Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T58970 | Target Info | |||
| Target Name | Extracellular signal-regulated kinase 2 (ERK2) | ||||
| Synonyms |
PRKM2; PRKM1; P42-MAPK; P42 Mitogen-activated protein kinase; Mitogen-activated protein kinase 2; Mitogen-activated protein kinase 1; MAPK 2; MAPK 1; MAP kinase isoform p42; MAP kinase 2; MAP kinase 1; ERT1; ERK-2
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| Target Type | Clinical trial Target | ||||
| Gene Name | MAPK1 | ||||
| Biochemical Class | Kinase | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 136 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Niclosamide
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Approved | Compound Info | ||
| Synonyms |
niclosamide; 50-65-7; Niclocide; 5-Chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxybenzamide; Tredemine; Bayluscid; Phenasal; Yomesan; Fenasal; Dichlosale; Helmiantin; Sagimid; Iomezan; Devermine; Atenase; Vermitid; Radeverm; Mansonil; Iomesan; Devermin; Cestocid; Sulqui; Lintex; Nasemo; Mato; Fedal-Telmin; Bayer 73; Radewerm; Zestocarp; Bayer 2353; 2',5-Dichloro-4'-nitrosalicylanilide; Chemagro 2353; BAY 2353; Benzamide, 5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxy-; 5-Chloro-2'-chloro-4'-nitrosalicylanilide; nicolsamide; HL 2447; Niclosamidum [I
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| Compound Name |
PMID25991433-Compound-P6
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Patented | Compound Info | ||
| Activity |
IC50 ~ 50000 nM
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[2] | |||
| Compound Name |
PMID25991433-Compound-P5
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Patented | Compound Info | ||
| Activity |
IC50 ~ 50000 nM
|
[3] | |||
| Compound Name |
XHPNYYOUZWOWNT-PYUWXLGESA-N
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Patented | Compound Info | ||
| Synonyms |
CHEMBL1922122; SCHEMBL3855548; XHPNYYOUZWOWNT-PYUWXLGESA-N; BDBM50358223; US8846696, (3RS,4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol; (3RS,4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol; (3RS, 4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol
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| Activity |
IC50 = 51000 nM
|
[4] | |||
| Compound Name |
AGGGWZCOULSEER-PYUWXLGESA-N
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Patented | Compound Info | ||
| Synonyms |
CHEMBL1922121; SCHEMBL3858001; AGGGWZCOULSEER-PYUWXLGESA-N; BDBM50358222; (3RS,4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol; US8846696, (3RS,4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol; (3RS, 4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol
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| Activity |
IC50 = 111000 nM
|
[4] | |||
| Compound Name |
JNJ-10198409
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Investigative | Compound Info | ||
| Synonyms |
JNJ-10198409; 627518-40-5; PDGFR Tyrosine Kinase Inhibitor IV; PDGF Receptor Tyrosine Kinase Inhibitor IV; CHEMBL120077; N-(3-fluorophenyl)-6,7-dimethoxy-1,4-dihydroindeno[1,2-c]pyrazol-3-amine; 3-Fluoro-N-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamine; ZDNURMVOKAERHZ-UHFFFAOYSA-N; SCHEMBL3088170; GTPL6020; CTK8E8807; jnj10198409; DTXSID70430890; MolPort-009-019-131; HMS3650O03; HMS3229I11; ZINC13677843; BDBM50179207; AKOS030525202; RWJ 540973; CCG-206773; NCGC00343986-02; RT-014973; KB-274227; SR-01000946814
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| Activity |
IC50 ~ 100000 nM
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[5] | |||
| Compound Name |
3-{[2-(3-Thienyl)pyridin-4-yl]amino}-4-{[(1R)-1-phenylethyl]amino}cyclobut-3-ene-1,2-dione
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL481248; BDBM50259638
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| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(2-(thiazol-2-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644627; BDBM50333991
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
N-[4-Bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(6,7-difluoro-2-oxoquinolin-1-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1822145; SCHEMBL3783987; US9796706, Compound 44; BDBM351600; BDBM50352614; n-(4-bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(6,7-difluoro-2-oxoquinolin-1(2h)-yl)acetamide
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| Activity |
IC50 ~ 50000 nM
|
[3] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644617; BDBM50334009
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
N-(4,4''-Bithiazol-5-yl)-2-(isoquinolin-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288160; SCHEMBL3713725; BDBM50332091; 2-isoquinolin-5-yl-N-[4-(1,3-thiazol-4-yl)-1,3-thiazol-5-yl]acetamide
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
CID 46179972
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1163016; BDBM50378568
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| Activity |
IC50 ~ 50000 nM
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[9] | |||
| Compound Name |
4-(6-Bromonaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644634; BDBM50334002
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
