Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
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| Target ID | T92328 | Target Info | |||
| Target Name | Ryanodine receptor 1 (RYR1) | ||||
| Synonyms |
Type 1 ryanodine receptor; Skeletal muscle-type ryanodine receptor; Skeletal muscle ryanodine receptor; Skeletal muscle calcium release channel; RyR1; RyR; RYR-1; RYDR; Cardiac muscleryanodine receptor-calcium release channel; Cardiac muscle-type ryanodine receptor; Brain-type ryanodine receptor; Brain ryanodine receptor-calcium release channel
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| Target Type | Discontinued Target | ||||
| Gene Name | RYR1 | ||||
| Biochemical Class | Ryanodine-inositol 1,4,5-triphosphate receptor calcium channel | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 1 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Bastadin-19
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL506286; (E,E)-Bastadin-19
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| Activity |
EC50 ~ 100000 nM
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[1] | |||
| References | Top | ||||
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| REF 1 | Open-chain half-bastadins mimic the effects of cyclic bastadins on calcium homeostasis in cultured neurons. Bioorg Med Chem Lett. 2008 Nov 1;18(21):5734-7. | ||||
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