-histidyl-lysine; Tripeptide-1; Gly-L-His-L-Lys; H-Gly-His-Lys-OH; Gly-L-His-L-Lys-OH; SCHEMBL259085; SCHEMBL19087235; CTK5D7156; KS-00000GCA; DTXSID30197831; Growth-modulating peptide (human); ANW-61320; BDBM50350478; MFCD00036754; ZINC13507674; AKOS016003505; DB11296; N(2)-(N-Glycyl-L-histidyl)-L-lysine; AC-31946; DS-14630; CS-0005654; Y-9228; 557G757

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Activity

Ki = 3090295.43 nM

[2]

Compound Name

Cefodizime

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Investigative

Compound Info

Synonyms

Cefodizima; Cefodizimum; UNII-Z31298J4HQ; HR 221 [AS SODIUM]; THR 221 [AS SODIUM]; Z31298J4HQ; S 77 1221 B [AS SODIUM]; THR-221; Cefodizime [INN:BAN]; Cefodizimum [INN-Latin]; Cefodizima [INN-Spanish]; Cefodizme; Diezime; Modivid; Timecef; Neucef; Cefodizime Acid; Cefodizime (INN); EC 700-301-3; HR-221 [As Sodium]; THR-221 [As Sodium]; SCHEMBL151101; CHEMBL2303613; DTXSID2022757; S-771221B [As Sodium]; EX-A1379; ZINC3871933; A0C261; BDBM50422690; HR-221; MFCD00864926; DB13470; HY-108402; CS-0028575; D07643; J-700161

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Activity

Ki = 8912509.38 nM

[2]

Compound Name

H-Pro-gly-gly-OH

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Investigative

Compound Info

Synonyms

Pro-gly-gly; Prolyl-glycyl-glycine; CHEMBL190343; 2-[[2-[[(2S)-pyrrolidine-2-carbonyl]amino]acetyl]amino]acetic acid; l-prolylglycylglycine; Pro-Gly-Gly-OH; Prolyl-glycyl-glycin; NSC 97937; Glycine,L-prolylglycyl-; L-Prolyl-glycyl-glycine; Glycine, L-prolylglycyl-; SCHEMBL10788841; CTK8D8729; Glycine, N-(N-L-prolylglycyl)-; ZINC4899450; 7229AH; BDBM50169143; MFCD00037877; AKOS010407662; 561P253; (S)-2-(2-(pyrrolidine-2-carboxamido)acetamido)acetic acid; {2-[(Pyrrolidine-2-carbonyl)-amino]-acetylamino}-acetic acid

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Ki = 10964781.96 nM

[2]

Compound Name

Cephapirin sodium

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Investigative

Compound Info

Synonyms

cefapirin sodium; Sodium cefapirin; Sodium cephapirin; Cefadyl; UNII-431LFF7I7J; Cefatrexyl; Ambrocef; Cefatrex; Cefapirin sodium salt; BLP 1322; Sodium 7-(pyrid-4-ylthioacetamido)cephalosporanate; Cephapirin sodium salt; 431LFF7I7J; BL-P 1322; Cefaloject; Cephatrexil; Cefa lak; Cela-Lak/ToDay; 7-(alpha-(4-Pyridylthio)acetamido)cephalosporanic acid sodium salt; DSSTox_CID_25574; DSSTox_RID_80971; DSSTox_GSID_45574; Brisfirina; Cephatrexyl; Brisporin; Bristocef; Cefapirina sodica; Cefadyl IM/IV; Cefa-Lak (Veterinary); Antibiotic BL-P 1322; 356C603; Cephapirin sodium [USAN:USP]; Prestwick_27; NCGC00017093-01; Cefadyl (TN); EINECS 246-194-2; NSC 179171; Cefapirin sodium (JAN); Cephapirin sodium (USP); Cephapirin sodium, >=96%; SCHEMBL64430; SPECTRUM1500167; CHEMBL1201043; DTXSID7045574; HMS500C04; HMS1570L03; HMS1920K13; HMS2091A16; Tox21_110772; BL-P-1322; CCG-38912; Cefapirin sodium, analytical standard; AKOS024282660; Tox21_110772_1; NCGC00093735-01; NCGC00162116-04; ST057376; EU-0100279; C 8270; C08101; D00908; Q27106128; Cefapirin sodium, European Pharmacopoeia (EP) Reference Standard; Cephapirin sodium, United States Pharmacopeia (USP) Reference Standard

