Co-Target(s) Information
Target General Information | Top | ||||
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Target ID | T59604 | Target Info | |||
Target Name | Growth hormone secretagogue receptor 1 (GHSR) | ||||
Synonyms |
Growth hormone secretagogue receptor; Ghrelin receptor; GHSR; GHS-R; GHRP; GH-releasing peptide receptor
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Target Type | Successful Target | ||||
Gene Name | GHSR | ||||
Biochemical Class | GPCR rhodopsin | ||||
UniProt ID |
Co-Targets of This Target | Top | |||||
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Co-Target Name | Ghrelin (GHRL) | Clinical trial Target | ||||
UniProt ID | GHRL_HUMAN | |||||
Gene Name | GHRL | |||||
Synonyms |
UNQ524/PRO1066; Motilin-related peptide; M46 protein; Growth hormone secretagogue; Growth hormone releasing peptide; Gastric peptide ghrelin; GHRL
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Representative Drug(s) | TZP-101 | Drug Info | Ki = 16 nM | [1] |
References | Top | ||||
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REF 1 | Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): Development of ulimorelin (TZP-101) from hit to clinic. J Med Chem. 2011 Dec 22;54(24):8305-20. |
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