N-[4-Cyano-3-(1h-1,2,4-Triazol-5-Yl)thiophen-2-Yl]-2-(2-Oxo-3,4-Dihydroquinolin-1(2h)-Yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682015; SCHEMBL3784549; US9796706, Compound 36; BDBM351592; BDBM50338293; Q27453534
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| Activity |
IC50 ~ 50000 nM
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[2] | |||
| Compound Name |
3-(5-Chloro-2-{[1-(dimethylamino)propan-2-yl]oxy}phenyl)-1-(5-cyanopyrazin-2-yl)urea
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Investigative | Compound Info | ||
| Synonyms |
urea-based inhibitor 2d; A-690002; CHEMBL425904; SCHEMBL5865729; BDBM14829; 1-[5-chloro-2-[1-(dimethylamino)propan-2-yloxy]phenyl]-3-(5-cyanopyrazin-2-yl)urea; (+/-)1-[5-Chloro-2-(2-dimethylamino-1-methyl-ethyloxy)-phenyl]-3-(5-cyano-pyrazin-2-yl)-urea
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| Activity |
IC50 ~ 50000 nM
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[10] | |||
| Compound Name |
Methyl 4-(6-(4-(methoxycarbonylamino)phenyl)-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
WYE-354; WYE 354; pyrazolo pyrimidine, 19; cc-506; MLS006011008; SCHEMBL300431; CHEMBL561708; GTPL9361; WYE354; BDBM35587; DTXSID00657912; C24H29N7O5; HMS3654N09; BCP02898; ZINC43013490; CCG-264882; CS-0183; SB19260; NCGC00242484-01; NCGC00242484-02; NCGC00242484-09; AC-28454; AS-55957; HY-12034; SMR004702806; BCP0726000260; DB-059456; FT-0675866; S1266; SW219671-1; X7422; W-5702; J-001552; J-514253; BRD-K77008974-001-01-6; Q27166532; mTOR Kinase Inhibitor II, WYE-354 - CAS 1062169-56-5
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| Activity |
IC50 ~ 50000 nM
|
[11] | |||
| Compound Name |
Schembl22388257
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1822151; SCHEMBL3780453; BDBM351666; US9796706, Compound 110; BDBM50352620; N-(4-bromo-3-(1H-1,2,4-triazol-3-yl)thiophen-2-yl)-2-(6-cyano-2-oxoquinolin-1(2H)-yl)acetamide; n-(4-bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(6-cyano-2-oxoquinolin-1(2h)-yl)acetamide; N-[4-bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(6-cyano-2-oxoquinolin-1-yl)acetamide
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| Activity |
IC50 ~ 50000 nM
|
[3] | |||
| Compound Name |
Methyl 4-(6-(4-aminophenyl)-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1095626; SCHEMBL3984085; BDBM50316252; methyl 4-[6-(4-aminophenyl)-4-morpholin-4-ylpyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carboxylate
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| Activity |
IC50 ~ 50000 nM
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[12] | |||
| Compound Name |
2-(Isoquinolin-5-yl)-n-(4-(1-methyl-1h-1,2,4-triazol-5-yl)thiazol-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288129; SCHEMBL3783552; BDBM50332089; 2-isoquinolin-5-yl-N-[4-(2-methyl-1,2,4-triazol-3-yl)-1,3-thiazol-5-yl]acetamide
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
5-Vinyl-3-pyridinecarbonitrile, 19
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL606245; BDBM35137
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| Activity |
IC50 ~ 50000 nM
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[13] | |||
| Compound Name |
4-(4-Methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1080994; SCHEMBL2934634; BDBM50311953
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| Activity |
IC50 ~ 50000 nM
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[14] | |||
| Compound Name |
4-(8-Aminonaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644636; BDBM50334004
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
2-Quinolin-5-yl-N-[2-(1H-1,2,4-triazol-5-yl)thiophen-3-yl]acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288099; SCHEMBL3777866; US9796706, Compound 25; BDBM351581; BDBM50332085; n-(2-(1h-1,2,4-triazol-5-yl)thiophen-3-yl)-2-(quinolin-5-yl)acetamide; N-(2-(4H-1,2,4-triazol-3-yl)thiophen-3-yl)-2-(quinolin-5-yl)acetamide
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
2-(Isoquinolin-5-yl)-n-(4-(pyrazin-2-yl)thiazol-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288159; SCHEMBL3713088; BDBM50332090; 2-isoquinolin-5-yl-N-(4-pyrazin-2-yl-1,3-thiazol-5-yl)acetamide
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
Methyl 4-(2-(naphthalen-1-yl)acetamido)-1H-pyrazole-3-carboxylate
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1287886; BDBM50332065
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
N-(2-(5-Amino-1H-1,2,4-triazol-3-yl)thiophen-3-yl)-2-(4-methoxyphenyl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288039; n-(2-(3-amino-1h-1,2,4-triazol-5-yl)thiophen-3-yl)-2-(4-methoxyphenyl)acetamide; N-[2-(3-amino-1H-1,2,4-triazol-5-yl)thiophen-3-yl]-2-(4-methoxyphenyl)acetamide; SCHEMBL3788513; US9796706, Compound 17; BDBM351573; BDBM50332080
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| Activity |
IC50 ~ 50000 nM
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[8] | |||
| Compound Name |
4-(8-Fluoronaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644635; BDBM50333998
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
3-(2-(Cyclohexylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1-(pyridin-4-ylmethyl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644642; BDBM50333980
