Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T67416 | Target Info | |||
| Target Name | Bifunctional aminoacyl-tRNA synthetase (EPRS) | ||||
| Synonyms |
QPRS; QARS; ProlinetRNA ligase; PIG32; GlutamatylprolyltRNA synthetase; Glutamatyl-prolyl-tRNA synthetase; GluRS; EPRS; Cell proliferationinducing gene 32 protein; Cell proliferation-inducing gene 32 protein; Bifunctional glutamate/prolinetRNA ligase; Bifunctional glutamate/proline--tRNA ligase; Bifunctional aminoacyltRNA synthetase
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| Target Type | Clinical trial Target | ||||
| Gene Name | EPRS | ||||
| Biochemical Class | Carbon-oxygen ligase | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 26 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
6-Bromo-2-(4-bromophenyl)-8-(trifluoromethyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL149973; SCHEMBL116080; BDBM50097104; 2-(4-Bromophenyl)-6-bromo-8-(trifluoromethyl)quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 6-bromo-2-(4-bromophenyl)-8-(trifluoromethyl)-; 6-Bromo-2-(4-bromo-phenyl)-8-trifluoromethyl-quinoline-4-carboxylic acid
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| Activity |
IC50 = 56000 nM
|
[1] | |||
| Compound Name |
2-(4-Bromophenyl)-7-fluoro-8-methylquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL346646; SCHEMBL117434; BDBM50097107; 2-(4-Bromo-phenyl)-7-fluoro-8-methyl-quinoline-4-carboxylic acid; 2-(4-bromophenyl)-7-fluoro-8-methyl-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-7-fluoro-8-methyl-
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| Activity |
IC50 = 60000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-7-bromo-8-methylquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL348184; SCHEMBL117482; BDBM50097093; 4-Quinolinecarboxylic acid, 7-bromo-2-(4-bromophenyl)-8-methyl-; 7-Bromo-2-(4-bromo-phenyl)-8-methyl-quinoline-4-carboxylic acid; 7-bromo-2-(4-bromophenyl)-8-methyl-quinoline-4-carboxylic acid
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| Activity |
IC50 = 70000 nM
|
[1] | |||
| Compound Name |
2-(4-Bromo-phenyl)-6-((E)-2-carboxy-vinyl)-quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL150306; BDBM50097087; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-[(E)-2-carboxyethenyl]-; 2-(4-Bromophenyl)-6-(3-oxo-3-hydroxy-1-propenyl)quinoline-4-carboxylic acid; 2-(4-bromophenyl)-6-[(E)-3-hydroxy-3-oxo-prop-1-enyl]quinoline-4-carboxylic acid
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| Activity |
IC50 = 80000 nM
|
[1] | |||
| Compound Name |
6-Amino-2-(4-bromophenyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL356452; SCHEMBL117388; BDBM50097099; 2-(4-Bromophenyl)-6-aminoquinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 6-amino-2-(4-bromophenyl)-; 6-Amino-2-(4-bromo-phenyl)-quinoline-4-carboxylic acid
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| Activity |
IC50 = 95000 nM
|
[1] | |||
| Compound Name |
