Target Poor or Non Binder(s) Information
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T00099 | Target Info | |||
| Target Name | HUMAN calpain-1/calpain small subunit 1 heterodimer (CAPN1/CAPNS1) | ||||
| Synonyms |
Calpain-1 large subunit/calpain small subunit 1 dimer
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| Biochemical Class | Peptidase C2 family | ||||
| UniProt ID | |||||
| Poor Binders of This Target (in total, 1 binders) | Download | Top | |||
|---|---|---|---|---|---|
| Compound Name |
[1-(1-Benzyl-2-diethylcarbamoyl-2-oxo-ethylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl ester
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|
Investigative | Compound Info | ||
| Synonyms |
CHEMBL117089; BDBM50042431
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| Activity |
Ki = 76000 nM
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[1] | |||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases. J Med Chem. 1993 Oct 29;36(22):3472-80. | ||||
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