Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T60182 | Target Info | |||
| Target Name | Glucagon receptor (GCGR) | ||||
| Synonyms |
GLR; GL-R
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| Target Type | Successful Target | ||||
| Gene Name | GCGR | ||||
| Biochemical Class | GPCR secretin | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 33 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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Investigative | Compound Info | ||
| Synonyms |
GSK137647A; GSK 137647; GSK-137647A; N-mesityl-4-methoxybenzenesulfonamide; CHEMBL3311308; MFCD02007969; 4-methoxy-N-(2,4,6-trimethylphenyl)-benzenesulfonamide; CBMicro_012617; Oprea1_349531; Oprea1_545891; SCHEMBL19357604; KS-00000TIW; AOB2991; ZINC184126; BCP17136; EX-A1097; GSK 137647A; SMSF0014079; BDBM50044849; STK899558; AKOS003261220; CB15818; CS-5549; GSK-137647; MCULE-5583867808; N-mesityl-4-methoxy-1-benzenesulfonamide; NCGC00387253-02; NCGC00387253-05; AK240703; AS-16737; HY-19995; BIM-0012523.P001; FFA4 (GPR120) agonist GSK137647A; B7793; EU-0076636; FT-0700296; S0001; ST50719559; GSK137647A, >=98% (HPLC); A14542; AJ-292/14925630; SR-01000478738; J-690285; SR-01000478738-1; [(4-methoxyphenyl)sulfonyl](2,4,6-trimethylphenyl)amine; 4-methoxy-N-(2,4,6-trimethylphenyl)benzene-1-sulfonamide; 4-Methoxy-N-(2,4,6-triMethylphenyl)benzenesulfonaMide, 97%
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| Activity |
EC50 ~ 50118.72 nM
|
[1] | |||
| Compound Name |
Naphthalen-1-yl-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-methanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL208053; BDBM50183181
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| Activity |
IC50 = 55000 nM
|
[2] | |||
| Compound Name |
1-(3,4-Dihydroxy-phenyl)-2-(5-phenyl-4H-[1,2,4]triazol-3-ylsulfanyl)-ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
MLS000074715; CHEMBL358546; SMR000011758; cid_654283; SCHEMBL13856448; BDBM32012; HMS2471L17; ZINC4373918; STK927379; AKOS000563318; MCULE-4509748009; 1-(3,4-dihydroxyphenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone; MLS-0029227.0001; SR-01000365237; SR-01000365237-1; 1-(3,4-Dihydroxyphenyl)-2-(5-phenyl-4H-1,2,4-triazole-3-ylthio)ethanone; 1-(3,4-dihydroxyphenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)thio]ethanone; 1-(3,4-dihydroxyphenyl)-2-[(5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethanone
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| Activity |
Ki = 55000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(5-nitro-1H-benzimidazole-2-ylthio)ethanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL147331; BDBM50068633; ZINC13782380; MCULE-5371844577; AI-204/36888010; 1-(3,4-Dihydroxy-phenyl)-2-(5-nitro-1H-benzoimidazol-2-ylsulfanyl)-ethanone; 1-(3,4-dihydroxyphenyl)-2-({5-nitro-1H-benzimidazol-2-yl}sulfanyl)ethanone
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| Activity |
Ki = 55000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzimidazol-2-ylsulfanyl)-1-(4-hydroxyphenyl)ethanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL149123; Oprea1_043471; ZINC41757; BDBM50068630; STK926148; AKOS002232648; MCULE-3131406309; ST50750526; SR-01000004910; SR-01000004910-1; 2-benzimidazol-2-ylthio-1-(4-hydroxyphenyl)ethan-1-one; 1-(4-Hydroxyphenyl)-2-(1H-benzimidazole-2-ylthio)ethanone; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(4-hydroxy-phenyl)-ethanone
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| Activity |
Ki ~ 60000 nM
|
[3] | |||
| Compound Name |
3-Chloro-4-hydroxy-5-methoxy-benzoic acid(4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL106058; BDBM50104097
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|
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| Activity |
IC50 = 60000 nM
|
[4] | |||
| Compound Name |
3-[[1-[3-(3,5-Dichlorophenyl)-5-(furan-2-yl)pyrazol-1-yl]-2,3-dihydro-1H-indene-5-carbonyl]amino]propanoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL3799656; BDBM50168095
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| Activity |
IC50 = 71800 nM
|
[5] | |||
| Compound Name |