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
N-(4-Cyano-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(isoquinolin-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682018; SCHEMBL3781602; US9796706, Compound 35; BDBM351591; BDBM50338264; N-[4-cyano-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-isoquinolin-5-ylacetamide
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| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
3-(2-(Cyclohexylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644618; BDBM50334008
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
6-Chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4H-pyrazolo[3,4-B]quinolin-4-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL207228; 9-hydroxy pyrazoloquinolinone 1; SCHEMBL21067944; BDBM15868; 6-chloro-9-hydroxy-1,3-dimethyl-1H,4H,9H-pyrazolo[3,4-b]quinolin-4-one; DB07218; Q27096139; 1,3-Dimethyl-6-chloro-9-hydroxy-1H-pyrazolo[3,4-b]quinoline-4(9H)-one
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| Activity |
IC50 ~ 50000 nM
|
[15] | |||
| Compound Name |
N-[4-(4-Naphthalen-2-yl-5-oxo-1H-1,2,4-triazol-3-yl)pyridin-2-yl]acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644629; BDBM50333999; N-(4-(4-(naphthalen-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)pyridin-2-yl)acetamide
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
4-(4-Methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrolidin-1-yl)prop-1-enyl)thieno[2,3-b]pyridine-5-carbonitrile
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL477817; SCHEMBL5520662; SCHEMBL5520668; BDBM50263132
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| Activity |
IC50 ~ 50000 nM
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[16] | |||
| Compound Name |
3-{5-Chloro-2-[(3-methyloxetan-3-yl)methoxy]phenyl}-1-(5-cyanopyrazin-2-yl)urea
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Investigative | Compound Info | ||
| Synonyms |
urea-based inhibitor 2e; A-641397; CHEMBL192161; BDBM14830; (+/-)1-[5-Chloro-2-(3-methyl-oxetan-3-ylmethoxy)-phenyl]-3-(5-cyano-pyrazin-2-yl)-urea
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| Activity |
IC50 ~ 50000 nM
|
[10] | |||
| Compound Name |
3-(2-(Cyclohexylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644638; BDBM50334000
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
N-[4-(4-Naphthalen-2-yl-5-oxo-1H-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644631; BDBM50334005; N-(4-(4-(naphthalen-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)pyridin-2-yl)benzamide
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| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
4-(6-Aminonaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644633; BDBM50334006
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| Activity |
IC50 ~ 50000 nM
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[7] | |||
| Compound Name |
n-(4-Bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(isoquinolin-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682016; SCHEMBL3783151; US9796706, Compound 32; BDBM351588; BDBM50338262; N-[4-bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-isoquinolin-5-ylacetamide
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| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644620; BDBM50333994
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| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
3-(7-(4-((1S,4S)-5-Methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)-2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl)phenol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1087650; SCHEMBL1015620; BDBM50311985
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| Activity |
IC50 ~ 50000 nM
|
[17] | |||
| Compound Name |
n-(4-Bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682013; SCHEMBL3780403; US9796706, Compound 34; BDBM351590; BDBM50338291; N-[4-bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1-yl)acetamide
Click to Show/Hide
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| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
n-(4-Methyl-3-(3-methyl-1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(quinolin-5-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682010; SCHEMBL3782459; US9796706, Compound 26; BDBM351582; BDBM50338287; N-[4-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)thiophen-2-yl]-2-quinolin-5-ylacetamide
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| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
2-(4-Methoxyphenyl)-N-(2-(5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl)thiophen-3-yl)acetamide
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288038; 2-(4-methoxyphenyl)-N-[2-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]thiophen-3-yl]acetamide; SCHEMBL2229021; US9796706, Compound 13; BDBM351569; BDBM50332079; 2-(4-methoxyphenyl)-n-(2-(3-(trifluoromethyl)-1h-1,2,4-triazol-5-yl)thiophen-3-yl)acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
3-[4-(4-Hydroxyphenyl)phenyl]-N-(pyridin-4-ylmethyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL242753; SCHEMBL6794625; BDBM50204693
