Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T90682 | Target Info | |||
| Target Name | GABA(A) receptor rho2 (GABRR2) | ||||
| Synonyms |
Gamma-aminobutyric acid receptor subunit rho-2; GABA(C) receptor2; GABA(A) receptor subunit rho-2
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| Target Type | Literature-reported Target | ||||
| Gene Name | GABRR2 | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 2 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
CACA
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Investigative | Compound Info | ||
| Synonyms |
cis-aminocrotonic acid; 4-aminocrotonic acid
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| Activity |
EC50 = 70000 nM
|
[1] | |||
| Compound Name |
4-Amino-2-methylbut-2-enoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL284115; 2-MeTACA; SCHEMBL22214; SCHEMBL17438080; BDBM50087274; AKOS006341839; (E)-2-Methyl-4-amino-2-butenoic acid; (E)-4-amino-2-methylbut-2-enoic acid; trans-4-amino-2-methylbut-2-enoic acid; 4-Amino-2-methyl-but-2-enoic acid (2-MeTACA)
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| Activity |
EC50 = 101000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology. J Med Chem. 2000 Apr 20;43(8):1427-47. | ||||
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