2-(1,3-Benzothiazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL148905; SCHEMBL3466913; cid_4066568; ZINC5629194; BDBM50068618; AKOS008906931; MCULE-4144107356; ST51025483; MLS-0315885.0001; AI-204/31680049; 1-(3,4-Dihydroxyphenyl)-2-(benzothiazole-2-ylthio)ethanone; 2-benzothiazol-2-ylthio-1-(3,4-dihydroxyphenyl)ethan-1-one; 2-(Benzothiazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-ethanone
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| Activity |
Ki = 73000 nM
|
[3] | |||
| Compound Name |
2-Chloro-4-[1-[4-(4-isopropylbenzyloxy)-3,5-dimethoxyphenyl]-(E)-methylideneaminosulfonamido]phenol
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL158886; SCHEMBL2664178; BDBM50110061
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|
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| Activity |
IC50 = 78300 nM
|
[6] | |||
| Compound Name |
3-[[[2-[2-(3,4-Dihydroxyphenyl)-2-oxoethylthio]-1H-benzimidazole-5-yl]oxy]methyl]benzoic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL149138; BDBM50068617; 3-{2-[2-(3,4-Dihydroxy-phenyl)-2-oxo-ethylsulfanyl]-1H-benzoimidazol-5-yloxymethyl}-benzoic acid
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| Activity |
Ki = 95000 nM
|
[3] | |||
| Compound Name |
4-(4-Hydroxy-naphthalen-1-ylmethylene-hydrazinocarbonyl)-benzoic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL322713; BDBM50104078
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (4-hydroxy-benzylidene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL107138; BDBM50104101
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (3-hydroxy-4-methoxy-benzylidene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL106738; BDBM50104074
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
3-Methoxy-benzoic acid (4-methoxy-naphthalen-1-ylmethylene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL107527; BDBM50104067
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Amino-benzoic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL320634; BDBM50104100
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
N'-[(E)-(4-Hydroxy-3-methoxyphenyl)methylidene]naphthalene-1-carbohydrazide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL419729; BDBM50104095; STK401646; ZINC32609432; AKOS003237913; ST50910897; N-[(1E)-2-(4-hydroxy-3-methoxyphenyl)-1-azavinyl]naphthylcarboxamide; Naphthalene-1-carboxylic acid (4-hydroxy-3-methoxy-benzylidene)-hydrazide
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
N-[(E)-(2,4-Dioxo-1H-pyrimidin-5-yl)methylideneamino]-4-hydroxy-3-methoxybenzamide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL107045; BDBM50104075; 4-Hydroxy-3-methoxy-benzoic acid (2,4-dioxo-1,2,3,4-tetrahydro-pyrimidin-5-ylmethylene)-hydrazide
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (1-naphthalen-1-yl-ethylidene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL430509; BDBM50104092
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-benzoic acid N''-naphthalen-1-ylmethyl-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL321461; BDBM50104065; ZINC13864079
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (4-methoxy-benzylidene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL419181; BDBM50104062
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-N-[(E)-(4-hydroxynaphthalen-1-yl)methylideneamino]-3-(morpholin-4-ylmethyl)benzamide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL107481; BDBM50104070; 4-Hydroxy-3-morpholin-4-ylmethyl-benzoic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
1H-Indole-5-carboxylic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL107480; BDBM50104084
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (5-methyl-1H-imidazol-4-ylmethylene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL439961; BDBM50104072
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
Quinoxaline-6-carboxylic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL107484; BDBM50104076
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
6-Hydroxy-nicotinic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL106950; BDBM50104090
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
5-Hydroxy-1H-indole-2-carboxylic acid (4-hydroxy-naphthalen-1-ylmethylene)-hydrazide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL108177; BDBM50104098
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
3-Chloro-N-[(E)-1-[3,5-dimethoxy-4-[(4-propan-2-ylphenyl)methoxy]phenyl]ethylideneamino]-4-hydroxybenzamide