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[18] | |||
| Compound Name |
3-[[2-(2-Fluorophenyl)pyridin-4-yl]amino]-4-[[(1R)-1-phenylethyl]amino]cyclobut-3-ene-1,2-dione
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL468125; 3-{[2-(2-Fluorophenyl)pyridin-4-yl]amino}-4-{[(1R)-1-phenylethyl]amino}cyclobut-3-ene-1,2-dione; SCHEMBL4371574; BDBM50259601
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[6] | |||
| Compound Name |
3-(4'-Hydroxybiphenyl-4-Yl)-N-(4-Hydroxycyclohexyl)-1,4-Dihydroindeno[1,2-C]pyrazole-6-Carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL438485; SCHEMBL4809259; SCHEMBL4809267; BDBM91830; BDBM50204694; ZINC100469705; ZINC253994709; Q27456666
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[18] | |||
| Compound Name |
N-(4-Methyl-3-(3-methyl-1H-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682012; SCHEMBL3784527; US9796706, Compound 15; BDBM351571; BDBM50338289
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
N-[4-(4-Naphthalen-2-yl-5-oxo-1H-1,2,4-triazol-3-yl)pyridin-2-yl]cyclopropanecarboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644630; BDBM50333984
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
Methyl 5-(2-(isoquinolin-5-yl)acetamido)thiazole-4-carboxylate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288127; SCHEMBL3712075; BDBM50332087; methyl 5-[(2-isoquinolin-5-ylacetyl)amino]-1,3-thiazole-4-carboxylate
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
N-[4-Methyl-3-(1h-1,2,4-Triazol-5-Yl)thiophen-2-Yl]-2-(2-Oxo-3,4-Dihydroquinolin-1(2h)-Yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1614820; n-(4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide; SCHEMBL3783179; US9796706, Compound 14; BDBM351570; BDBM50338290; Q27456956; N-[4-methyl-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1-yl)acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
Tert-Butyl 4-(6-(4-aminophenyl)-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carboxylate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1095627; SCHEMBL3991434; BDBM50316253
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[12] | |||
| Compound Name |
6-Methyl-4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1080995; SCHEMBL2934911; BDBM50311954
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[14] | |||
| Compound Name |
n-(4-Bromo-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(quinolin-5-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682019; SCHEMBL3783257; US9796706, Compound 33; BDBM351589; BDBM50338265; N-[4-bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-quinolin-5-ylacetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
6-Chloro-9-hydroxy-1-methyl-3-(trifluoromethyl)-1H,4H,9H-pyrazolo[3,4-b]quinolin-4-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
Kinome_3393; CHEMBL207400; 9-hydroxy pyrazoloquinolinone 2; BDBM15869
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[15] | |||
| Compound Name |
3-(2-(Cyclopropylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644623; BDBM50333986
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
5-[2-(Cyclohexylamino)pyridin-4-Yl]-4-Naphthalen-2-Yl-2-(Tetrahydro-2h-Pyran-4-Yl)-2,4-Dihydro-3h-1,2,4-Triazol-3-One
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644639; BDBM50334001; Q27455545
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(2-(pyridin-2-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644625; SCHEMBL16573741; BDBM50333982
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
n-(4-Chloro-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682014; SCHEMBL3782279; US9796706, Compound 18; BDBM351574; BDBM50338292; N-[4-chloro-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1-yl)acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
n-(4-Chloro-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(quinolin-5-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682020; SCHEMBL3782088; US9796706, Compound 21; BDBM351577; BDBM50338266; N-[4-chloro-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-quinolin-5-ylacetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
N-[3-(2-Pyridin-4-ylpyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1089082; SCHEMBL4656083; BDBM50314051; N-(3-(2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-3-(trifluoromethyl)benzamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[19] | |||
| Compound Name |
Methyl 3-(2-(isoquinolin-5-yl)acetamido)thiophene-2-carboxylate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288215; BDBM50332050
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1-(tetrahydrofuran-3-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644640; BDBM50333996
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
2-(4-Methoxyphenyl)-N-(2-(2-methyl-1H-imidazol-4-yl)thiophen-3-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288069; SCHEMBL3782262; BDBM50332083; 2-(4-methoxyphenyl)-N-[2-(2-methyl-1H-imidazol-5-yl)thiophen-3-yl]acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
(3R)-N-(3-Chloro-4-hydroxyphenyl)-1-[2-[4-[4-(4-methoxyphenyl)phenyl]piperazin-1-yl]-2-oxoethyl]pyrrolidine-3-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3398595; SCHEMBL10236155; BDBM50063576
