Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T32821 | Target Info | |||
| Target Name | Lysophosphatidic acid acyltransferase beta (LPAATB) | ||||
| Synonyms |
Lysophosphatidic acid acyltransferase-beta; LPAAT-beta; AGPAT2; 1-acylglycerol-3-phosphate O-acyltransferase 2; 1-AGPAT 2; 1-AGP acyltransferase 2
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| Target Type | Literature-reported Target | ||||
| Gene Name | AGPAT2 | ||||
| Biochemical Class | Acyltransferase | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 5 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
[4-Chloro-3-(6-methyl-benzothiazol-2-yl)-phenyl]-carbamic acid methyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL35964; BDBM50141299
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| Activity |
IC50 ~ 64000 nM
|
[1] | |||
| Compound Name |
[4-Chloro-3-(5-phenyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL36197; BDBM50141264
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| Activity |
IC50 = 64000 nM
|
[1] | |||
| Compound Name |
[4-Methoxy-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL35211; BDBM50141267
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| Activity |
IC50 = 64000 nM
|
[1] | |||
| Compound Name |
[4-Fluoro-3-(5-methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester
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Investigative | Compound Info | ||
| Synonyms |
CHEMBL35254; BDBM50141286
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| Activity |
IC50 ~ 64000 nM
|
[1] | |||
| Compound Name |
[3-(5-Methyl-benzooxazol-2-yl)-phenyl]-carbamic acid methyl ester
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL35255; BDBM50141253
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| Activity |
IC50 ~ 64000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Synthesis and SAR of 2-arylbenzoxazoles, benzothiazoles and benzimidazoles as inhibitors of lysophosphatidic acid acyltransferase-beta. Bioorg Med Chem Lett. 2004 Mar 22;14(6):1455-9. | ||||
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