2-(Pyridin-4-yl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-pyridin-4-ylquinoline-4-carboxylic acid; 2-(4-pyridinyl)-4-quinolinecarboxylic acid; 2-Pyridin-4-yl-quinoline-4-carboxylic acid; NSC360211; 4-Quinolinecarboxylic acid, 2-(4-pyridinyl)-; CINCHONINIC ACID, 2-(4-PYRIDYL)-; 2-(4-pyridyl)quinoline-4-carboxylic acid; CHEMBL415737; NSC-360211; 2-(4-Pyridyl)cinchoninic acid; NSC 360211; 2-(4-Pyridyl)cinchoninsaeure [German]; BRN 0017972; 2-(4-Pyridyl)cinchoninsaeure; Kyselin 2-(4-pyridyl)-cinchoninova [Czech]; Kyselin 2-(4-pyridyl)-cinchoninova; Cambridge id 5542580; NCIStruc1_000902; NCIStruc2_000832; Oprea1_338008; Oprea1_758729; 5-25-05-00236 (Beilstein Handbook Reference); SCHEMBL116042; CTK0I1174; ZINC65268; DTXSID90161997; ALBB-000774; 4267AD; AR3149; BBL009856; BDBM50097097; CCG-37557; MFCD00687610; NCGC00014819; NCI360211; SBB011934; STK364547; AKOS000121700; AB06957; MCULE-6246568887; NCGC00014819-02; NCGC00014819-03; NCGC00097920-01; AS-45535; NCI60_003280; ST078406; AB0086917; DB-042620; 2-(4-Pyridinyl)quinoline-4-carboxylic acid; BB 0217752; CS-0116568; FT-0637038; 4-Quinolinecarboxylicacid, 2-(4-pyridinyl)-; EN300-00687; W-7482; AB00088210-01; AB00088210-04; 228P230; SR-01000908315; SR-01000908315-1; Z56792374; F1142-0435
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| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Cinchophen
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Investigative | Compound Info | ||
| Synonyms |
2-Phenylquinoline-4-carboxylic acid; 2-Phenyl-4-quinolinecarboxylic acid; Cinchopen; 2-Phenylcinchoninic acid; Cinconal; Atophan; Cinchophene; Phenoquin; Quinofen; Quinophan; Quinophen; Tervalon; Atofan; Cinchophenic acid; Aciphenochinolinium; Polyphlogin; Aminophan; Artexin; Cincosal; Ikterosan; Mylofanol; Phenophan; Rhematan; Rheumin; Tophosan; Traubofan; Viophan; Agotan; Alutyl; Artam; Atigoa; Atocin; Tophol; Vantyl; Aciphenochinoline; CINCOPHEN; 2-Phenylcinchonic acid; 4-Quinolinecarboxylic acid, 2-phenyl-; Cinchoninic acid, 2-phenyl-; 2-Phenyl-quinoline-4-carboxylic acid; NSC 2617; UNII-39Y533Z02M; MLS000053018; CHEMBL348000; MFCD00006750; 39Y533Z02M; NCGC00018221-06; NCGC00018221-08; Acifenokinolin; Artamin; SMR000059017; Aciphenochinolinum; DSSTox_CID_20705; DSSTox_RID_79555; DSSTox_GSID_40705; Cincofene [DCIT]; Cinchophenum; Cincofene; Cincofeno; WLN: T66 BNJ CR & EVQ; Cincofeno [INN-Spanish]; Cinchophene [INN-French]; Cinchophenum [INN-Latin]; Phenylcinchoninic Acid; HSDB 2085; 2-Phenylquinoline-4-carboxlic acid; SR-01000000141; EINECS 205-067-1; BRN 0192803; Cinchophen [INN:BAN:NF]; Rheumatan; Alutyo; AI3-15400; Cinchophen (BAN); Cincain (TN); ACMC-209bpl; Opera_ID_819; N-Cyclohexyl-2-phenyl-4-chinolincarboxamid; Cambridge id 5117240; TimTec1_001239; Oprea1_652483; SCHEMBL25519; 5-22-03-00484 (Beilstein Handbook Reference); MLS000069591; MLS001074296; DTXSID0040705; CTK0H5112; NSC2617; HMS1537I07; HMS2236H09; HMS3264N13; HMS3369G13; HMS3652D09; Pharmakon1600-01504508; ZINC125047; HY-B0972; KS-00000UU3; NSC-2617; NSC70178; Tox21_110841; Tox21_400022; ANW-19447; BBL011719; BDBM50097100; CCG-34161; NSC-70178; NSC758887; SBB000885; STK076256; 2-phenyl-4-quinoline-carboxylic acid; 2-Phenylquinolinecarboxylic acid-(4); 4-Quinolinecarboxylicacid, 2-phenyl-; AKOS000264299; Tox21_110841_1; CS-4461; DB13551; MCULE-5908309566; NE10455; NSC-758887; SB18446; NCGC00018221-01; NCGC00018221-02; NCGC00018221-03; NCGC00018221-04; NCGC00018221-05; NCGC00018221-07; NCGC00018221-09; NCGC00018221-10; NCGC00018221-13; NCGC00021229-04; NCGC00021229-05; NCGC00021229-06; AS-56238; ST013890; 2-Phenyl-4-quinolinecarboxylic acid, 99%; SBI-0207075.P001; DB-000656; EU-0096447; FT-0623825; P1301; S4190; SW089640-2; X6853; 4-Quinolinecarboxylic acid, 2-phenyl- (9CI); A16453; D07280; AB00275103-10; AB00275103-16; AB00275103_18; AB00275103_19; AE-641/00678051; J-006195; Q5120196; SR-01000000141-2; SR-01000000141-4; BRD-K72915123-001-01-7; BRD-K72915123-001-11-6; Z56782585; F0391-0013