Click to Show/Hide
|
||||
| Activity |
IC50 = 50000 nM
|
[20] | |||
| Compound Name |
2-(4-Methoxyphenyl)-N-(2-(pyrazin-2-yl)thiophen-3-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288098; SCHEMBL3713053; BDBM50332084; 2-(4-methoxyphenyl)-N-(2-pyrazin-2-ylthiophen-3-yl)acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
2-(Isoquinolin-5-yl)-N-(2-(thiazol-4-yl)thiophen-3-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288100; SCHEMBL3713199; BDBM50332086; 2-isoquinolin-5-yl-N-[2-(1,3-thiazol-4-yl)thiophen-3-yl]acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
4-(Naphthalen-2-yl)-1-(pyridin-2-ylmethyl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644615; BDBM50334007
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
n-(4-Methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(quinolin-5-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1682011; SCHEMBL3776306; US9796706, Compound 23; BDBM351579; BDBM50338288; N-[4-methyl-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-quinolin-5-ylacetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
4-(Naphthalen-2-yl)-3-(2-(phenylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644624; BDBM50334003
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
4-(6-Fluoronaphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644632; BDBM50333990
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
9-Isopropyl-N*6*-(3-methyl-but-2-enyl)-9H-purine-2,6-diamine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL77155; BDBM50113679
Click to Show/Hide
|
||||
| Activity |
IC50 = 50000 nM
|
[21] | |||
| Compound Name |
Methyl 3-[2-(2-thienyl)acetamido]thiophene-2-carboxylate
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288895; Methyl 3-[(Thiophen-2-Ylacetyl)amino]thiophene-2-Carboxylate; Oprea1_862132; ZINC82427; HMS3745A11; methyl 3-[(2-thiophen-2-ylacetyl)amino]thiophene-2-carboxylate; BDBM50332040; CCG-45435; AKOS001327224; MCULE-1255934042; SR-01000635201-1; Q27162609; methyl3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylate; methyl 3-(2-(thiophen-2-yl)acetamido)thiophene-2-carboxylate
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[2] | |||
| Compound Name |
3-(2-(Cyclopentylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644621; BDBM50333985
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
3-(2-(Cyclobutylamino)pyridin-4-yl)-4-(naphthalen-2-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644622; BDBM50333992
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
2-(4-Methoxyphenyl)-N-(2-(1-methyl-1H-imidazol-4-yl)thiophen-3-yl)acetamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1288067; SCHEMBL3782326; BDBM50332081; 2-(4-methoxyphenyl)-N-[2-(1-methylimidazol-4-yl)thiophen-3-yl]acetamide
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[8] | |||
| Compound Name |
(3R)-1-[2-[4-(4-Acetylphenyl)piperazin-1-yl]-2-oxoethyl]-N-(2-chloro-4-hydroxyphenyl)pyrrolidine-3-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3356125; SCHEMBL13119169; BDBM50030878
Click to Show/Hide
|
||||
| Activity |
IC50 = 50000 nM
|
[22] | |||
| Compound Name |
4-(Naphthalen-2-yl)-1-(pyridin-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1644641; BDBM50333981
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 50000 nM
|
[7] | |||
| Compound Name |
2-Phenyl-5H-pyrrolo[2,3-b]pyrazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3628249; SCHEMBL12605504; BDBM50127021; ZINC584652510
Click to Show/Hide
|
||||
| Activity |
IC50 = 50100 nM
|
[23] | |||
| Compound Name |
(3S)-3-[[6-(Benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2-methylpentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922217; SCHEMBL3876741; BDBM50358242
Click to Show/Hide
|
||||
| Activity |
IC50 = 52000 nM
|
[24] | |||
| Compound Name |
(3RS,4S)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922210; SCHEMBL1376090; BDBM50358236; (4S)-2-methyl-4-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]hexan-3-ol; (3RS, 4S)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 67000 nM
|
[4] | |||
| Compound Name |
2-Pyridin-3-yl-5H-pyrrolo[2,3-b]pyrazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3628360; BDBM50127030
Click to Show/Hide
|
||||
| Activity |
IC50 = 71500 nM
|
[23] | |||
| Compound Name |
(3R)-3-[[9-Propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922114; BDBM50358215
Click to Show/Hide
|
||||
| Activity |
IC50 = 73000 nM
|
[24] | |||
| Compound Name |
Chembl4210146
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
BDBM50456345; ERZ
Click to Show/Hide
|
||||
| Activity |
IC50 = 76000 nM
|
[25] | |||
| Compound Name |
(3S)-3-[[9-Propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922204; BDBM50358230
Click to Show/Hide
|
||||
| Activity |
IC50 = 77000 nM
|
[24] | |||
| Compound Name |
(4S)-4-[[9-Propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922205; SCHEMBL1378854; BDBM50358231; (3RS,4S)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 80000 nM
|
[24] | |||
| Compound Name |
N-(5,6-Dimethoxy-1,3-benzothiazol-2-yl)-2-[(4-fluorophenoxy)methyl]-1,3-thiazole-4-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3752694; BDBM50139004; ZINC13011838; AKOS001458415; MCULE-4851709338; Z296307320
