Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T58496 | Target Info | |||
| Target Name | Transient receptor potential cation channel V3 (TRPV3) | ||||
| Synonyms |
Vanilloid receptor-like 3; VRL-3; TrpV3
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| Target Type | Clinical trial Target | ||||
| Gene Name | TRPV3 | ||||
| Biochemical Class | Transient receptor potential catioin channel | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 1 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
(R)-8-{5-[3-Methyl-4-(trifluoromethyl)phenyl]oxazol-2-ylamino}-1,2,3,4-tetrahydronaphthalen-2-ol
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL1173240; SCHEMBL472366; BDBM50321851; US8796328, D
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| Activity |
IC50 ~ 100000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Synthesis and biological evaluation of 5-substituted and 4,5-disubstituted-2-arylamino oxazole TRPV1 antagonists. Bioorg Med Chem. 2010 Jul 1;18(13):4821-9. | ||||
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