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(5-Chlorothiophen-2-yl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-(5-Chloro-thiophen-2-yl)-quinoline-4-carboxylic acid; 2-(5-chloro-2-thienyl)quinoline-4-carboxylic acid; 2-(5-chlorothien-2-yl)quinoline-4-carboxylic acid; CHEMBL153072; Oprea1_512722; MLS000759674; SCHEMBL117380; cid_625773; CTK4G9587; ZINC35849; DTXSID00347780; HMS2712K24; ALBB-000434; BBL013760; BDBM50097098; MFCD01114913; STK386169; AKOS000121725; MCULE-8974043994; 2-[5-Chloro-2-thienyl]cinchoninic acid; SMR000369410; ST005651; VS-03988; DB-028322; FT-0730091; EN300-00851; W-7881; SR-01000597066; 2-(5-Chloro-2-thienyl)-4-quinolinecarboxylic acid; J-018944; SR-01000597066-1; 2-(5-Chloro-2-thienyl)-4-quinolinecarboxylic acid #; 4-Quinolinecarboxylic acid, 2-(5-chloro-2-thienyl)-; Z56827509
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6-chloro-8-methylquinoline-4-carboxylic acid 1H-tetrazole-5-yl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL151039; BDBM50097086; 2-(4-Bromo-phenyl)-6-chloro-8-methyl-quinoline-4-carboxylic acid 1H-tetrazol-5-yl ester
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6-sulfoquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL153066; SCHEMBL117224; BDBM50097085; 2-(4-Bromo-phenyl)-6-sulfo-quinoline-4-carboxylic acid
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Methoxyphenyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-(4-Methoxy-phenyl)-quinoline-4-carboxylic acid; 2-(4-methoxyphenyl)-4-quinolinecarboxylic acid; 4'-Methoxycinchophen; CHEMBL149961; Oprea1_106318; Oprea1_135261; SCHEMBL116026; ARONIS017295; CTK1D7649; ZINC39344; DTXSID80350277; KUC108632N; ALBB-000126; KS-00001W7J; BBL012121; BDBM50097112; MFCD00160581; SBB004431; STK007581; AKOS000121627; CCG-202937; KSC-19-181; MCULE-4252177423; NCGC00276472-01; ST056047; DB-019462; FT-0635247; L-3576; 2-(4-methoxyphenyl)-quinoline-4-carboxylic acid; 4-Quinolinecarboxylicacid, 2-(4-methoxyphenyl)-; AB01276973-01; 3Y-0940; 4-Quinolinecarboxylic acid, 2-(4-methoxyphenyl)-; AK-968/37166243; SR-01000597040; J-506050; SR-01000597040-1; F0267-4406
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-5-methyl-7-chloroquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL151769; SCHEMBL116073; BDBM50097084; 2-(4-Bromo-phenyl)-7-chloro-5-methyl-quinoline-4-carboxylic acid; 2-(4-bromophenyl)-7-chloro-5-methyl-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-7-chloro-5-methyl-
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6-(trifluoromethoxy)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL153295; SCHEMBL116058; BDBM50097113; 2-(4-Bromo-phenyl)-6-trifluoromethoxy-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-(trifluoromethoxy)-
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(Naphthalen-2-yl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-naphthalen-2-ylquinoline-4-carboxylic acid; 2-Naphthalen-2-yl-quinoline-4-carboxylic acid; 2-(2-naphthyl)quinoline-4-carboxylic acid; CHEMBL345300; 2-(2-naphthalenyl)-4-quinolinecarboxylic acid; 4-Quinolinecarboxylicacid, 2-(2-naphthalenyl)-; 4-Quinolinecarboxylic acid, 2-(2-naphthalenyl)-; C20H13NO2; PubChem6192; Oprea1_554721; Oprea1_709918; SCHEMBL117387; 2-Naphthylchinolin-4-carbonsaure; CTK0H1853; ZINC44904; DTXSID60350472; ALBB-011584; 3951AD; BBL016804; BDBM50097101; MFCD00622213; STK435043; AKOS001598328; MCULE-3605957758; VS-05583; FT-0705525; R3550; ST50908823; 2-Naphthalen-2-yl-quinoline-4-carboxylicacid; A807022
