Multi-target agents
Target Pair | Drug Name | |
---|---|---|
CAI --- CAIX | 2-cyclohexylamido-5-sulfonamidoindane | Drug Info |
Aurora --- VEGFR | 7-(1H-indol-2-yl)isoindolin-1-one | Drug Info |
AuroraA --- STK1 | (Z)-N-(3-{[3-(3-Morpholino-3-oxopropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-2-yl]methylene}-2-oxoindolin-5-yl)benzenesulfonamide | Drug Info |
AuroraA --- STK1 | (R)-N-(5-(2-fluoro-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-4-(4-methylpiperazin-1-yl)benzamide | Drug Info |
AuroraA --- STK1 | 6-Methyl-3-(1H-pyrazol-4-yl)-N-[3-[(3,3,4,4-tetrafluoro-1-pyrrolidinyl)methyl]-5-isothiazolyl]imidazo[1,2-a]pyrazin-8-amine Hydrochloride | Drug Info |
AuroraA --- STK1 | 3-methyl-N-(6-(morpholinomethyl)-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)isothiazol-5-amine | Drug Info |
AuroraA --- STK1 | N-(4-(4-(5-methyl-1H-pyrazol-3-ylamino)-6-(piperidin-1-yl)pyrimidin-2-ylthio)phenyl)propionamide | Drug Info |
AuroraA --- STK1 | 4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine | Drug Info |
AuroraA --- STK1 | (R)-1-(2-amino-6-(3-amino-1H-indazol-6-yl)pyrimidin-4-yl)-N-phenylpiperidine-3-carboxamide | Drug Info |
AuroraA --- STK1 | N-(3-fluorophenyl)-2-(3-(7-(3-((2-hydroxyethyl)(propyl)amino)propoxy)-6-methoxyquinazolin-4-ylamino)-1H-pyrazol-5-yl)acetamide | Drug Info |
B1R --- B2R | H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH (JMV1639) | Drug Info |
Beta PDGFR --- CABL | (E)-4-(3-(hydroxyamino)-3-oxoprop-1-enyl)-N-(4-methyl-3-(4-(pyridin-3-yl)thiazol-2-ylamino)phenyl)benzamide | Drug Info |
BNOS --- Hepatocyte NOS | 7,8-Difluoro-4-((2-(4-methylthiazol-5-yl)-1H-benzo[d]imidazol-1-yl)methyl)quinolin-2(1H)-one | Drug Info |
BNOS --- Hepatocyte NOS | 4-Isopropyl-pyrrolidin-(2Z)-ylideneamine | Drug Info |
BNOS --- Hepatocyte NOS | Azepan-(2Z)-ylideneamine | Drug Info |
BNOS --- Hepatocyte NOS | N-(4-Carbamimidoylsulfanylmethyl-phenyl)-acetamidine | Drug Info |
BNOS --- Hepatocyte NOS | (R)-N-(1-(2-(3-Hydroxypyrrolidin-1-yl)ethyl)indolin-6-yl)-thiophene-2-carboximidamide | Drug Info |
BNOS --- Hepatocyte NOS | SID11111542 | Drug Info |
BNOS --- Hepatocyte NOS | 4-ethylpyridin-2-amine | Drug Info |
BNOS --- Hepatocyte NOS | 3-Methyl-pyrrolidin-(2Z)-ylideneamine | Drug Info |
BNOS --- Hepatocyte NOS | (3aR,9bS)-8-chloro-2,3,3a,9b-tetrahydro-1H-cyclopenta[c]quinolin-4-amine | Drug Info |
BNOS --- Hepatocyte NOS | 4-Trifluoromethyl-piperidin-(2Z)-ylideneamine | Drug Info |
Pagination
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