Click to Show/Hide
|
||||
| Activity |
IC50 = 82000 nM
|
[26] | |||
| Compound Name |
(3RS,4S)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2-methyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922215; SCHEMBL4487926; BDBM50358240; (3RS, 4S)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2-methyl-hexan-3-ol; (4S)-4-[[6-(benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2-methylhexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 88000 nM
|
[24] | |||
| Compound Name |
2-(4-Methoxyphenyl)-5H-pyrrolo[2,3-b]pyrazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3628253; BDBM50127025
Click to Show/Hide
|
||||
| Activity |
IC50 = 89700 nM
|
[23] | |||
| Compound Name |
(3R)-3-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922123; SCHEMBL1376524; BDBM50358210; (3R)-2-methyl-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 91000 nM
|
[4] | |||
| Compound Name |
N-(3-Methoxyphenyl)-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3782023
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
3-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-7-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780571
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
(4S,6E)-18-Hydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1668419; BDBM50336461
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[28] | |||
| Compound Name |
N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781159
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-Ethyl-3-[3-[(6-methoxypyridin-3-yl)amino]pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3695655; SCHEMBL14506629; BDBM142697; US8937068, 190
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780515
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
2-(3,4-Dihydroxybenzylidene)benzofuran-3(2H)-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3361128; BDBM50038423; ZINC16052822; (E)-2-(3,4-Dihydroxybenzylidene)benzofuran-3(2H)-one
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[30] | |||
| Compound Name |
1-[3-(4-Chloroanilino)pyrido[2,3-b]pyrazin-6-yl]-3-ethylurea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5477088; CHEMBL3695630; BDBM142671; US8937068, 159
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-Ethyl-3-[3-(4-fluoroanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5449855; CHEMBL3695637; BDBM142678; US8937068, 167
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-Ethyl-3-[3-(naphthalen-2-ylamino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5447745; CHEMBL3695662; BDBM47102; US8937068, 178
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780543
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-4-yl]-3-(2-phenylethyl)urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318035; SCHEMBL1932182; BDBM50050861
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
1-Benzyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-4-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318034; SCHEMBL1932160; BDBM50050860
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
N-(3-Ethynylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780350
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
7-Chloro-1-(3,4-dichlorophenyl)-6-methoxy-3,4-dihydroisoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1087421; BDBM50415616
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[32] | |||
| Compound Name |
1-Ethyl-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780985
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-[3-[(2-Chloropyridin-4-yl)amino]pyrido[2,3-b]pyrazin-6-yl]-3-ethylurea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3695649; SCHEMBL14506638; BDBM142691; US8937068, 184
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-(3-Methoxyphenyl)-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780768
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-[7-(3,4-Dimethoxyphenyl)-1,5-naphthyridin-4-yl]-3-ethylurea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318008; SCHEMBL1933460; BDBM50050855
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
N-Phenyl-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781538
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-Tert-butyl-3-[7-(4-hydroxy-3-methoxyphenyl)-1,5-naphthyridin-4-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318031; SCHEMBL1932385; BDBM50050857
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
2,3-[Ethyliminobis[ethyleneoxyethylene(1H-indole-1,3-diyl)]]maleimide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL103055; SCHEMBL4346022; BDBM50132310
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[33] | |||
| Compound Name |
6-Methoxy-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole-1-carboxylic acid
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL395157; 6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-1-carboxylic acid; 6-METHOXY-1H,2H,3H,4H,9H-PYRIDO[3,4-B]INDOLE-1-CARBOXYLIC ACID; SCHEMBL608164; SCHEMBL12660570; CTK0H2172; DTXSID00397280; BDBM50215483; MFCD00010826; STL525685; AKOS015894383; MCULE-5714246217; ST065834; 952M635; J-011460; Z2216905627; 6-methoxy-1,2,3,4-tetrahydrobeta-carbolinecarboxylic acid; 6-Methoxy-1,2,3,4-tetrahydro-beta-carboline-1-carboxylic acid; 6-methoxy-2,3,4,9-tetrahydro-1h-beta-carboline-1-carboxylic acid; 1H-Pyrido[3,4-b]indole-1-carboxylic acid, 2,3,4,9-tetrahydro-6-methoxy-; 1H-Pyrido[3,4-b]indole-1-carboxylicacid, 2,3,4,9-tetrahydro-6-methoxy-; 6-methoxy-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-2-ium-1-carboxylate; 6-Methoxy-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole-1-carboxylic acid, 97%