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
(3,4-Dichlorophenyl)methyl 2-(4-bromophenyl)-6-chloro-8-methyl-quinoline-4-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL345331; SCHEMBL117389; BDBM50097095; 2-(4-Bromo-phenyl)-6-chloro-8-methyl-quinoline-4-carboxylic acid 3,4-dichloro-benzyl ester; 2-(4-Bromophenyl)-6-chloro-8-methylquinoline-4-carboxylic acid 3,4-dichlorobenzyl ester; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-chloro-8-methyl-, (3,4-dichlorophenyl)methyl ester
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6-chloro-8-(hydroxymethyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL150407; SCHEMBL116064; BDBM50097109; 2-(4-Bromo-phenyl)-6-chloro-8-hydroxymethyl-quinoline-4-carboxylic acid
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6-iodo-quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL357572; SCHEMBL117405; ZINC8443064; BDBM50097082; AKOS015970429; 2-(4-Bromo-phenyl)-6-iodo-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-iodo-
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
(4-Phenylphenyl)methyl 2-(4-bromophenyl)-6-chloro-8-methyl-quinoline-4-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL153564; BDBM50097108; 2-(4-Bromo-phenyl)-6-chloro-8-methyl-quinoline-4-carboxylic acid biphenyl-4-ylmethyl ester; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-chloro-8-methyl-, [1,1'-biphenyl]-4-ylmethyl ester
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(Furan-2-yl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-Furan-2-yl-quinoline-4-carboxylic acid; 2-(2-furyl)-4-quinolinecarboxylic acid; 2-(2-furyl)quinoline-4-carboxylic acid; CC-PMLSC-DMA-P117; 2-(2-furanyl)-4-quinolinecarboxylic acid; 2-furan-2-yl-quinoline-4-carboxylic-acid; CHEMBL150924; 4-Quinolinecarboxylic acid, 2-(2-furanyl)-; SMR000069873; 2-furylcinchoninic acid; Enamine_001353; 2-(2-furyl)cinchoninic acid; MLS000061543; MLS000889043; SCHEMBL116036; cid_697640; BDBM35453; CTK1A5851; ZINC74195; HMS1397N11; HMS2217P07; HMS3334M10; ALBB-011592; CCG-1199; 6799AD; BBL013207; MFCD00092384; SBB011784; STK411135; AKOS000114785; 2-fur-2-ylquinoline-4-carboxylic acid; MCULE-6589570485; SDCCGMLS-0025966.P003; 2-(2-furyl)quinoline-4 carboxylic acid; 2-furan-2-ylquinoline-4-carboxylic acid; NCGC00055957-02; VS-03704; 2-(2-Furanyl)quinoline-4-carboxylic acid; 4-Quinolinecarboxylicacid, 2-(2-furanyl)-; AB0130041; DB-045108; ST4140007; FT-0637952; EN300-00804; L-3586; 146F252; SR-01000597065; SR-01000597065-1; BRD-K16705470-001-09-3; BRD-K16705470-001-11-9; F0267-5724
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-6,8-dimethylquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL150993; Oprea1_178464; SCHEMBL117228; CTK6B4716; ALBB-000561; ZINC4651885; BBL017513; BDBM50097088; MFCD03075244; STK449262; AKOS003295686; MCULE-6990068534; VS-06233; R6470; ST50831691; AK-968/41171788; 2-(4-bromophenyl)-6,8-dimethyl-4-quinolinecarboxylic acid; 2-(4-Bromo-phenyl)-6,8-dimethyl-quinoline-4-carboxylic acid; 2-(4-bromophenyl)-6,8-dimethyl-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6,8-dimethyl-
