Target Validation Information
Target ID T40016
Target Name Glucocorticoid receptor
Target Type
Successful
Drug Potency against Target GW685698X Drug Info IC50 = 69000 nM [552644]
ZK-230211 Drug Info IC50 = 16 nM [525950]
References
Ref 552644Structure-activity relationships of selective GABA uptake inhibitors. Curr Top Med Chem. 2006;6(17):1861-82.
Ref 525950J Med Chem. 2000 Dec 28;43(26):5010-6.Synthesis and biological activity of a novel, highly potent progesterone receptor antagonist.

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