TTD_Target_ID	Target_Name	TTD_Drug_ID	Drug_Name	Drug_Highest_Status	Drug_PubchemID	Molecular_Formula	Molecular_Weight	Canonical_SMILES	Activity	Binder_Type
T72849	Adipocyte-derived leucine aminopeptidase	B0U5EM	2-[[[1-Amino-3-(3-hydroxyphenyl)propyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid	Investigative	118720631	C19H24NO5P	377.4	C1=CC=C(C=C1)CC(CP(=O)(C(CCC2=CC(=CC=C2)O)N)O)C(=O)O	Ki = 87100 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B1G5XA	Methyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate	Investigative	118734258	C23H30N4O5	442.5	CCCC[C@@H](C(=O)NC1=C(C=CC(=C1)C(=O)N[C@@H](CC2=CC=C(C=C2)O)C(=O)OC)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B4ZMH0	[(2R)-2-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid	Investigative	137653412	C35H40N3O4P	597.7	C1=CC=C(C=C1)CC[C@H](N)P(=O)(C[C@H](CC(C2=CC=CC=C2)C3=CC=CC=C3)C(=O)N[C@@H](CC4=CC=CC=C4)C(=O)N)O	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B6OB2T	(2S)-2-[(3,4-Diaminobenzoyl)amino]-3-(1H-indol-3-yl)propanoic acid	Investigative	118734273	C18H18N4O3	338.4	C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)O)NC(=O)C3=CC(=C(C=C3)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B86GZE	Methyl 4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoate	Investigative	118734163	C18H21N3O4	343.4	COC(=O)C1=CC(=C(C=C1)N)NC(=O)[C@H](CCC2=CC=C(C=C2)O)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B8PD3N	Methyl (2S)-6-amino-2-[(3,4-diaminobenzoyl)amino]hexanoate	Investigative	118734270	C14H22N4O3	294.35	COC(=O)[C@H](CCCCN)NC(=O)C1=CC(=C(C=C1)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B8R6FT	Methyl 3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoate	Investigative	118734265	C18H21N3O3	327.4	COC(=O)C1=CC(=C(C=C1)NC(=O)[C@H](CCC2=CC=CC=C2)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	B9NI8O	Methyl 4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoate	Investigative	118734165	C14H21N3O3	279.33	CCCC[C@@H](C(=O)NC1=C(C=CC(=C1)C(=O)OC)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BIC47U	Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoate	Investigative	118734254	C42H41N5O5	695.8	C1=CC=C(C=C1)COC2=CC=C(C=C2)CC[C@@H](C(=O)NC3=C(C=CC(=C3)C(=O)N[C@@H](CC4=CNC5=CC=CC=C54)C(=O)OCC6=CC=CC=C6)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BKL9P8	Methyl (2S)-6-amino-2-[[3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]hexanoate	Investigative	118734285	C23H31N5O5	457.5	COC(=O)[C@H](CCCCN)NC(=O)C1=CC(=C(C=C1)NC(=O)[C@H](CC2=CC=C(C=C2)O)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BLC0O3	Methyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate	Investigative	118734292	C23H30N4O5	442.5	CCCC[C@@H](C(=O)NC1=C(C=C(C=C1)C(=O)N[C@@H](CC2=CC=C(C=C2)O)C(=O)OC)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BM6AW9	[(2R)-3-[[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[(3,5-diphenylphenyl)methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid	Investigative	137640549	C40H42N3O4P	659.8	C1=CC=C(C=C1)CC[C@H](N)P(=O)(C[C@H](CC2=CC(=CC(=C2)C3=CC=CC=C3)C4=CC=CC=C4)C(=O)N[C@@H](CC5=CC=CC=C5)C(=O)N)O	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BPKL71	Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-methylbutanoate	Investigative	71817806	C29H34N4O4	502.6	CC(C)[C@@H](C(=O)OCC1=CC=CC=C1)NC(=O)C2=CC(=C(C=C2)N)NC(=O)[C@H](CCC3=CC=CC=C3)N	IC50 = 95500 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BT4CF0	Methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate	Investigative	118734181	C26H28N4O6	492.5	COC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)C2=CC(=C(C=C2)N)NC(=O)[C@H](CC3=CC=C(C=C3)O)N	IC50 = 110000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BU2OB6	Methyl (2S,3R)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-hydroxybutanoate	Investigative	118734182	C21H26N4O6	430.5	C[C@H]([C@@H](C(=O)OC)NC(=O)C1=CC(=C(C=C1)N)NC(=O)[C@H](CC2=CC=C(C=C2)O)N)O	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BU45WQ	Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]hexanoate	Investigative	118734173	C31H39N5O5	561.7	COC(=O)[C@H](CCCCN)NC(=O)C1=CC(=C(C=C1)N)NC(=O)[C@H](CCC2=CC=C(C=C2)OCC3=CC=CC=C3)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BW5I7M	Benzyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoate	Investigative	118734290	C25H34N4O4	454.6	CCCC[C@@H](C(=O)NC1=C(C=C(C=C1)C(=O)N[C@@H](C(C)C)C(=O)OCC2=CC=CC=C2)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BX6BP8	Benzyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoate	Investigative	118734256	C25H34N4O4	454.6	CCCC[C@@H](C(=O)NC1=C(C=CC(=C1)C(=O)N[C@@H](C(C)C)C(=O)OCC2=CC=CC=C2)N)N	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BY1ZC6	4-Amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoic acid	Investigative	118734161	C16H17N3O4	315.32	C1=CC(=CC=C1C[C@@H](C(=O)NC2=C(C=CC(=C2)C(=O)O)N)N)O	IC50 ~ 100000 nM	Poor binder
T72849	Adipocyte-derived leucine aminopeptidase	BZ74KI	Methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]hexanoate	Investigative	118734172	C24H33N5O5	471.5	COC(=O)[C@H](CCCCN)NC(=O)C1=CC(=C(C=C1)N)NC(=O)[C@H](CCC2=CC=C(C=C2)O)N	IC50 ~ 100000 nM	Poor binder