Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T15848 | Target Info | |||
| Target Name | Tyrosine-protein kinase Tec (PSCTK4) | ||||
| Synonyms |
Tec protein tyrosine kinase
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| Target Type | Patented-recorded Target | ||||
| Gene Name | TEC | ||||
| Biochemical Class | Kinase | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 1 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
Staurosporine
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Phase 2 | Compound Info | ||
| Synonyms |
staurosporine; Staurosporin; (+)-Staurosporine; Antibiotic 230; 62996-74-1; Antibiotic AM 2282; CCRIS 3272; AM-2282; UNII-H88EPA0A3N; Alkaloid AM-2282 from Streptomyces; H88EPA0A3N; CHEMBL388978; CHEBI:15738; CGP 39360; 8,12-Epoxy-1H,8H-2,7b,12a-triazadibenzo(a,g)cyclonona(cde)trinden-1-one, 2,3,9,10,11,12-hexahydro-9-methoxy-8-methyl-10-(methylamino)-, (8alpha,9beta,10beta,12alpha)-(+)-
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| Activity |
IC50 = 128000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Discovery and optimization of selective FGFR4 inhibitors via scaffold hopping. Bioorg Med Chem Lett. 2017 Jun 1;27(11):2420-2423. | ||||
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