Target Poor or Non Binder(s) Information
Target General Information | Top | ||||
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Target ID | T68066 | Target Info | |||
Target Name | Steroid hormone receptor ERR (ESRR) | ||||
Synonyms |
Nuclear receptor subfamily 3 group B; NR3B; ERR
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Target Type | Successful Target | ||||
Gene Name | ESRRA; ESRRB; ESRRG | ||||
Biochemical Class | Nuclear hormone receptor | ||||
UniProt ID |
Poor Binders of This Target (in total, 5 binders) | Download | Top | |||
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Compound Name |
(2-Aminophenyl)-[1-(3-phenylmethoxyphenyl)triazol-4-yl]methanone
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2381361; BDBM50434085
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Activity | Estrogen-related receptor alpha |
IC50 ~ 50000 nM
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[1] | ||
Compound Name |
3-[4-(2-Aminobenzoyl)triazol-1-yl]benzoic acid
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2381367; BDBM50434079
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Activity | Estrogen-related receptor alpha |
IC50 ~ 50000 nM
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[1] | ||
Compound Name |
[1-(4-Propan-2-ylphenyl)triazol-4-yl]-[2-(trifluoromethyl)phenyl]methanone
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2381475; BDBM50434100
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Activity | Estrogen-related receptor alpha |
IC50 ~ 50000 nM
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[1] | ||
Compound Name |
3-[4-(2-Aminobenzoyl)triazol-1-yl]benzenesulfonamide
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2381366; BDBM50434080
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Activity | Estrogen-related receptor alpha |
IC50 ~ 50000 nM
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[1] | ||
Compound Name |
3-[4-(2-Aminobenzoyl)triazol-1-yl]benzonitrile
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Investigative | Compound Info | ||
Synonyms |
CHEMBL2381365; BDBM50434081
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Activity | Estrogen-related receptor alpha |
IC50 ~ 50000 nM
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[1] |
References | Top | ||||
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REF 1 | 1-Phenyl-4-benzoyl-1H-1,2,3-triazoles as orally bioavailable transcriptional function suppressors of estrogen-related receptor alpha. J Med Chem. 2013 Jun 13;56(11):4631-40. |
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