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[34] | |||
| Compound Name |
N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781584
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-4-yl]-3-phenylurea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318033; SCHEMBL1934333; BDBM50050859
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
1-Ethyl-3-[3-(4-methoxyanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5452117; CHEMBL3695629; BDBM142670; US8937068, 158
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-Ethyl-3-[3-(3-hydroxy-4-methylanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3695653; SCHEMBL14506635; BDBM142695; US8937068, 188
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
N-Benzyl-N-methyl-4-(phenylsulfamoyl)benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3355482; BDBM50043416; ZINC17334508; AKOS008571954; Z31474376
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[35] | |||
| Compound Name |
N-(2-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781543
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
Meridianin E
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol; CHEMBL296682; SCHEMBL2787193; BDBM10842
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[36] | |||
| Compound Name |
1-Ethyl-3-[3-(pyridin-3-ylamino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5458507; CHEMBL3695631; BDBM142672; US8937068, 161
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-Ethyl-3-[3-(4-ethylanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5456518; CHEMBL3695632; BDBM142673; US8937068, 162
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
1-Tert-butyl-3-[7-(3,4-dimethoxyphenyl)-1,5-naphthyridin-4-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3318009; SCHEMBL1933604; BDBM50050856
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[31] | |||
| Compound Name |
1-Ethyl-3-[3-(3-methylanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL5458922; CHEMBL3695658; BDBM47097; US8937068, 157
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
(3S,5E)-1-Methyl-3-(pyridin-2-ylmethyl)-5-(pyridin-2-ylmethylidene)piperidin-4-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2338335; BDBM50431025
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[37] | |||
| Compound Name |
(3R)-N-(3-Chloro-4-hydroxyphenyl)-1-[2-[4-[4-(4-fluorophenyl)phenyl]piperazin-1-yl]-2-oxoethyl]pyrrolidine-3-carboxamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3398592; SCHEMBL13118946; BDBM50063533
Click to Show/Hide
|
||||
| Activity |
IC50 = 100000 nM
|
[20] | |||
| Compound Name |
N-(3-Chloro-4-fluorophenyl)-3-phenylpyrido[3,4-b]pyrazin-8-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780151
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
(4S,6E,12E)-18-Hydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1668418; BDBM50336459
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[28] | |||
| Compound Name |
(3R,5E)-1-Methyl-3-(pyridin-2-ylmethyl)-5-(pyridin-2-ylmethylidene)piperidin-4-one
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2338334; BDBM50431026
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[37] | |||
| Compound Name |
7-Chloro-1-(3-chlorophenyl)-6-methoxy-3,4-dihydroisoquinoline
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1088633; BDBM50415620
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[32] | |||
| Compound Name |
N-(4-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3781566
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
Chembl4276946
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
GTPL9965; compound 3a [Pipionne et al, 2018]; 1-[5-amino-4-(3,4-dichlorophenyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-one
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[38] | |||
| Compound Name |
2-(4-Methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-amine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3780637
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[27] | |||
| Compound Name |
3-[6-(Ethylcarbamoylamino)pyrido[2,3-b]pyrazin-3-yl]benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
SCHEMBL4684786; CHEMBL3695628; BDBM142668; US8937068, 155
Click to Show/Hide
|
||||
| Activity |
IC50 ~ 100000 nM
|
[29] | |||
| Compound Name |
(3RS,4R)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922200; SCHEMBL4490773; BDBM50358226; (3RS, 4R)4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-hexan-3-ol; (4R)-4-[[6-(benzylamino)-9-propan-2-ylpurin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 103000 nM
|
[24] | |||
| Compound Name |
(4S)-2,2-Dimethyl-4-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922207; SCHEMBL1381128; BDBM50358233; (3RS,4S)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 137000 nM
|
[24] | |||
| Compound Name |
