TTD_Target_ID Target_Name TTD_Drug_ID Drug_Name Drug_Highest_Status Drug_PubchemID Molecular_Formula Molecular_Weight Canonical_SMILES Activity Binder_Type T27466 Bromodomain and PHD finger containing 3 B2ISO1 4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamide Investigative 137636309 C20H19N3O3S 381.4 CCC1=CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=C(C=C3)C#N)N(C1=O)CC IC50 ~ 100000 nM Poor binder T27466 Bromodomain and PHD finger containing 3 B9C1SD 1-Methyl-2-oxo-N-phenylquinoline-6-sulfonamide Investigative 137639742 C16H14N2O3S 314.4 CN1C2=C(C=CC1=O)C=C(C=C2)S(=O)(=O)NC3=CC=CC=C3 IC50 ~ 100000 nM Poor binder T27466 Bromodomain and PHD finger containing 3 D03BTJ PMID25408830C3 Investigative 15990224 C22H26N4O3 394.5 CN1C2=C(C=C(C(=C2)NC(=O)C3=CC=CC=C3OC)N4CCCCC4)N(C1=O)C IC50 ~ 100000 nM Poor binder