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(3,4-Dichlorophenyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-(3,4-Dichlorophenyl)-4-quinolinecarboxylic acid; CHEMBL150249; 4-Quinolinecarboxylicacid, 2-(3,4-dichlorophenyl)-; 2-(3,4-Dichloro-phenyl)-quinoline-4-carboxylic acid; ACMC-20duv5; Oprea1_411697; Oprea1_830927; SCHEMBL117357; CTK0G9622; ZINC69324; DTXSID10351272; 2-(3,4-DICHLORO-PHENYL)-QUINOLINE-4-CARBOXYLICACID; ALBB-000431; 4581AD; BBL016546; BDBM50097083; MFCD01414694; SBB027728; STK424517; AKOS000300926; MCULE-6021816792; KS-00001P44; NCGC00281303-01; VS-05354; ST4039566; R4528; AB01280379-01; SR-01000520462; SR-01000520462-1; 4-Quinolinecarboxylic acid, 2-(3,4-dichlorophenyl)-
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
2-(4-Bromo-phenyl)-quinoline-4-carboxylic acid; CHEMBL440534; 2-(4-bromophenyl)-4-quinolinecarboxylic acid; 2-(4-bromo-phenyl)quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-; C16H10BrNO2; NeomycinsulphateB; NSC25669; ACMC-20ctyz; PubChem5995; Oprea1_581627; Oprea1_594120; SCHEMBL116022; ARONIS017250; CTK0I3312; ZINC35846; DTXSID50282374; ZERENEX E/6110121; ALBB-000127; KS-000026AB; 7835AC; BBL002046; BDBM50097094; MFCD00160560; NSC-25669; SBB001346; STK089680; AKOS000114879; GS-6357; MCULE-2588579343; BC003083; ST005648; AB0132996; DB-040494; FT-0642547; EN300-00789; Y-9251; AK-968/37166242; SR-01000597068; SR-01000597068-1
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-[4-(Trifluoromethyl)phenyl]quinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL151890; SCHEMBL116029; CTK7I7148; BDBM50097110; 2-(4-Trifluoromethyl-phenyl)-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-[4-(trifluoromethyl)phenyl]-
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| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
Methyl 2-[[2-(4-bromophenyl)-6-chloro-8-methyl-quinoline-4-carbonyl]amino]-3-phenyl-propanoate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL434852; BDBM50097092; Phenylalanine, N-[[2-(4-bromophenyl)-6-chloro-8-methyl-4-quinolinyl]carbonyl]-, methyl ester
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
2-(4-Bromophenyl)-5,7-dichloroquinoline-4-carboxylic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL358675; SCHEMBL117257; BDBM50097091; 2-(4-Bromo-phenyl)-5,7-dichloro-quinoline-4-carboxylic acid; 2-(4-bromophenyl)-5,7-dichloro-quinoline-4-carboxylic acid; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-5,7-dichloro-
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| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Compound Name |
2-Furylmethyl 2-(4-bromophenyl)-6-chloro-8-methyl-quinoline-4-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL150266; SCHEMBL117392; BDBM50097102; 2-(4-Bromo-phenyl)-6-chloro-8-methyl-quinoline-4-carboxylic acid furan-2-ylmethyl ester; 2-(4-Bromophenyl)-6-chloro-8-methylquinoline-4-carboxylic acid 2-furanylmethyl ester; 4-Quinolinecarboxylic acid, 2-(4-bromophenyl)-6-chloro-8-methyl-, 2-furanylmethyl ester
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| Activity |
IC50 ~ 100000 nM
|
[1] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| References | Top | ||||
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| REF 1 | A series of quinoline analogues as potent inhibitors of C. albicans prolyl tRNA synthetase. Bioorg Med Chem Lett. 2001 Feb 26;11(4):541-4. | ||||
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