(R)-3-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2-methyl-pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922203; SCHEMBL4488751; BDBM50358229; (3R)-3-[[6-(benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2-methylpentan-2-ol
Click to Show/Hide
|
||||
| Activity |
IC50 = 149000 nM
|
[24] | |||
| Click to Show/Hide the Information of All Poor Binders | |||||
| Non Binders of This Target (in total, 15 non binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
(3R)-3-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922118; SCHEMBL4496436; BDBM50358219; (3R)-2-methyl-3-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]pentan-2-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
2-Bromo-5H-pyrrolo[2,3-b]pyrazine
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
5-BROMO-4,7-DIAZAINDOLE; 2-bromo-5H-pyrrolo[3,2-b]pyrazine; CHEMBL3628247; MFCD09834822; 5H-Pyrrolo[2,3-b]pyrazine, 2-bromo-; PubChem16377; PubChem20664; SCHEMBL421369; CTK3E8037; DTXSID50648618; 5-methyl-3-pyridine-1H-pyrazole; BCP27240; KS-000002TO; ANW-51807; BDBM50127013; CB0143; MFCD22989332; SC1651; ZINC21303791; AKOS006326434; AKOS028109150; ACN-025231; CM14228; CS-W008866; FS-3280; 2-bromanyl-5H-pyrrolo[2,3-b]pyrazine; AC-23734; AK-23813; BC004105; BP-30046; BR-23813; QC-10946; SC-45298; SY007444; AB0009963; DB-023135; AM20070392; FT-0648057; C-2047; 781B434; A842277; J-517067; W-205236
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[23] | |||
| Compound Name |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2,2-dimethyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922117; SCHEMBL1380702; BDBM50358218; (4R)-2,2-dimethyl-4-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
(3S)-2-Methyl-3-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]pentan-2-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1921805; SCHEMBL1378506; BDBM50358234; (3S)-3-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-pentan-2-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
3-(5H-Pyrrolo[2,3-b]pyrazin-2-yl)benzamide
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3628250; BDBM50127022
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[23] | |||
| Compound Name |
(4S)-2-Methyl-4-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922206; SCHEMBL1381821; BDBM50358232; (3RS,4S)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
3-(5H-Pyrrolo[2,3-b]pyrazin-2-yl)phenol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL3628251; BDBM50127023
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[23] | |||
| Compound Name |
(3RS,4R)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2,2-dimethyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922202; SCHEMBL4489114; BDBM50358228; (3RS, 4R)-4(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2,2-dimethyl-hexan-3-ol; (4R)-4-[[6-(benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2,2-dimethylhexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922116; SCHEMBL1380041; BDBM50358217; (4R)-2-methyl-4-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
(3RS,4S)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2,2-dimethyl-hexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922216; SCHEMBL4488384; BDBM50358241; (3RS, 4S)-4-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-2,2-dimethyl-hexan-3-ol; (4S)-4-[[6-(benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2,2-dimethylhexan-3-ol
Click to Show/Hide
|
||||
| Activity |
IC50 > 200000 nM
|
[24] | |||
| Compound Name |
(4R)-4-[[6-(Benzylamino)-9-propan-2-ylpurin-2-yl]amino]-2-methylhexan-3-ol
Click to Show/Hide
|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922201; SCHEMBL4484946; BDBM50358227
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| Activity |
IC50 > 200000 nM
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[24] | |||
| Compound Name |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-2-ylmethyl)-amino]-9H-purin-2-ylamino}-hexan-3-ol
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL1922115; SCHEMBL1381885; BDBM50358216; (4R)-4-[[9-propan-2-yl-6-(pyridin-2-ylmethylamino)purin-2-yl]amino]hexan-3-ol
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| Activity |
IC50 = 230000 nM
|
[24] | |||
| Compound Name |
(4R)-5-(1H-Benzimidazol-2-ylmethyl)-4-(5-methyl-1H-imidazol-4-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2297161; BDBM50489125
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| Activity |
Ki = 1000000 nM
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[39] | |||
| Compound Name |
2-[[(8-Methylimidazo[1,2-a]pyridin-2-yl)methyl-propan-2-ylamino]methyl]-3H-quinazolin-4-one
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL2297163; BDBM50489128
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| Activity |
Ki = 1000000 nM
|
[39] | |||
| Compound Name |
(4S)-5-(1H-Benzimidazol-2-ylmethyl)-4-(5-methyl-1H-imidazol-4-yl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL2297162; BDBM50489131
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| Activity |
Ki = 1000000 nM
|
[39] | |||
| Click to Show/Hide the Information of All Non Binders | |||||
| References | Top | ||||
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