Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T67339 | Target Info | |||
| Target Name | Channel-activating protease 1 (CAP1) | ||||
| Synonyms |
Serine protease 8; Prostasin; CAP1
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| Target Type | Literature-reported Target | ||||
| Gene Name | PRSS8 | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 2 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Benzyl (S)-1-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-oxohexan-2-ylamino)-4-methyl-1-oxopentan-2-ylcarbamate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL509923; BDBM50246983
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| Activity |
Ki ~ 100000 nM
|
[1] | |||
| Compound Name |
Benzyl (S)-1-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-oxohexan-2-ylamino)-1-oxo-4-phenylbutan-2-ylcarbamate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL508055; BDBM50246984
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| Activity |
Ki ~ 100000 nM
|
[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Discovery of inhibitors of the channel-activating protease prostasin (CAP1/PRSS8) utilizing structure-based design. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5895-9. | ||||
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