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Activity

Ki = 11100000 nM

[2]

Compound Name

Cefuroxime

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Investigative

Compound Info

Synonyms

Cephuroxime; Cefuroximo; Cefuroxim; Cefuroximum; Zinacef Danmark; Zinacef; Cefuroximum [INN-Latin]; Cefuroximo [INN-Spanish]; UNII-O1R9FJ93ED; Biofuroksym; Cefuril; O1R9FJ93ED; Q63409033; Cefuroxime [USAN:INN:BAN]; C16H16N4O8S; EINECS 259-560-1; BRN 5783190; Cefuroximine; Cefuroxime [USAN:BAN:INN]; Cefuroxime (TN); Cefuroxime (USAN/INN); Prestwick3_000720; CHEMBL1436; BSPBio_000939; BIDD:GT0619; BPBio1_001033; SCHEMBL1821942; HY-B1256A; ZINC3830485; BDBM50422689; MFCD00864889; AKOS015962849; AC-4539; DB01112; KS-5162; AB0010602; CS-0013520; EN300-53016; C06894; Cefuroxime, VETRANAL(TM), analytical standard; D00262; 268C752; A830563; Cefuroxime, Antibiotic for Culture Media Use Only; W-105575; BRD-K02733959-236-02-8; BRD-K02733959-236-07-7

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Activity

Ki = 12589254.12 nM

[2]

Compound Name

Cefotaxime

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Investigative

Compound Info

Synonyms

Cephotaxime; Cefotaxime acid; E-cefotaxime; UNII-N2GI8B1GK7; Cefotaximum; Cefotaxima; N2GI8B1GK7; Omnatax; Taxim; HR 756; Cefotaxime [INN:BAN]; RU 24756; Cefotaximum [INN-Latin]; Cefotaxima [INN-Spanish]; Cefotaxime (INN); EINECS 264-299-1; Cefotaxim Hikma (TN); RU 24662; Prestwick2_000139; Prestwick3_000139; Claforan (*Sodium salt*); CHEMBL1730; Lopac0_000278; BSPBio_000218; BPBio1_000240; SCHEMBL3731931; DTXSID6022761; HY-A0088A; HMS2090M11; ZINC3830437; AC-217; BDBM50482777; MFCD00864971; s4720; AKOS015951267; DB00493; SDCCGSBI-0050266.P002; AS-12690; clo[4.2.0]oct-2-ene-2-carboxylic acid; CS-0013515; C06885; D07647; J90010; 527C526; BRD-K78364995-236-03-5; Q27262497; Di- poundg-chlorotetrakis[2,4-dimethyl-6-(2-quinolinyl-KN)phenyl-KC]di-iridium

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Activity

Ki = 19952623.15 nM

[2]

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References

Top

REF 1

Differential recognition of beta -lactam antibiotics by intestinal and renal peptide transporters, PEPT 1 and PEPT 2. J Biol Chem. 1995 Oct 27;270(43):25672-7.

REF 2

Fragmental modeling of hPepT2 and analysis of its binding features by docking studies and pharmacophore mapping. Bioorg Med Chem. 2011 Aug 1;19(15):4544-51.

REF 3

Interaction of anionic cephalosporins with the intestinal and renal peptide transporters PEPT 1 and PEPT 2. Biochim Biophys Acta. 1997 Mar 13;1324(2):296-308.

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