TTD_Target_ID Target_Name TTD_Drug_ID Drug_Name Drug_Highest_Status Drug_PubchemID Molecular_Formula Molecular_Weight Canonical_SMILES Activity Binder_Type T67339 Channel-activating protease 1 B82VGZ Benzyl (S)-1-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-oxohexan-2-ylamino)-4-methyl-1-oxopentan-2-ylcarbamate Investigative 44563619 C27H34N4O5 494.6 CC(C)C[C@@H](C(=O)N[C@@H](CCCCN)C(=O)C1=NC2=CC=CC=C2O1)NC(=O)OCC3=CC=CC=C3 Ki ~ 100000 nM Poor binder T67339 Channel-activating protease 1 BISK59 Benzyl (S)-1-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-oxohexan-2-ylamino)-1-oxo-4-phenylbutan-2-ylcarbamate Investigative 44563620 C31H34N4O5 542.6 C1=CC=C(C=C1)CC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)C2=NC3=CC=CC=C3O2)NC(=O)OCC4=CC=CC=C4 Ki ~ 100000 nM Poor binder