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL160521; BDBM50110075
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|
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| Activity |
IC50 ~ 100000 nM
|
[6] | |||
| Compound Name |
4-Hydroxy-3-methoxy-benzoic acid (4-styryl-benzylidene)-hydrazide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL431650; BDBM50104085
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|
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| Activity |
IC50 ~ 100000 nM
|
[4] | |||
| Compound Name |
1-[4-[1-[3-(3,5-Dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]piperidine-3-carboxylic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3798731; BDBM50168083
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|
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| Activity |
IC50 = 112200 nM
|
[5] | |||
| Compound Name |
1-[4-[1-[3-(3,5-Dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]pyrrolidine-3-carboxylic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3798548; BDBM50168084
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|
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| Activity |
IC50 = 131100 nM
|
[5] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(quinoline-2-ylthio)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL147634; BDBM50068634; 1-(3,4-Dihydroxy-phenyl)-2-(quinolin-2-ylsulfanyl)-ethanone
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|
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| Activity |
Ki = 160000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(4,5-diphenyl-1H-imidazole-2-ylthio)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL359177; BDBM50068637; 1-(3,4-Dihydroxy-phenyl)-2-(4,5-diphenyl-1H-imidazol-2-ylsulfanyl)-ethanone
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| Activity |
Ki = 180000 nM
|
[3] | |||
| Compound Name |
5-[(1H-Benzimidazole-2-ylthio)acetyl]-2-hydroxybenzoic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL148045; BDBM50068643; 5-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-2-hydroxy-benzoic acid
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| Activity |
Ki = 200000 nM
|
[3] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 15 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(benzoxazole-2-ylthio)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL148645; cid_4450383; ZINC5628740; BDBM50068635; AKOS001297585; MCULE-8537204386; UPCMLD0ENAT5731231:001; ST51025484; MLS-0315886.0001; Z19651549; 2-benzoxazol-2-ylthio-1-(3,4-dihydroxyphenyl)ethan-1-one; 2-(Benzooxazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-ethanone; 2-(1,3-benzoxazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethan-1-one
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|
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| Activity |
Ki = 250000 nM
|
[3] | |||
| Compound Name |
1-(3-Hydroxyphenyl)-2-(1H-benzimidazole-2-ylthio)ethanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL147173; BDBM50068628; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-hydroxy-phenyl)-ethanone
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| Activity |
Ki = 380000 nM
|
[3] | |||
| Compound Name |
3-[(1H-Benzimidazole-2-ylthio)acetyl]benzoic acid
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL148750; BDBM50068625; 3-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzoic acid
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(1H-imidazole-2-ylthio)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL357318; BDBM50068623; 1-(3,4-Dihydroxy-phenyl)-2-(1H-imidazol-2-ylsulfanyl)-ethanone
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzimidazol-2-ylsulfanyl)-1-(3,4-dimethoxyphenyl)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL147177; Oprea1_067342; Oprea1_584943; ZINC344642; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dimethoxy-phenyl)-ethanone; BDBM50068615; STK859647; AKOS000560262; MCULE-2409209260; 1-(3,4-Dimethoxyphenyl)-2-(1H-benzimidazole-2-ylthio)ethanone
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
4-[2-(1H-Benzoimidazol-2-ylsulfanyl)-1-hydroxy-ethyl]-2-chloro-phenol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL347544; BDBM50068613; 1-(3-Chloro-4-hydroxyphenyl)-2-(1H-benzimidazole-2-ylthio)ethanol
