Target and Its Patented Drug(s)
| Target General Information | Top | ||||
|---|---|---|---|---|---|
| Target ID | T03279 | Target Info | |||
| Target Name | Ribosomal protein S6 kinase alpha-3 (RSK3) | ||||
| Synonyms | pp90RSK2; p90RSK3; p90-RSK 3; S6K-alpha-3; Ribosomal S6 kinase 2; RSK2; RSK-2; MAPKAPK1B; MAPKAPK-1b; MAPKAP kinase 1b; MAPK-activated protein kinase 1b; MAP kinase-activated protein kinase 1b; Insulin-stimulated protein kinase 1; ISPK1; ISPK-1; 90 kDa ribosomal protein S6 kinase 3 | ||||
| Target Type | Patented-recorded Target | ||||
| Gene Name | RPS6KA3 | ||||
| Biochemical Class | Kinase | ||||
| UniProt ID | |||||
| Patent(s) and the Corresponding Patented Drug(s) | Top | ||||
|---|---|---|---|---|---|
| United States Patent and Trademark Office (USPTO) | |||||
| Patent ID | US9150577 | ||||
| Title | Heterocyclic Compounds Containing An Indole Core. | ||||
| Representative Drug(s) | D01IOH | Drug Info | IC50 = 600 to 7700 nM | [1] | |
| Patent ID | US7687506 | ||||
| Title | Selective Serine/Threonine Kinase Inhibitors. | ||||
| Representative Drug(s) | D0X8YV | Drug Info | N.A. | [1] | |
| Patent ID | US8765802 | ||||
| Title | Kinase Inhibitors, Compositions Thereof, and Methods of Use Therewith. | ||||
| Representative Drug(s) | D0O6TG | Drug Info | IC50 < 1000 nM | [1] | |
| Patent ID | US7605241 | ||||
| Title | Synthesis of Inhibitors of P90Rsk. | ||||
| References | Top | ||||
|---|---|---|---|---|---|
| REF 1 | Ribosomal S6 kinase (RSK) modulators: a patent review.Expert Opin Ther Pat. 2016 Sep;26(9):1061-78. | ||||
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