Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T72319 | Target Info | |||
| Target Name | Chromobox protein homolog 7 (CBX7) | ||||
| Synonyms |
Chromobox 7
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|
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| Target Type | Literature-reported Target | ||||
| Gene Name | CBX7 | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 35 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(2-bicyclo[2.2.1]heptanylamino)hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3932467; BDBM50194427
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|
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| Activity |
IC50 = 51000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(dimethylamino)hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3954152; BDBM50194431
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|
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| Activity |
IC50 = 51000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-pyrrolidin-1-ylhexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3945426; BDBM50194249
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|
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| Activity |
IC50 = 53000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234154; BDBM50009472
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|
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| Activity |
IC50 = 53000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[[2-[(4-carboxyphenyl)sulfonylamino]acetyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234185; BDBM50009503
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|
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| Activity |
IC50 = 53000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-benzamidopropanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234173; BDBM50009491
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|
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| Activity |
IC50 = 57000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(4-methoxycarbonylphenyl)sulfonylamino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234439; BDBM50009524
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|
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| Activity |
IC50 = 57000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234179; BDBM50009497
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|
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| Activity |
IC50 = 58000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234181; BDBM50009499
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|
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| Activity |
IC50 = 58000 nM
|
[2] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-6-[azetidin-3-yl(methyl)amino]-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3918626; BDBM50194467
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(cyclohexylamino)hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3906755; BDBM50194426
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-Benzamidopropanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-3-hydroxy-1-methoxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3965363; BDBM50194472
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(cyclopentylamino)hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3907836; BDBM50194478
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[[[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-Benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-3-hydroxy-1-methoxy-1-oxopropan-2-yl]amino]-6-oxohexyl]amino]-(dimethylamino)methylidene]-dimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3946489; BDBM50194253
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-6-(2-adamantylamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3982833; BDBM50194470
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-Benzamidoacetyl)-methylamino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-3-hydroxy-1-methoxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3963110; BDBM50194386
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(propan-2-ylamino)hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3978346; BDBM50194388
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-6-[acetyl(2-bicyclo[2.2.1]heptanyl)amino]-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3922982; BDBM50194252
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-6-(1-azabicyclo[2.2.2]octan-3-ylamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3908012; BDBM50194254
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-Benzamidopropanoyl]amino]-4-methylpentanoyl]amino]-6-(methylamino)-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3942638; BDBM50194460
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-Benzamidoacetyl)amino]-3-phenylpropanoyl]-methylamino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-3-hydroxy-1-methoxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3951389; BDBM50194356
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Benzamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]pentyl-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3898819; BDBM50194464
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
Methyl (2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-benzamidoacetyl)amino]-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoate
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3916833; BDBM50194459
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|
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| Activity |
IC50 ~ 60000 nM
|
[1] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234141; BDBM50009459
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|
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| Activity |
IC50 = 62000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-3,3-dimethylbutanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234139; BDBM50009457
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|
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| Activity |
IC50 = 67000 nM
|
[2] | |||
| Compound Name |
1-[4-(2,3-Dimethoxybenzoyl)piperazin-1-yl]-2-(3-methylphenoxy)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
MS37452; CHEMBL3827954; 1-(2,3-dimethoxybenzoyl)-4-[(3-methylphenoxy)acetyl]piperazine; 1-[4-(2,3-Dimethoxybenzoyl)-1-piperazinyl]-2-(3-methylphenoxy)-ethanone; Oprea1_185108; SCHEMBL20013899; AOB5774; ZINC779542; BDBM50189780; STK146391; AKOS000551086; MCULE-7891456476; NCGC00402347-02; AS-16919; MS37452, >=98% (HPLC); AT-057/43316446; Q27454416; 1-(4-(2,3-Dimethoxybenzoyl)piperazin-1-yl)-2-(m-tolyloxy)ethanone; 1-{4-[(2,3-dimethoxyphenyl)carbonyl]piperazin-1-yl}-2-(3-methylphenoxy)ethanone
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|
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| Activity |
IC50 = 67000 nM
|
[3] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-(1H-indole-3-carbonylamino)propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234178; BDBM50009496
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|
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| Activity |
IC50 = 67000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234145; 4mn3; BDBM50009463
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|
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| Activity |
IC50 = 73000 nM
|
[4] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(1R)-1-carboxy-2-hydroxyethyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234158; BDBM50009476
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|
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| Activity |
IC50 = 79000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[[2-(2-bromophenyl)acetyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234176; BDBM50009494
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|
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| Activity |
IC50 = 89000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-(pyridine-3-carbonylamino)propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234174; BDBM50009492
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|
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| Activity |
IC50 = 91000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-[[2-[(2-phenylacetyl)amino]acetyl]amino]propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234180; BDBM50009498
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|
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| Activity |
IC50 = 100000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxo-6-(propylamino)hexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234165; BDBM50009483
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|
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| Activity |
IC50 = 102000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethylamino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234169; BDBM50009487
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|
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| Activity |
IC50 = 105000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]hexanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234153; BDBM50009471
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| Activity |
IC50 = 120000 nM
|
[2] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 11 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[1-(hydroxymethyl)cyclopentyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234163; BDBM50009481
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[(1-hydroxy-3-methylbutan-2-yl)amino]-6-oxohexyl]-trimethylazanium
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234160; BDBM50009478
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-[[(2S)-2-[(4-methylphenyl)sulfonylamino]-3-phenylpropanoyl]amino]propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234437; BDBM50009522
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[(4-methoxyphenyl)sulfonylamino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234182; BDBM50009500
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-[[(1S,2S)-2-hydroxycyclohexyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234162; BDBM50009480
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-4-methyl-2-[[(2S)-2-(pyridin-3-ylsulfonylamino)propanoyl]amino]pentanoyl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234183; BDBM50009501
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|
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| Activity |
IC50 > 250000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]-6-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]amino]-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234155; BDBM50009473
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|
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| Activity |
IC50 > 500000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-6-(1-hydroxypentan-2-ylamino)-6-oxohexyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234161; BDBM50009479
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|
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| Activity |
IC50 > 500000 nM
|
[2] | |||
| Compound Name |
[(5S)-5-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-phenylpropanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-5-carboxypentyl]-trimethylazanium
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234159; BDBM50009477
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| Activity |
IC50 = 560000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-(benzylamino)propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234187; BDBM50009507
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| Activity |
IC50 > 2000000 nM
|
[2] | |||
| Compound Name |
[(5S)-6-[[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]amino]-5-[[(2S)-2-[[(2S)-2-[(4-carboxyphenyl)methylamino]propanoyl]amino]-4-methylpentanoyl]amino]-6-oxohexyl]-trimethylazanium
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3234186; BDBM50009504
Click to Show/Hide
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| Activity |
IC50 > 2000000 nM
|
[2] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Structure-Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains. J Med Chem. 2016 Oct 13;59(19):8913-8923. | ||||
| REF 2 | Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7). J Med Chem. 2014 Apr 10;57(7):2874-83. | ||||
| REF 3 | Methyllysine binding domains: Structural insight and small molecule probe development. Eur J Med Chem. 2017 Aug 18;136:14-35. | ||||
| REF 4 | Selective Inhibition of CBX6: A Methyllysine Reader Protein in the Polycomb Family. ACS Med Chem Lett. 2015 Dec 7;7(2):139-44. | ||||
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