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxy-phenyl)-ethanone O-methyl-oxime
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL146374; BDBM50068624
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-4-(1H-benzimidazole-2-ylthio)-1-butanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL146545; BDBM50068622; 4-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-butan-1-one
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzimidazol-2-ylsulfanyl)-1-phenylethanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL147345; 2-((1H-benzo[d]imidazol-2-yl)thio)-1-phenylethanone; Enamine_000106; 2-phenacylthiobenzimid-azole; CBDivE_001158; CBDivE_002748; CBDivE_004649; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-phenyl-ethanone; ZINC50018; BBL001876; BDBM50068642; MFCD00226073; STK325626; AKOS000666762; Benzimidazole, 2-(benzoylmethylthio)-; MCULE-3370650931; ST066964; 2-benzimidazol-2-ylthio-1-phenylethan-1-one; 10.14272/NRCVVKRZQAPHQO-UHFFFAOYSA-N; 1-Phenyl-2-(1H-benzimidazole-2-ylthio)ethanone; doi:10.14272/NRCVVKRZQAPHQO-UHFFFAOYSA-N; SR-01000508660; 2(1-H-Benzimidazol-2-yl-sulfanyl)-1-phenylethanone; Ethanone, 2-(1H-benzimidazol-2-ylthio)-1-phenyl-; SR-01000508660-1; 2-(1H-Benzimidazol-2-ylsulfanyl)-1-phenylethanone #; 2-[(1H-Benzimidazol-2-yl)sulfanyl]-1-phenylethanone; F0081-0093
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|
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dichlorophenyl)-2-(1H-benzimidazole-2-ylthio)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL342535; CBDivE_002609; ZINC192237; BDBM50068621; AKOS003625587; MCULE-1879545196; AB00074173-01; F0017-0025; 2-((1H-benzo[d]imidazol-2-yl)thio)-1-(3,4-dichlorophenyl)ethanone; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dichloro-phenyl)-ethanone
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(1-methyl-1H-benzimidazole-2-ylthio)ethanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL147679; BDBM50068640; 2-(3,4-dihydroxyphenacylthio)-1-methylbenzimidazole; 1-(3,4-Dihydroxy-phenyl)-2-(1-methyl-1H-benzoimidazol-2-ylsulfanyl)-ethanone
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
4-[(1H-Benzimidazole-2-ylthio)acetyl]benzoic acid
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL146181; BDBM50068629; 4-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzoic acid
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzimidazol-2-ylsulfanyl)-1-(3,5-dihydroxyphenyl)ethanone
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2112026; BDBM50408685
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|
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxy-phenyl)-ethanone O-benzyl-oxime
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL149067; BDBM50068632
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|
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| Activity |
Ki > 500000 nM
|
[3] | |||
| Compound Name |
1-(3,4-Dihydroxyphenyl)-2-(1H-benzimidazol-2-ylthio)-1-pentanone
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL146399; BDBM50068619; 2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-pentan-1-one
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| Activity |
Ki > 500000 nM
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[3] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
| References | Top | ||||
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| REF 1 | Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120). Bioorg Med Chem Lett. 2014 Jul 15;24(14):3100-3. | ||||
| REF 2 | Novel substituted naphthalen-1-yl-methanone derivatives as anti-hyperglycemic agents. Bioorg Med Chem Lett. 2006 May 15;16(10):2719-23. | ||||
| REF 3 | Discovery and structure-activity relationship of the first non-peptide competitive human glucagon receptor antagonists. J Med Chem. 1998 Dec 17;41(26):5150-7. | ||||
| REF 4 | Identification of alkylidene hydrazides as glucagon receptor antagonists. J Med Chem. 2001 Sep 13;44(19):3141-9. | ||||
| REF 5 | Design, synthesis, structure-activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists. Bioorg Med Chem. 2016 Jun 15;24(12):2852-63. | ||||
| REF 6 | Human glucagon receptor antagonists based on alkylidene hydrazides. Bioorg Med Chem Lett. 2002 Feb 25;12(4):663-6. | ||||
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